CC(C)Cn1cc(CNS(=O)(=O)C2CC2)c2ccc(-c3ccccc3C(F)(F)F)cc21 CHEMBL5434615 EC50 6.0 nM
CC(C)Cn1cc(C(C)NS(=O)(=O)C2CC2)c2ccc(-c3ccccc3C(F)(F)F)cc21 CHEMBL5408866 EC50 7.0 nM
CC(C)Cc1cn(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccncc3)cc12 CHEMBL5419854 EC50 10.0 nM
CC(C)Cc1cn(CCNS(=O)(=O)N(C)C)c2ncc(-c3ccncc3)cc12 CHEMBL5417493 EC50 20.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccncc3)cc21 CHEMBL5424373 EC50 20.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)C2CC2)c2ccc(-c3ccncc3)cc21 CHEMBL5407367 EC50 25.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)C2CC2)c2ccc(-c3ccccc3C(F)(F)F)cc21 CHEMBL5404180 EC50 40.0 nM
Cc1cc(Cl)ccc1CN(Cc1ccc(Cl)cc1)Cc1ccc([N+](=O)[O-])s1 CHEMBL2381196 EC50 50.0 nM
Cc1cc(Cl)cc(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)c1 CHEMBL4761268 EC50 50.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccccc3Cl)cc21 CHEMBL5436011 EC50 50.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)C(C)C)c2ccc(-c3ccncc3)cc21 CHEMBL5424215 EC50 54.0 nM
O=[N+]([O-])c1ccc(CN(Cc2ccc(Cl)cc2)Cc2ccccc2F)s1 CHEMBL2381198 EC50 63.0 nM
CC(C)(C)Oc1ccc(OC[C@@H]2Cc3cc(F)ccc3CN2C(=O)c2cccc3ccccc23)cc1 CHEMBL4781178 EC50 68.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccccc3)cc21 CHEMBL5439268 EC50 70.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccccc3C(F)(F)F)cc21 CHEMBL5412941 EC50 70.0 nM
CCCOc1ccc(OCC2Cc3ccccc3CN2C(=O)c2cccc3ccccc23)cc1 CHEMBL2030074 EC50 77.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(C3CC3)cc21 CHEMBL5434147 EC50 80.0 nM
CCOc1ccc(OCC2Cc3ccccc3CN2C(=O)c2cccc3ccccc23)cc1 CHEMBL2030073 EC50 97.0 nM
O=[N+]([O-])c1ccc(CN(Cc2ccccc2)Cc2ccc(Cl)cc2)s1 CHEMBL2381197 EC50 100.0 nM
CC(C)Cn1cc(C(NS(=O)(=O)C2CC2)C(F)(F)F)c2ccc(-c3ccccc3C(F)(F)F)cc21 CHEMBL5432192 EC50 110.0 nM
COc1ccc(OCC2Cc3ccccc3CN2C(=O)c2cccc3ccccc23)cc1 CHEMBL2030072 EC50 120.0 nM
O=C(c1cccc2ccccc12)N1Cc2ccccc2CC1COc1ccc(-n2cncn2)cc1 CHEMBL2030077 EC50 120.0 nM
Cc1ccc2c(CCNS(=O)(=O)N(C)C)cn(CC(C)C)c2c1 CHEMBL5435001 EC50 120.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N2CCCC2)c2ccc(-c3ccncc3)cc21 CHEMBL5438917 EC50 123.0 nM
CC(C)(C)Oc1ccc(OCC2Cc3ccccc3CN2C(=O)c2cccc3ccccc23)cc1 CHEMBL2030075 EC50 140.0 nM
COCCNc1oc(-c2ccc(N(C)Cc3ccc(Cl)cc3)cc2)nc1C#N CHEMBL4763333 EC50 150.0 nM
O=[N+]([O-])c1ccc(CN(Cc2ccc(F)cc2)Cc2cccnc2)s1 CHEMBL2381202 EC50 160.0 nM
Cc1ccc(CN(Cc2cccnc2)Cc2ccc([N+](=O)[O-])s2)cc1 CHEMBL2381201 EC50 160.0 nM
O=[N+]([O-])c1ccc(CN(Cc2ccc(Cl)cc2)Cc2cccnc2)s1 CHEMBL2381200 EC50 160.0 nM
CC(C)CCN(Cc1ccc(Cl)cc1)Cc1ccc([N+](=O)[O-])s1 CHEMBL2381199 EC50 160.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3cccnc3)cc21 CHEMBL5429567 EC50 160.0 nM
N#Cc1ccc(CN(Cc2cccnc2)Cc2ccc(F)c(F)c2)s1 CHEMBL2381193 EC50 200.0 nM
N#Cc1ccc(CN(Cc2ccc(F)cc2)Cc2cccnc2)s1 CHEMBL2381214 EC50 200.0 nM
N#Cc1ccc(CN(Cc2ccc(Cl)cc2)Cc2cccnc2)s1 CHEMBL2381208 EC50 200.0 nM
COc1ccc(CN(Cc2cccnc2)Cc2ccc([N+](=O)[O-])s2)cc1 CHEMBL2381205 EC50 200.0 nM
Cc1cccc(CN(Cc2cccnc2)Cc2ccc([N+](=O)[O-])s2)c1 CHEMBL2381204 EC50 200.0 nM
Cc1ccccc1CN(Cc1cccnc1)Cc1ccc([N+](=O)[O-])s1 CHEMBL2381203 EC50 200.0 nM
Cc1sc(CN(Cc2ccc(Cl)cc2)Cc2cccnc2)cc1Br CHEMBL2381209 EC50 250.0 nM
COc1ccc(OCC2Cc3ccccc3CN2C(=O)c2cccc3ccccc23)cc1OC CHEMBL2030081 EC50 330.0 nM
COc1ccccc1-c1ccc2c(CCNS(=O)(=O)N(C)C)cn(CC(C)C)c2c1 CHEMBL5435835 EC50 330.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3cccc(C#N)c3)cc21 CHEMBL5396141 EC50 370.0 nM
CC(C)Cn1cc(C(C)(C)NS(=O)(=O)C2CC2)c2ccc(-c3ccccc3C(F)(F)F)cc21 CHEMBL5432560 EC50 390.0 nM
CC(C)(C)OC(=O)CN(Cc1ccc(Cl)cc1)Cc1ccc([N+](=O)[O-])s1 CHEMBL1961795 EC50 400.0 nM
O=C(Nc1ccc([N+](=O)[O-])cc1)N1CCC(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)C1 CHEMBL2059696 EC50 400.0 nM
Clc1ccc(CN(Cc2cccnc2)Cc2cc3ccccc3s2)cc1 CHEMBL2381210 EC50 400.0 nM
O=[N+]([O-])c1ccc(CN(Cc2cccnc2)Cc2cccc(C(F)(F)F)c2)s1 CHEMBL2381207 EC50 400.0 nM
COc1cccc(CN(Cc2cccnc2)Cc2ccc([N+](=O)[O-])s2)c1 CHEMBL2381206 EC50 400.0 nM
O=[N+]([O-])c1ccc(CN(Cc2ccc(Cl)cc2)CC2CCN(S(=O)(=O)c3cccc4ccccc34)C2)s1 CHEMBL2059700 EC50 450.0 nM
CCOC(=O)C1Cc2ccccc2CN1C(=O)c1ccc(SC)s1 CHEMBL4754504 EC50 470.0 nM
Cn1nc(Oc2cc(C(F)(F)F)ccc2-c2ccsc2Cl)c2sccc2c1=O CHEMBL4795406 EC50 520.0 nM
CS(=O)(=O)N1CCC(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)C1 CHEMBL2059697 EC50 570.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccccc3O)cc21 CHEMBL5418070 EC50 580.0 nM
O=C(c1cccc2ccccc12)N1Cc2ccccc2CC1COc1ccc(OC(F)(F)F)cc1 CHEMBL2030076 EC50 600.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3cccc(F)c3)cc21 CHEMBL5401858 EC50 610.0 nM
CCCCCNC(=O)N1CCC(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)C1 CHEMBL1961797 IC50 620.0 nM
COc1cccc(OCC2Cc3ccccc3CN2C(=O)c2cccc3ccccc23)c1 CHEMBL2030079 EC50 620.0 nM
O=C(Nc1ccccc1)N1CCC(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)C1 CHEMBL2059573 EC50 620.0 nM
CCOC(=O)N1CCC(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)C1 CHEMBL1961796 EC50 620.0 nM
O=[N+]([O-])c1ccc(CN(Cc2ccc(Cl)cc2)CC2CCN(S(=O)(=O)Cc3ccccc3)C2)s1 CHEMBL2059699 EC50 630.0 nM
N#Cc1ccc(CN(Cc2cccnc2)Cc2cc(F)ccc2F)s1 CHEMBL2381194 EC50 630.0 nM
COc1ccc(CN(Cc2cccnc2)Cc2ccc(C#N)s2)cc1 CHEMBL2380321 EC50 630.0 nM
Clc1ccc(CN(Cc2cccnc2)Cc2sccc2-n2cccc2)cc1 CHEMBL2381211 EC50 630.0 nM
O=C(c1cccc2ccccc12)N1Cc2ccccc2CC1COCc1ccccc1 CHEMBL2030064 EC50 650.0 nM
O=C(c1cccc2ccccc12)N1Cc2ccccc2CC1COc1ccc(-c2ccccc2)cc1 CHEMBL2030071 EC50 650.0 nM
C=CCOC(=O)N1CCC(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)C1 CHEMBL2059572 EC50 670.0 nM
CCCCNC(=O)N1CCC(CN(Cc2ccc(Cl)cc2)Cc2ccc([N+](=O)[O-])s2)C1 CHEMBL2059574 EC50 670.0 nM
O=C(c1cccc2ccccc12)N1Cc2ccccc2CC1COc1ccc(F)cc1F CHEMBL2030082 EC50 710.0 nM
CN(C)c1cccc(OCC2Cc3ccccc3CN2C(=O)c2cccc3ccccc23)c1 CHEMBL2030080 EC50 780.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccc(F)cc3)cc21 CHEMBL5407293 EC50 790.0 nM
O=C(c1cccc2ccccc12)N1Cc2ccccc2CC1COc1ccc(F)cc1 CHEMBL2030070 EC50 800.0 nM
CC(C)(C)OC(=O)CN(Cc1ccc([N+](=O)[O-])s1)S(=O)(=O)c1cccc2ccccc12 CHEMBL2059549 EC50 800.0 nM
O=C(c1cccc2ccccc12)N1Cc2ccccc2CC1COc1ccccc1 CHEMBL2029898 EC50 840.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccc(OC(F)(F)F)cc3)cc21 CHEMBL5425667 EC50 890.0 nM
COc1cccc(-c2ccc3c(CCNS(=O)(=O)N(C)C)cn(CC(C)C)c3c2)c1 CHEMBL5434847 EC50 930.0 nM
Cc1cccc(-c2ccc3c(CCNS(=O)(=O)N(C)C)cn(CC(C)C)c3c2)c1 CHEMBL5396987 EC50 950.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccccc21 CHEMBL5440000 EC50 990.0 nM
CC(C)Cn1cc(CCNS(=O)(=O)N(C)C)c2ccc(-c3ccccn3)cc21 CHEMBL5427835 EC50 1000.0 nM