CCCCC[C@H](CC(=O)NO)C(=O)N[C@H](C(=O)N1CCC[C@H]1CO)C(C)C CHEMBL308333 Ki 0.3 nM
CCCC[C@H](CC(=O)NO)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL122067 IC50 1.0 nM
Cc1cnc(NC(=O)[C@@H]2CC3(CC3)CN2C(=O)[C@@H](CC(=O)NO)CC2CCCC2)s1 CHEMBL4637933 IC50 2.78 nM
Cc1csc(NC(=O)[C@@H]2CC3(CC3)CN2C(=O)[C@@H](CC(=O)NO)CC2CCCC2)n1 CHEMBL4638057 IC50 2.99 nM
Cc1ccc(NC(=O)[C@@H]2CC3(CC3)CN2C(=O)[C@@H](CC(=O)NO)CC2CCCC2)cc1 CHEMBL4632607 IC50 3.58 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccccc2)no1)NO CHEMBL4641062 IC50 3.77 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccc(F)cc2C(F)(F)F)no1)NO CHEMBL4635911 IC50 4.11 nM
CCCCc1ccc(-c2noc([C@@H]3CC4(CC4)CN3C(=O)[C@@H](CC(=O)NO)CC3CCCC3)n2)cc1 CHEMBL4643984 IC50 4.24 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccc(C(F)(F)F)cc2F)no1)NO CHEMBL4649534 IC50 4.85 nM
CCCC[C@H](CC(=O)NO)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1ccc(F)cn1 CHEMBL4639327 IC50 4.92 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccc(F)cn2)no1)NO CHEMBL4641416 IC50 5.01 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccc(C3CC3)cc2)no1)NO CHEMBL4636545 IC50 5.01 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccc(Br)cc2)no1)NO CHEMBL4643967 IC50 5.48 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1ccc(F)cn1)NO CHEMBL4636221 IC50 5.87 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1cnccn1)NO CHEMBL4634572 IC50 5.87 nM
CN(C)C(=O)[C@@H](NC(=O)[C@H](CC1CCCCC1)CN(O)C=O)C(C)(C)C CHEMBL90193 IC50 6.0 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1ccc(Br)cc1)NO CHEMBL4637166 IC50 6.12 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1ccccc1)NO CHEMBL4640974 IC50 6.42 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccc(C(F)(F)F)cc2Cl)no1)NO CHEMBL4645966 IC50 6.47 nM
CCCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL431210 IC50 7.0 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1ccc(F)cc1C(F)(F)F)NO CHEMBL4635093 IC50 7.01 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2cc(F)cc(F)c2F)no1)NO CHEMBL4637631 IC50 7.08 nM
C=C1C[C@@H](C(=O)Nc2ccc(F)cn2)N(C(=O)[C@@H](CC(=O)NO)CC2CCCC2)C1 CHEMBL4642360 IC50 7.15 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2ccc(C(F)(F)F)cc2)no1)NO CHEMBL4635263 IC50 7.19 nM
CN(C)C(=O)[C@@H](NC(=O)[C@H](CC1CCCC1)CN(O)C=O)C(C)(C)C CHEMBL316099 IC50 8.0 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1nccs1)NO CHEMBL4645936 IC50 8.74 nM
CCc1ccc(-c2noc([C@@H]3CC4(CC4)CN3C(=O)[C@@H](CC(=O)NO)CC3CCCC3)n2)cc1 CHEMBL4646467 IC50 8.81 nM
Cc1cnc(NC(=O)[C@@H]2CCCN2C(=O)[C@@H](CC(=O)NO)CC2CCCC2)s1 CHEMBL4641901 IC50 8.94 nM
Cc1ccc(-c2noc([C@@H]3CC4(CC4)CN3C(=O)[C@@H](CC(=O)NO)CC3CCCC3)n2)cc1 CHEMBL4640884 IC50 9.26 nM
CCCC[C@H](CC(=O)NO)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1ncc(C)s1 CHEMBL4644600 IC50 9.42 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1ccncn1)NO CHEMBL4638180 IC50 9.53 nM
CCCCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL96864 IC50 10.0 nM
CC(C)C[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL413726 IC50 10.0 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CCC[C@H]1C(=O)Nc1ccc(F)cn1)NO CHEMBL4636076 IC50 10.9 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1C(=O)Nc1cccnn1)NO CHEMBL4645201 IC50 13.1 nM
O=C(C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(-c2cnccn2)no1)NO CHEMBL4643686 IC50 16.1 nM
CCCC[C@H](CS)C(=O)N[C@@H](CCCCN)C(=O)Nc1ccc([N+](=O)[O-])cc1 CHEMBL325246 Ki 19.0 nM
C=CCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL540441 IC50 20.0 nM
CN(C)C(=O)[C@@H](NC(=O)[C@@H](CN(O)C=O)C1CCCC1)C(C)(C)C CHEMBL328502 IC50 20.0 nM
CC(C)CC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL91882 IC50 20.0 nM
CCSC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL91835 IC50 20.0 nM
CN(C)C(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)CN(O)C=O)C(C)(C)C CHEMBL328688 IC50 20.0 nM
Cc1noc([C@@H]2CC3(CC3)CN2C(=O)[C@@H](CC(=O)NO)CC2CCCC2)n1 CHEMBL4649755 IC50 29.3 nM
CC#CC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL91461 IC50 30.0 nM
C=CC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL93648 IC50 30.0 nM
CCCCCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL315668 IC50 30.0 nM
CCCCC[C@H](CC(=O)NO)C(=O)N[C@H](C(=O)N1CCC[C@@H]1CO)C(C)C CHEMBL5191348 IC50 30.0 nM
Cn1cc(NC(=O)[C@@H]2CC3(CC3)CN2C(=O)[C@@H](CC(=O)NO)CC2CCCC2)cn1 CHEMBL4641571 IC50 30.2 nM
CCCCCCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL88314 IC50 40.0 nM
CC(C)[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL90378 IC50 50.0 nM
CCCCCCCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL314241 IC50 50.0 nM
CCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL327700 IC50 50.0 nM
CC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL90091 IC50 70.0 nM
CCCC[C@@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL93332 IC50 70.0 nM
CCCCC(CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL84969 IC50 70.0 nM
C[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL92692 IC50 100.0 nM
COc1ccc(C[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C)cc1 CHEMBL94197 IC50 200.0 nM
CCCC[C@H](CC(=O)O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL422256 IC50 200.0 nM
CCCC[C@H](CC(=O)NN)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL120479 IC50 200.0 nM
CN(C)C(=O)[C@@H](NC(=O)[C@@H](CN(O)C=O)c1ccc(Cl)cc1)C(C)(C)C CHEMBL94198 IC50 500.0 nM
CCCC[C@@H](C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C)C(C)N(O)C=O CHEMBL91105 IC50 600.0 nM
CCCC[C@H](CCN(O)C=O)C(=O)N[C@H](C(=O)N(C)C)C(C)(C)C CHEMBL93365 IC50 1000.0 nM