CC#Cc1ccc2c(=O)[nH]c(CSc3ncccn3)nc2c1C CHEMBL5191676 IC50 14.0 nM
Cc1ccc2c(=O)[nH]c(-c3ccc(C(C)(C)O)cc3)cn12 CHEMBL5199558 IC50 67.0 nM
CC#Cc1ccc2c(=O)[nH]c(CSc3ccc(C(=O)O)cc3)nc2c1C CHEMBL5207717 IC50 99.0 nM
Cn1ncnc1[C@H]1c2n[nH]c(=O)c3cc(F)cc(c23)N[C@@H]1c1ccc(F)cc1 CHEMBL3137320 IC50 140.0 nM
Cc1cccc2c(=O)[nH]c(CSc3ncccn3)nc12 CHEMBL5187963 IC50 200.0 nM
COc1ccc(OC)c2c1sc1nnc(N)n12 CHEMBL5404785 IC50 240.0 nM
Cc1ccc2c(c1)sc1nnc(N)n12 CHEMBL5431108 pIC50 467.74 nM
Cc1ccc2c(=O)[nH]c(CSc3ncccn3)nc2c1C CHEMBL5186007 IC50 550.0 nM
