Cc1ccc(-c2nc3ccccn3c2-c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)cc1 CHEMBL5419651 EC50 0.0 nM
CCc1ccc(-c2nc3ccccn3c2-c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)cc1 CHEMBL5397029 EC50 0.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2cnn(Cc3ccc(Cl)c(Cl)c3)c2)cc1 CHEMBL5440796 EC50 0.0 nM
COC(=O)c1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5425254 EC50 0.0 nM
Fc1ccc(-c2nc3ccccn3c2-c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)cc1 CHEMBL5426747 EC50 1.0 nM
FC(F)(F)c1ccc(-c2nc3ccccn3c2-c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)cc1 CHEMBL5434244 EC50 1.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2cn(Cc3ccccc3)nn2)cc1 CHEMBL5419791 EC50 1.0 nM
CC(=O)c1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5429867 EC50 1.0 nM
OCc1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5400735 EC50 1.0 nM
Clc1ccc(Cn2cc(-c3c(-c4ccc(Cl)c(Cl)c4)nc4ccccn34)nn2)cc1Cl CHEMBL5396305 EC50 2.0 nM
Clc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)cc1 CHEMBL5439022 EC50 2.0 nM
Clc1ccc(-c2nc3sccn3c2-c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)cc1 CHEMBL5408637 EC50 3.0 nM
O=[N+]([O-])c1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5425742 EC50 4.0 nM
Clc1ccc(-c2nc3sccn3c2/C=N/OCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL458603 EC50 5.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)cc1 CHEMBL5401908 EC50 5.0 nM
Nc1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5435896 EC50 6.0 nM
Clc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4sccn34)nn2)cc1 CHEMBL5397287 EC50 7.0 nM
Clc1ccc(-c2nc3sccn3c2-c2cn(Cc3ccccc3)nn2)cc1 CHEMBL5411992 EC50 7.0 nM
O/N=C/c1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5437829 EC50 7.0 nM
O=Cc1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5423627 EC50 8.0 nM
CS(=O)(=O)c1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)cc1 CHEMBL5437100 EC50 9.0 nM
COCc1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5398624 EC50 9.0 nM
Clc1ccc(-c2nc3sccn3c2-c2cn(Cc3ccccn3)nn2)cc1 CHEMBL5421493 EC50 10.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2cc(Cc3ccc(Cl)c(Cl)c3)no2)cc1 CHEMBL5396096 EC50 10.0 nM
CSc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)cc1 CHEMBL5432712 EC50 11.0 nM
CCC(=O)c1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5399445 EC50 11.0 nM
O=C(Nc1ccc2c(c1)N(C(=O)Cn1cccc1)c1ccccc1CC2)OC1CCCCC1 CHEMBL3763793 IC50 11.7 nM
Clc1ccc(-c2nc3sccn3c2-c2csc(Cc3ccc(Cl)c(Cl)c3)n2)cc1 CHEMBL5433607 EC50 13.0 nM
O=C(Nc1ccc2c(c1)N(C(=O)Cn1cccc1)c1ccccc1CC2)OC1CCCC1 CHEMBL3763399 IC50 13.9 nM
Clc1ccc(-c2nc3sccn3c2-c2nc(Cc3ccc(Cl)c(Cl)c3)no2)cc1 CHEMBL5434877 EC50 14.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2nnc(Cc3ccc(Cl)c(Cl)c3)s2)cc1 CHEMBL5438918 EC50 15.0 nM
Clc1ccc(Cn2cc(-c3c(-c4ccc(Cl)c(Cl)c4)nc4sccn34)nn2)cc1Cl CHEMBL5409045 EC50 16.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2cccn2Cc2ccc(Cl)c(Cl)c2)cc1 CHEMBL5399505 EC50 17.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2csc(Cc3ccc(Cl)c(Cl)c3)n2)cc1 CHEMBL5440050 EC50 18.0 nM
COc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)cc1OC CHEMBL5435703 EC50 19.0 nM
CC(C)OC(=O)Nc1ccc2c(c1)N(C(=O)COC1CCCC1)c1ccccc1CC2 CHEMBL3763536 IC50 19.5 nM
O=C(Nc1ccc2c(c1)N(C(=O)Cn1cccc1)c1ccccc1CC2)OC1CCC1 CHEMBL3763664 IC50 20.1 nM
CC(C)OC(=O)Nc1ccc2c(c1)N(C(=O)Cn1cccc1)c1ccccc1CC2 CHEMBL3764750 IC50 20.9 nM
CC(C)OC(=O)Nc1ccc2c(c1)N(C(=O)COCC(C)(C)C)c1ccccc1CC2 CHEMBL3765064 IC50 21.2 nM
O=C(Nc1ccc2c(c1)N(C(=O)Cn1cccc1)c1ccccc1CC2)OC1CC1 CHEMBL3763725 IC50 22.1 nM
Clc1ccc(-c2nc3ccccn3c2-c2nnc(Cc3ccc(Cl)c(Cl)c3)o2)cc1 CHEMBL5409712 EC50 23.0 nM
CC(C)OC(=O)Nc1ccc2c(c1)N(C(=O)COC1CCCCC1)c1ccccc1CC2 CHEMBL3764168 IC50 24.1 nM
CC(C)(C)OC(=O)Nc1ccc2c(c1)N(C(=O)Cn1cccc1)c1ccccc1CC2 CHEMBL3764583 IC50 31.9 nM
Clc1ccc(-c2nc3ccccn3c2-c2nc(Cc3ccc(Cl)c(Cl)c3)no2)cc1 CHEMBL5417795 EC50 35.0 nM
CCC(C)OCC(=O)N1c2ccccc2CCc2ccc(NC(=O)OC(C)C)cc21 CHEMBL3765692 IC50 35.3 nM
CCOC(=O)Nc1ccc2c(c1)N(C(=O)Cn1cccc1)c1ccccc1CC2 CHEMBL3763695 IC50 37.0 nM
CC(C)OC(=O)Nc1ccc2c(c1)N(C(=O)COC1CCC1)c1ccccc1CC2 CHEMBL3764324 IC50 37.6 nM
COc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)cc1 CHEMBL5434075 EC50 40.0 nM
Clc1ccc(-c2nc3ccccn3c2-c2cn(CCc3ccc(Cl)c(Cl)c3)nn2)cc1 CHEMBL5400588 EC50 40.0 nM
CC(c1ccccc1)n1cc(-c2c(-c3ccc(Cl)cc3)nc3ccccn23)nn1 CHEMBL5405148 EC50 40.0 nM
N#Cc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)cc1 CHEMBL5413864 EC50 60.0 nM
CC(C)OCC(=O)N1c2ccccc2CCc2ccc(NC(=O)OC(C)C)cc21 CHEMBL3763758 IC50 60.1 nM
Clc1ccc(-c2nc3ccccn3c2-c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)c(Cl)c1 CHEMBL5428723 EC50 62.0 nM
CCOC(=O)Nc1ccc2c(c1)N(C(=O)COC(C)(C)C)c1ccccc1CC2 CHEMBL3765243 IC50 70.8 nM
Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1ccnc1 CHEMBL104 IC50 80.0 nM
CC(C)OC(=O)Nc1ccc2c(c1)N(C(=O)COC1CC1)c1ccccc1CC2 CHEMBL3763979 IC50 81.5 nM
CC(C)OCC(=O)N1c2ccccc2CCc2ccc(NC(=O)OC(C)(C)C)cc21 CHEMBL3763569 IC50 116.0 nM
CCCN(CCC)CC(=O)N1c2ccccc2CCc2ccc(NC(=O)OC(C)C)cc21 CHEMBL3764215 IC50 116.4 nM
CC(=O)Nc1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5434255 EC50 134.0 nM
Fc1ccc(-c2nc3sccn3c2CNCCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4563092 EC50 150.0 nM
COc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4sccn34)nn2)cc1OC CHEMBL5416598 EC50 150.0 nM
CCCN(CCC)CC(=O)N1c2ccccc2CCc2ccc(NC(=O)OC(C)(C)C)cc21 CHEMBL3764619 IC50 152.9 nM
Clc1ccc(-c2nc3sccn3c2COCCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4438442 EC50 190.0 nM
CCCN(CCC)CC(=O)N1c2ccccc2CCc2ccc(NC(=O)OCC)cc21 CHEMBL3764049 IC50 210.0 nM
CC(C)(C)OC(=O)Nc1ccc2c(c1)N(C(=O)CN1CCCCC1)c1ccccc1CC2 CHEMBL3764753 IC50 216.2 nM
CCOC(=O)Nc1ccc2c(c1)N(C(=O)CN1CCOCC1)c1ccccc1CC2 CHEMBL3765016 IC50 235.0 nM
Clc1ccc(CCNCc2c(-c3ccccc3)nc3sccn23)cc1Cl CHEMBL4442038 EC50 240.0 nM
CC(C)OC(=O)Nc1ccc2c(c1)N(C(=O)CN1CCCCC1)c1ccccc1CC2 CHEMBL3763803 IC50 249.0 nM
COC(=O)Nc1ccc2c(c1)N(C(=O)CCN1CCOCC1)c1ccccc1CC2 CHEMBL3765163 IC50 288.0 nM
CON(C)C(=O)c1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5399035 EC50 313.0 nM
CCOC(=O)Nc1ccc2c(c1)N(C(=O)CCN1CCOCC1)c1ccccc1CC2 CHEMBL3765146 IC50 320.0 nM
Clc1ccc(CO/N=C/c2c(-c3ccc4ccccc4c3)nc3occn23)cc1Cl CHEMBL4465050 EC50 370.0 nM
Clc1ccc(CO/N=C/c2c(-c3ccc4ccccc4c3)nc3sccn23)cc1Cl CHEMBL4454940 EC50 380.0 nM
CCC(C)N(C)C(=O)c1cc2ccccc2c(-c2ccccc2Cl)n1 CHEMBL481537 IC50 390.0 nM
Clc1ccc(-c2nc3sccn3c2CNCCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4527619 EC50 400.0 nM
Clc1ccc(-c2nc3occn3c2/C=N/OCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4439746 EC50 410.0 nM
Cc1ccc(-c2nc3sccn3c2CNCCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4437007 EC50 440.0 nM
Clc1ccc(-c2nc3sccn3c2CNC2Cc3ccccc3C2)cc1 CHEMBL4442397 EC50 460.0 nM
FC(F)(F)c1ccc(CO/N=C/c2c(-c3ccc4ccccc4c3)nc3occn23)cc1 CHEMBL4449508 EC50 470.0 nM
Clc1ccc(CO/N=C/c2c(-c3ccc(Br)cc3)nc3sccn23)cc1Cl CHEMBL4562469 EC50 480.0 nM
Cc1ccc(-c2nc3sccn3c2/C=N/OCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4452961 EC50 490.0 nM
COc1ccc(-c2nc3sccn3c2/C=N/OCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4463067 EC50 490.0 nM
Nc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)cc1 CHEMBL5396120 EC50 500.0 nM
Cc1ccc(Nc2c(F)cccc2Cl)c(CC(=O)O)c1 CHEMBL404108 AC50 550.0 nM
Clc1ccc(CCNCc2c(-c3ccc(Br)cc3)nc3sccn23)cc1Cl CHEMBL4577011 EC50 560.0 nM
CCC(C)(C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@H]21 CHEMBL1064 AC50 570.0 nM
Clc1ccc(CO/N=C/c2c(-c3ccccc3)nc3sccn23)cc1Cl CHEMBL4457645 EC50 580.0 nM
CC(C)c1ccc(-c2nc3sccn3c2/C=N/OCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4469650 EC50 590.0 nM
NC(=O)c1cc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4ccccn34)nn2)ccc1Cl CHEMBL5408469 EC50 611.0 nM
CCOC(=O)Nc1ccc2c(c1)N(C(=O)CN1CCCCC1)c1ccccc1CC2 CHEMBL3763550 IC50 620.0 nM
Clc1ccc(CCNCc2c(-c3ccc(Cl)cc3)nc3sccn23)cc1 CHEMBL4522917 EC50 650.0 nM
COc1ccc(Cn2cc(-c3c(-c4ccc(Cl)cc4)nc4sccn34)nn2)cc1 CHEMBL5432241 EC50 656.0 nM
c1ccc2c(c1)CC(NCc1c(-c3ccc4ccccc4c3)nc3occn13)C2 CHEMBL4473295 EC50 660.0 nM
COc1ccc(-c2nc3sccn3c2CNCCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4574159 EC50 670.0 nM
Fc1ccc(-c2nc3sccn3c2/C=N/OCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4565112 EC50 670.0 nM
CCN(CC)CC(=O)N1c2ccccc2CCc2ccc(NC(=O)OC(C)C)cc21 CHEMBL3764651 IC50 680.0 nM
CCOC(=O)Nc1ccc2c(c1)N(C(=O)CN(CC)CC)c1ccccc1CC2 CHEMBL1622371 IC50 687.0 nM
COc1cccc(-c2nc3ccccc3c(=S)[nH]2)c1 CHEMBL3823873 EC50 690.0 nM
Clc1ccc(-c2nc3sccn3c2CNCCc2ccccc2)cc1 CHEMBL4449535 EC50 740.0 nM
C(=N/OCc1ccccc1)\c1c(-c2ccc3ccccc3c2)nc2occn12 CHEMBL4576432 EC50 840.0 nM
FC(F)(F)c1ccc(-c2nc3sccn3c2/C=N/OCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4452491 EC50 880.0 nM
Clc1ccc(-c2nc3ncccn3c2CNCCc2ccc(Cl)c(Cl)c2)cc1 CHEMBL4474143 EC50 920.0 nM
Clc1cccc(-c2nc3sccn3c2CNCCc2ccc(Cl)c(Cl)c2)c1 CHEMBL4453764 EC50 930.0 nM
Clc1ccc(CO/N=C/c2c(-c3cccc4ccccc34)nc3sccn23)cc1Cl CHEMBL4445350 EC50 940.0 nM
C(=N/OC1Cc2ccccc2C1)\c1c(-c2ccc3ccccc3c2)nc2occn12 CHEMBL4580898 EC50 980.0 nM
Clc1ccc(CO/N=C/c2c(-c3ccc4ccccc4c3)nc3occn23)cc1 CHEMBL4456609 EC50 990.0 nM