N#Cc1cn(-c2c[nH]n(-c3cc(N4CC(F)(F)C4)ncn3)c2=O)nn1 CHEMBL3115317 IC50 70.0 nM
N#Cc1cn(-c2c[nH]n(-c3cc(N4CC(F)(F)C4)ncn3)c2=O)cn1 CHEMBL3640646 IC50 90.0 nM
N#Cc1cn(-c2c[nH]n(-c3cc(N4CCC(F)(F)C4)ncn3)c2=O)nn1 CHEMBL3640645 IC50 130.0 nM
N#Cc1cn(-c2c[nH]n(-c3cc(N4CCCCO4)ncn3)c2=O)nn1 CHEMBL3642645 IC50 170.0 nM
O=c1c(-c2cccnc2)c[nH]n1-c1cc(N2CCOCC2)ncn1 CHEMBL3651449 IC50 180.0 nM
N#Cc1cn(-c2c[nH]n(-c3cc(N4CCCOCC4)ncn3)c2=O)cn1 CHEMBL3642643 IC50 180.0 nM
O=C(O)c1ccc(-c2ccc(C(=O)O)cn2)nc1 CHEMBL332005 IC50 185.0 nM
O=C(O)c1ccc(-n2[nH]cc(-c3cncc(Br)c3)c2=O)nc1 CHEMBL3640754 IC50 260.0 nM
CCOc1ccc(NC(=O)c2ccc(-c3ccc(C(=O)O)cn3)nc2)cc1 CHEMBL124527 IC50 320.0 nM
N#Cc1cn(-c2c[nH]n(-c3cc(N4CCCOCC4)ncn3)c2=O)nn1 CHEMBL3642644 IC50 380.0 nM
O=c1c(-c2ccc(Cl)nc2)c[nH]n1-c1cc(N2CCOCC2)ncn1 CHEMBL3651450 IC50 480.0 nM
O=C(O)C1CN(c2cc(-n3[nH]cc(-n4ccnc4)c3=O)ncn2)C1 CHEMBL3640643 IC50 540.0 nM
Cc1cc(C)n(-c2cc(-n3[nH]cc(-c4cccnc4)c3=O)ncn2)n1 CHEMBL3651451 IC50 700.0 nM
CN(C)C1CN(c2cc(-n3[nH]cc(-n4ccnn4)c3=O)ncn2)C1 CHEMBL3640644 IC50 760.0 nM
O=c1c(-c2cccnc2)c[nH]n1-c1nnc(-c2ccc(Cl)cc2)s1 CHEMBL3651452 IC50 880.0 nM
O=c1c(-n2ccnn2)c[nH]n1-c1cc(N2CCN(C3CCC3)CC2)ncn1 CHEMBL3640642 IC50 880.0 nM
COCCN1CCN(c2cc(-n3[nH]cc(-c4cccnc4)c3=O)ncn2)CC1 CHEMBL3651453 IC50 890.0 nM
O=C(NCc1ccnc(-n2[nH]cc(-c3cccnc3)c2=O)c1)Nc1c(Cl)cccc1Cl CHEMBL3640757 IC50 900.0 nM
CC(C)(C)NC(=O)c1ccc(-n2[nH]cc(-c3cccnc3)c2=O)nc1 CHEMBL3640755 IC50 910.0 nM
O=c1c(-c2cccnc2)c[nH]n1-c1cnccn1 CHEMBL3651454 IC50 930.0 nM
COc1ccc(S(=O)(=O)NC(=O)c2ccc(C(=O)[O-])nc2)cc1 CHEMBL1744254 IC50 1000.0 nM