CC(C)(C)NS(=O)(=O)c1ccc2c(c1)C(=O)c1ccccc1C2=O CHEMBL4290650 Kd 1.45 nM
Cc1ncc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(Cc3sc(C)nc3C)c2=O)s1 CHEMBL4290666 EC50 4.8 nM
Cc1nc(C)c(Cn2c(=O)n(Cc3cnn(C)c3)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)s1 CHEMBL4282478 EC50 6.0 nM
Cc1ncc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(CC3CC3)c2=O)s1 CHEMBL4290954 EC50 19.0 nM
Cn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(CF)CC4)ccc3n(Cc3ccn(C)n3)c2=O)cn1 CHEMBL4459798 IC50 20.0 nM
Cn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(Cc3ccn(C)n3)c2=O)cn1 CHEMBL4518815 IC50 20.0 nM
Cc1cc(Cn2c(=O)n(Cc3cnn(C)c3)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)n(C)n1 CHEMBL4293745 EC50 23.0 nM
Cc1cc(Cn2c(=O)n(Cc3cnc(C)s3)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)n(C)n1 CHEMBL4286938 EC50 26.0 nM
Cn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(CC3CC3)c2=O)cn1 CHEMBL4278621 EC50 29.0 nM
[2H]C([2H])([2H])C1(NS(=O)(=O)c2ccc3c(c2)c(=O)n(Cc2cnn(C)c2)c(=O)n3Cc2ccn(C)n2)CC1 CHEMBL4459166 IC50 30.0 nM
Cc1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(Cc3cc(C)nn3C)c2=O)on1 CHEMBL4294475 EC50 38.0 nM
C#CCn1c(=O)n(Cc2cnc(C)s2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4290350 EC50 45.0 nM
Cc1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(CC3CC3)c2=O)on1 CHEMBL4286164 EC50 49.0 nM
C#CCn1c(=O)n(Cc2cnn(C)c2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4289269 EC50 52.0 nM
Cc1cc(Cn2c(=O)n(Cc3nnc(C)s3)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)n(C)n1 CHEMBL4293317 EC50 64.0 nM
Cn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(CC3COC3)c2=O)cn1 CHEMBL4285867 EC50 69.0 nM
C#CCn1c(=O)n(Cc2cc(C)no2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4294064 EC50 76.0 nM
CCn1c(=O)n(Cc2cnn(C)c2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4282082 EC50 78.0 nM
CCn1c(=O)n(Cc2cnn(C)c2)c(=O)c2cc(S(=O)(=O)NC3(CF)CC3)ccc21 CHEMBL4438105 IC50 80.0 nM
Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OC[C@H]2NC[C@H](O)[C@@H]2O)[C@@H](O)[C@H]1O CHEMBL1230692 IC50 120.0 nM
CCn1c(=O)n(Cc2cc(C)no2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4282778 EC50 120.0 nM
CCn1c(=O)n(Cc2nnc(C)s2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4287646 EC50 120.0 nM
Cc1nc(C)c(Cn2c(=O)n(C)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)s1 CHEMBL4285012 EC50 180.0 nM
C#CCn1c(=O)n(CC#N)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4287255 EC50 250.0 nM
C#CCn1c(=O)n(C)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4285603 EC50 250.0 nM
CC1(NS(=O)(=O)c2ccc3c(c2)c(=O)n(CC#N)c(=O)n3CC2CC2)CC1 CHEMBL4277012 EC50 270.0 nM
Cc1cc(Cn2c(=O)n(CC#N)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)n(C)n1 CHEMBL4279324 EC50 280.0 nM
Cc1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(CC3COC3)c2=O)on1 CHEMBL4283898 EC50 280.0 nM
Cn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(CF)CC4)ccc3n(C)c2=O)cn1 CHEMBL4452307 IC50 290.0 nM
Cn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C(F)F)CC4)ccc3n(Cc3ccn(C)n3)c2=O)cn1 CHEMBL4456850 IC50 320.0 nM
Cn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(C)c2=O)cn1 CHEMBL4283111 IC50 330.0 nM
Cn1c(=O)n(Cc2cnn(CC#N)c2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4283434 EC50 370.0 nM
Cc1cc(Cn2c(=O)n(C)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)n(C)n1 CHEMBL4292216 EC50 380.0 nM
Cn1c(=O)n(Cc2cn[nH]c2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4286783 EC50 380.0 nM
Cn1c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc2n(CC2CC2)c1=O CHEMBL4290899 EC50 440.0 nM
COc1ccc(Cn2c(=O)n(C)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)cc1 CHEMBL4281824 EC50 450.0 nM
CCn1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(C)c2=O)cn1 CHEMBL4278860 EC50 450.0 nM
Cc1nnc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(C)c2=O)s1 CHEMBL4279282 EC50 470.0 nM
Cc1cc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(C)c2=O)on1 CHEMBL4279961 EC50 470.0 nM
Cc1ncc(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(C)c2=O)s1 CHEMBL4291874 EC50 480.0 nM
Cn1c(=O)n(Cc2cnc(N)s2)c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc21 CHEMBL4291445 EC50 480.0 nM
Cn1c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc2n(Cc2ccc(F)cc2)c1=O CHEMBL4277949 EC50 530.0 nM
Cn1c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc2n(CC2CCCCC2)c1=O CHEMBL4283025 EC50 560.0 nM
Cc1noc(C)c1Cn1c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc2n(C)c1=O CHEMBL4287190 EC50 620.0 nM
Cc1oncc1Cn1c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc2n(C)c1=O CHEMBL4295120 EC50 770.0 nM
COc1cccc(Cn2c(=O)n(C)c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc32)c1 CHEMBL4293083 EC50 860.0 nM
Cc1nnsc1Cn1c(=O)c2cc(S(=O)(=O)NC3(C)CC3)ccc2n(C)c1=O CHEMBL4290368 EC50 880.0 nM
Cc1nc(C)c(Cn2c(=O)c3cc(S(=O)(=O)NC4(C)CC4)ccc3n(C)c2=O)s1 CHEMBL4283598 EC50 910.0 nM