CCOc1ccc(OC2CCN(c3ncc(C(=O)NO)cn3)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 CHEMBL3936651 IC50 0.13 nM
CCCc1nn(C)c2c(O)nc(-c3cc(C(C)=O)ccc3OCC)nc12 CHEMBL377168 IC50 0.9 nM
CCc1ccc([C@@H]2c3[nH]c4ccccc4c(=O)c3CN2c2ncc(-c3ccccn3)cn2)s1 CHEMBL4217054 IC50 1.2 nM
COCCNc1cc(O)c2c(=O)c3c(-c4nccs4)[nH]c(Cc4ccc5c(c4)OCO5)c3oc2c1 CHEMBL4218772 IC50 1.2 nM
CCCc1nn(C)c2c(O)nc(-c3cc(C(=O)CN4CCOCC4)ccc3OCC)nc12 CHEMBL209460 IC50 1.4 nM
CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)s4)ccc3OCC)nc12 CHEMBL4212186 IC50 1.4 nM
CCc1ccc([C@@H]2c3[nH]c4ccccc4c(=O)c3CN2c2ncc(-c3ccccn3)cn2)o1 CHEMBL4217579 IC50 1.5 nM
CCc1ccc(C2c3[nH]c4ccccc4c(=O)c3CN2c2ncc(-c3ccccn3)cn2)o1 CHEMBL4212630 IC50 2.3 nM
CCOc1ccc(CC2CC(C(=O)NO)C2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 CHEMBL3900593 IC50 2.6 nM
CCc1ccc(C2c3[nH]c4ccccc4c(=O)c3CN2c2ncccn2)s1 CHEMBL4218398 IC50 3.7 nM
CCc1ccc([C@H]2c3[nH]c4ccccc4c(=O)c3CN2c2ncc(-c3ccccn3)cn2)o1 CHEMBL4208249 IC50 3.8 nM
CCc1ccc(C2c3[nH]c4ccccc4c(=O)c3CN2c2ncc(-c3ccccn3)cn2)s1 CHEMBL4209716 IC50 4.8 nM
CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)NCCCCCCO)ccc3OCC)nc12 CHEMBL3401745 IC50 5.2 nM
CCc1ccc(C2c3[nH]c4ccccc4c(=O)c3CN2c2ncccn2)o1 CHEMBL4204725 IC50 6.2 nM
CCN1Cc2nc3ccc(C#N)cc3c(NCc3ccc(OC)c(Cl)c3)c2C1=O CHEMBL4072903 IC50 6.6 nM
CCc1ccc([C@H]2c3[nH]c4ccccc4c3C[C@@H]3C(=O)N(CC)C(=O)N23)o1 CHEMBL4284224 IC50 10.0 nM
CCN1C(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3sccc3C)N2C1=O CHEMBL4285199 IC50 13.0 nM
CCCOc1ccc(NC(=O)CN2CCN(C)CC2)cc1-c1nc(CC)c(CC)c(=O)[nH]1 CHEMBL4462192 IC50 19.8 nM
CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCN(C)CC4)ccc3OCC)nc12 CHEMBL192 IC50 24.0 nM
COc1ccc(CNc2c3c(nc4ccc(C#N)cc24)CCN(C(C)=O)C3)cc1Cl CHEMBL4062273 IC50 30.1 nM
CCc1ccc([C@H]2c3[nH]c4ccccc4c(=O)c3CN2c2ncc(-c3ccccn3)cn2)s1 CHEMBL4205338 IC50 34.1 nM
CCCOc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1-c1nc(CC)c(CC)c(=O)[nH]1 CHEMBL2180945 IC50 45.6 nM
CCc1ccc([C@@H]2c3[nH]c4ccccc4c3C[C@H]3C(=O)N(CC)C(=O)N23)s1 CHEMBL4277243 IC50 56.0 nM
CCN1C(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccc(C)o3)N2C1=O CHEMBL4292389 IC50 62.0 nM
CCCCN1C(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccc(CC)s3)N2C1=O CHEMBL4280648 IC50 107.0 nM
CCc1ccc([C@@H]2c3[nH]c4ccccc4c3C[C@H]3C(=O)N(CC)C(=O)N23)o1 CHEMBL4281766 IC50 127.0 nM
CN1CC(=O)N2[C@H](c3ccc(Br)s3)c3[nH]c4ccccc4c3C[C@@H]2C1=O CHEMBL4289471 IC50 136.0 nM
CCCCOc1ncc(C(C)=O)cc1-c1nc(O)c2nn(Cc3ccccn3)c(CCC)c2n1 CHEMBL210603 IC50 183.0 nM
CCc1ccc(C2c3[nH]c4ccccc4c3C(=O)CN2c2ncc(-c3ccc(OC)c(OC)c3)cn2)s1 CHEMBL4287438 IC50 253.0 nM
CCc1ccc(C2c3[nH]c4ccccc4c3C(=O)CN2c2ncc(-c3ccc(OC)c(OC)c3)cn2)o1 CHEMBL4292970 IC50 288.0 nM
CCc1c2nc(-c3cc(S(=O)(=O)N4CCN(CC)CC4)cnc3OCCOC)[nH]c(=O)c2nn1Cc1ccccn1 CHEMBL209157 IC50 386.0 nM
CN1CC(=O)N2[C@H](c3ccc4c(c3)OCO4)c3[nH]c4ccccc4c3C[C@@H]2C1=O CHEMBL779 IC50 402.0 nM
O=c1n(Cc2ccc(Cl)cc2)c2sc3c(c2c2ncnn12)CCCC3 CHEMBL1463540 IC50 460.0 nM
CCCCOc1ncc(C(C)=O)cc1-c1nc(O)c2nn(C3CN(CC)C3)c(CC)c2n1 CHEMBL210930 IC50 840.0 nM