CC(C)c1ccc(CC(=O)N2CCN(c3ccc(Cl)nn3)CC2)cc1 CHEMBL5082138 IC50 0.4 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc(Cl)nn3)CC2)cc1 CHEMBL363699 IC50 0.7 nM
CC(C)c1ccc(CC(=O)N2CCN(c3ccc(C#N)nn3)CC2)cc1 CHEMBL5077276 IC50 1.0 nM
CC(C)c1ccc(CC(=O)N2CCN(c3cnc(Cl)cn3)CC2)cc1 CHEMBL5094733 IC50 1.8 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc(C#N)nn3)CC2)cc1 CHEMBL5078496 IC50 4.0 nM
CC(C)c1ccc(CC(=O)N2CCN(c3cnc(C#N)nc3)CC2)cc1 CHEMBL5085732 IC50 10.0 nM
CC(C)c1ccc(OC(=O)N2CCN(c3ccc(C#N)nn3)CC2)cc1 CHEMBL5082695 IC50 10.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc([N+](=O)[O-])cn3)CC2)cc1 CHEMBL5093027 IC50 20.0 nM
CSc1cccc(NC(=O)CCc2c(C)nc3c4cccnc4nn3c2C)c1 CHEMBL3410246 IC50 25.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3cnc(C#N)cn3)CC2)cc1 CHEMBL5075383 IC50 29.0 nM
CC(C)c1ccc(CC(=O)N2CCN(c3ccc(C#N)cn3)CC2)cc1 CHEMBL5078248 IC50 60.0 nM
CC(C)(C)c1ccc(CC(=O)N2CCN(c3ccc(C#N)cn3)CC2)cc1 CHEMBL5092780 IC50 60.0 nM
CC(C)c1ccc(NC(=O)CCc2nc(O)c3c4c(sc3n2)CCC4)cc1 CHEMBL3410245 IC50 120.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3nccc(C#N)n3)CC2)cc1 CHEMBL5088913 IC50 140.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ncc(Br)cn3)CC2)cc1 CHEMBL5088098 IC50 160.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3cnc(C#N)nc3)CC2)cc1 CHEMBL5092773 IC50 170.0 nM
CCS(=O)(=O)Nc1ccc(C(=O)NC2CC3CCC2C3)cc1 CHEMBL3410244 IC50 180.0 nM
N#Cc1ccc(N2CCN(C(=O)Cc3ccc(C4CC4)cc3)CC2)nc1 CHEMBL5073319 IC50 200.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc(Br)cn3)CC2)cc1 CHEMBL5076791 IC50 220.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc(Cl)cn3)CC2)cc1 CHEMBL5070550 IC50 220.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3cc(C#N)ccn3)CC2)cc1 CHEMBL5079891 IC50 230.0 nM
CC(C)c1ccc(CC(=O)N2CCN(c3nccc(Cl)n3)CC2)cc1 CHEMBL5086917 IC50 270.0 nM
CC(=O)Nc1ccc(NC(=O)CCc2c(C)nc3c4cccnc4nn3c2C)cc1 CHEMBL3410400 IC50 350.0 nM
CC(C)c1ccc(OC(=O)N2CCN(c3ccc(C#N)cn3)CC2)cc1 CHEMBL5085445 IC50 420.0 nM
CC(C)Cc1ccc(NC(=O)N2CCN(c3ccc(C#N)cn3)CC2)cc1 CHEMBL5089188 IC50 490.0 nM
CC(C)(C)c1ccc(NC(=O)N2CCN(c3ccc(C#N)cn3)CC2)cc1 CHEMBL5075792 IC50 510.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc(C#N)cc3)CC2)cc1 CHEMBL5089505 IC50 580.0 nM
Cc1nc2c3cccnc3nn2c(C)c1CCC(=O)Nc1cccc(F)c1 CHEMBL3410256 IC50 620.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc(C#N)cn3)CC2)cc1 CHEMBL5074576 IC50 640.0 nM
CC(C)c1ccc(NC(=O)N2CCN(c3ccc(C(F)(F)F)cn3)CC2)cc1 CHEMBL5093358 IC50 770.0 nM
Cc1nc2c3cccnc3nn2c(C)c1CCC(=O)Nc1cccc(C(F)(F)F)c1 CHEMBL3410398 IC50 830.0 nM
CC(C)c1ccc(C(O)C(=O)N2CCN(c3ccc(C#N)cn3)CC2)cc1 CHEMBL5086368 IC50 990.0 nM