O=C1NC[C@@H](c2ccccn2)[C@@H](O)c2cc(Cl)c(Cl)cc21 CHEMBL5189477 IC50 362.0 nM
O=C1NCC(c2ccccn2)[C@@H](O)c2cc(Cl)c(Cl)cc21 CHEMBL5284069 IC50 362.0 nM
Nc1ncc2c(n1)CNC(=O)c1[nH]c(Br)c(Br)c1-2 CHEMBL5172255 IC50 427.0 nM
NC(=O)c1cccc(NC(=O)/C=C\C(=O)N2CCN(c3ccc(F)cc3)CC2)c1 CHEMBL4089522 IC50 560.0 nM
Cn1ncnc1[C@H]1c2n[nH]c(=O)c3cc(F)cc(c23)N[C@@H]1c1ccc(F)cc1 CHEMBL3137320 Kd(app) 1000.0 nM
