O=C(Nc1ccc(-c2nc3cc(NC(=O)C4CC4)ccc3[nH]2)cc1)c1ccccc1Cl CHEMBL386138 EC50 35.0 nM
COC(=O)CCCCC1SCC2NC(=O)NC21O CHEMBL1391310 IC50 139.1 nM
CC(C)C(=O)Nc1ccc2[nH]c(-c3ccc(NC(=O)c4ccccc4Cl)cc3)nc2c1 CHEMBL213426 EC50 147.0 nM
C[C@@H]1NC(=O)N[C@@H]1CCCCCC(=O)O CHEMBL1232381 IC50 149.12 nM
Cn1c(SCC(=O)Nc2cccc(Br)c2)nnc1-c1cc2ccccc2o1 CHEMBL1602811 IC50 167.27 nM
O=C(Nc1ccc(-c2nc3cc(NC(=O)c4ccccc4Cl)ccc3[nH]2)cc1)c1ccccc1F CHEMBL384623 EC50 170.0 nM
Cc1ccc(-c2cc(-c3ccc(F)cc3)nc3ncnc(N)c23)cc1 CHEMBL1384281 IC50 177.87 nM
Cc1ccc(-c2cc(-c3ccccc3)c3c(N)ncnc3n2)cc1 CHEMBL1575389 IC50 177.89 nM
COC(=O)c1cc2n3ccccc3c(C)c(-c3ccccc3)c-2c1C(=O)OC CHEMBL1326814 IC50 185.5 nM
COc1ccc(-c2cc(-c3ccccc3)c3c(N)ncnc3n2)cc1 CHEMBL1324779 IC50 220.17 nM
O=C(Nc1ccc(-c2nc3cc(NC(=O)[C@@H]4C[C@H]4F)ccc3[nH]2)cc1)c1ccccc1Cl CHEMBL212336 EC50 260.0 nM
Cc1ccccc1C(=O)Nc1ccc(-c2nc3cc(NC(=O)c4ccccc4Cl)ccc3[nH]2)cc1 CHEMBL213665 EC50 260.0 nM
O=C(Nc1ccc(-c2nc3cc(NC(=O)c4ccccc4Cl)ccc3[nH]2)cc1)c1ccccc1 CHEMBL215539 EC50 270.0 nM
COC(=O)c1c(Cl)c2n3ccccc3c(C)c(-c3ccccc3)c-2c1C(=O)OC CHEMBL1544403 IC50 303.35 nM
CCCCOc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2)cc1 CHEMBL1433074 IC50 330.11 nM
O=C(Nc1ccc(-c2nc3cc(NC(=O)C4(c5ccccc5)CC4)ccc3[nH]2)cc1)c1ccccc1Cl CHEMBL214562 EC50 370.0 nM
COC(=O)CCCC[C@H]1SC[C@H]2NC(=O)N[C@]21O CHEMBL1454198 IC50 389.38 nM
Cc1ccc(NC(=O)CSc2nc3ccccc3c3nc(CCc4c(C)n[nH]c4C)nn23)cc1F CHEMBL1565040 IC50 473.9 nM
Cc1ccc(S(=O)(=O)NC(=O)Nc2ccc(N(C)C)cc2)cc1 CHEMBL312032 IC50 748.25 nM
C=CCn1c(SCC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)nnc1-c1ccccc1 CHEMBL1482670 IC50 774.16 nM
Cc1nc2ccc3nc(NC(=O)c4ccc5c(c4)OCCO5)sc3c2s1 CHEMBL1417231 IC50 812.55 nM
COc1ccc(C(=O)Nc2nc3ccc4nc(C)sc4c3s2)cc1 CHEMBL1392806 IC50 861.97 nM
O=C(Nc1ccc(-c2nc3cc(NC(=O)C4CCC4)ccc3[nH]2)cc1)c1ccccc1Cl CHEMBL214445 EC50 986.0 nM