CC(=O)c1ccc(Cn2nc3c(c2Nc2ccc(F)c(C)c2)C(=O)N(C)C2=NC(C)(C)CN23)cc1 CHEMBL3678507 Ki 0.1 nM
CC(=O)c1ccc(Cn2nc3c(c2Nc2ccc(F)cc2)C(=O)N(C)C2=NC(C)(C)CN23)cc1 CHEMBL3678504 Ki 0.2 nM
CC(=O)c1ccc(Cn2nc3c(c2Nc2ccc(F)c(F)c2)C(=O)N(C)C2=NC(C)(C)CN23)cc1 CHEMBL3678506 Ki 0.3 nM
CC(O)c1ccc(Cn2nc3c(c2Nc2ccc(F)cc2)C(=O)N(C)C2=NC(C)(C)CN23)cc1 CHEMBL3678505 Ki 0.5 nM
COc1ccc2c([C@H]3CCc4ccc(Cl)cc43)nccc2c1OC CHEMBL3601563 IC50 2.0 nM
COc1ccc2c(N[C@@H](C)Cc3cc(C)[nH]n3)ncnc2c1OC CHEMBL4128481 IC50 42.0 nM
CC(C)c1n[nH]c2c(=O)[nH]c(Cc3cccc(Cl)c3)nc12 CHEMBL512790 IC50 54.0 nM
CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)NCCCCCCO)ccc3OCC)nc12 CHEMBL3401745 IC50 62.0 nM
COc1ccc2c(NC(C)Cc3cc(C)[nH]n3)ncnc2c1OC CHEMBL4127641 IC50 118.0 nM
CC1=C(C(=O)O[C@H](C)c2ccccc2)C(c2ccc3c(cnn3C)c2)C(C(=O)O[C@H](C)c2ccccc2)=C(C)N1 CHEMBL5180169 IC50 145.0 nM
CCOCCCCOc1ccc2cc1Oc1ccc(cc1)C[C@H]1c3cc(c(OC)cc3CCN1C)Oc1c(OC)c(OC)cc3c1[C@@H](C2)N(C)CC3 CHEMBL454806 IC50 350.0 nM
C[C@@H](c1ccc2ncccc2c1)c1nnc2ccc(-c3ccc(F)c(F)c3)nn12 CHEMBL2431822 IC50 452.0 nM
C[C@@H](c1ccc2ncccc2c1)c1nnc2ccc(-c3cccc(C#N)c3)nn12 CHEMBL2431826 IC50 462.0 nM
C[C@@H](c1ccc2ncccc2c1)c1nnc2ccc(-c3cnn(C)c3)nn12 CHEMBL2431819 IC50 580.0 nM
CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCN(C)CC4)ccc3OCC)nc12 CHEMBL192 IC50 600.0 nM
COc1ccc2c(N[C@H](C)Cc3cc(C)[nH]n3)ncnc2c1OC CHEMBL4129844 IC50 777.0 nM
CC(C)c1nn(C)c2c(=O)[nH]c(Cc3ccccc3OCCN3CCOCC3)nc12 CHEMBL466474 IC50 790.0 nM