Cn1ncnc1[C@H]1c2n[nH]c(=O)c3cc(F)cc(c23)N[C@@H]1c1ccc(F)cc1 CHEMBL3137320 Kd(app) 0.7 nM
O=C(c1cc(Cc2n[nH]c(=O)c3ccccc23)ccc1F)N1CCn2c(nnc2-c2ccc(Br)o2)C1 CHEMBL5402698 IC50 1.0 nM
O=C(c1cc(Cc2n[nH]c(=O)c3ccccc23)ccc1F)N1CCN(C(=O)C2CC2)CC1 CHEMBL521686 IC50 13.5 nM
C[C@]1(c2nc3c(C(N)=O)cccc3[nH]2)CCCN1 CHEMBL506871 Kd(app) 105.0 nM
Cn1ncnc1[C@@H]1c2n[nH]c(=O)c3cc(F)cc(c23)N[C@H]1c1ccc(F)cc1 CHEMBL3764816 IC50 254.0 nM
NC(=O)c1cccc2cn(-c3ccc([C@@H]4CCCNC4)cc3)nc12 CHEMBL1094636 Kd(app) 272.0 nM
O=C1NCC2c3c(cccc31)CCN2C(=O)Cc1cccnc1 CHEMBL595018 IC50 440.0 nM
Cc1cc(C)c2nc(CSc3ncccn3)[nH]c(=O)c2c1 CHEMBL5198711 IC50 500.0 nM
CNCc1ccc(-c2[nH]c3cc(F)cc4c3c2CCNC4=O)cc1 CHEMBL1173055 Kd(app) 503.0 nM
O=C1NCC2c3c(cccc31)CCN2C(=O)CCc1cnccn1 CHEMBL609002 IC50 660.0 nM
CN(C)CC(=O)Nc1ccc2[nH]c(=O)c3ccccc3c2c1 CHEMBL372303 pIC50 758.58 nM
Cc1cc(Br)cc2c(=O)[nH]c(CSc3ncccn3)nc12 CHEMBL5181770 IC50 800.0 nM
Cc1cc(I)cc2c(=O)[nH]c(CSc3ccc(C(=O)O)cc3)nc12 CHEMBL5200299 IC50 800.0 nM