CN(C)C(=O)c1ccc(N(Cc2cc(Br)cs2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4591977 IC50 5.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(Br)s2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4551410 IC50 8.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(I)o2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4519504 IC50 11.0 nM
Cc1nc(N2C[C@@H](c3ccc(C(=O)O)[nH]3)C[C@H]2CO)c2c(n1)[nH]c1c(C3CC3)cccc12 CHEMBL5087040 IC50 12.2 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(Br)o2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4575355 IC50 13.0 nM
Cc1nc(N2C[C@@H](c3ccc(C(N)=O)[nH]3)C[C@H]2CO)c2c(n1)[nH]c1c(C3CC3)cccc12 CHEMBL5072731 IC50 17.8 nM
CN(C)C(=O)c1ccc(N(Cc2ncc(Br)s2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4461160 IC50 20.0 nM
Cc1cnc(Cl)nc1-c1ccc(N(Cc2ccc(CNC(=O)C(F)F)cc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL3727577 IC50 21.0 nM
Cc1nc2[nH]c3c(C4CC4)cccc3c2cc1-c1nnc(C(NC(=O)CCc2ccccc2)C(C)C)o1 CHEMBL5079107 IC50 24.1 nM
Cc1nc2[nH]c3c(C4CC4)cccc3c2cc1-c1nnc(C(CC(=O)NCc2ccccc2)C(C)C)o1 CHEMBL5087238 IC50 32.9 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(O)cc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4540811 IC50 34.0 nM
CC[C@@H]1C[C@H](c2ccc(C(=O)O)[nH]2)CN1c1nc(C)nc2[nH]c3c(C4CC4)cccc3c12 CHEMBL5089800 IC50 40.6 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(F)cc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4558944 IC50 52.0 nM
Cc1ccc(CN(C(=O)c2ccc(O)cc2O)c2ccc(C(=O)N(C)C)cc2)o1 CHEMBL4558837 IC50 52.0 nM
Cc1nc2[nH]c3c(C4CC4)cccc3c2cc1-c1nnc([C@@H](CC(=O)N[C@H](C)c2ccccc2)C(C)C)o1 CHEMBL5090085 IC50 61.5 nM
CN(C)C(=O)c1ccc(N(Cc2ccccc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL3729572 IC50 66.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccco2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4570690 IC50 69.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(Cl)o2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4587341 IC50 82.0 nM
O=C1c2ccccc2C(=O)c2c1cccc2-c1cnn(C2CCNCC2)c1 CHEMBL4471264 IC50 84.0 nM
CN(C)C(=O)c1ccc(N(Cc2cnc(Br)s2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4452536 IC50 87.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(C#N)s2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4513465 IC50 89.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc([N+](=O)[O-])cc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4539698 IC50 99.0 nM
CC(C(=O)O)n1cc(-c2cccc3c2C(=O)c2ccccc2C3(O)C(F)(F)F)cn1 CHEMBL4439097 IC50 143.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(Cl)cc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4534284 IC50 169.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc3ccccc3c2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4533214 IC50 234.0 nM
Cc1nc(N2C[C@@](Cc3ccccc3)(C(N)=O)C[C@H]2CO)c2c(n1)[nH]c1c(C3CC3)cccc12 CHEMBL5079949 IC50 260.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(C(F)(F)F)cc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4470843 IC50 273.0 nM
NC(=O)C[C@H](N)C(=O)N1CCC(Nc2ccc3c(c2)CN(S(=O)(=O)c2ccc(O)cc2O)C3)CC1 CHEMBL4103350 IC50 284.0 nM
CCCc1nnc(-c2cc3c(nc2C)[nH]c2c(C4CC4)cccc23)o1 CHEMBL5085080 IC50 292.0 nM
Cc1nc(N2C[C@](CO)(Cc3ccccc3)C[C@H]2CO)c2c(n1)[nH]c1c(C3CC3)cccc12 CHEMBL5092915 IC50 292.0 nM
CC(=O)Nc1ccc(CN(C(=O)c2ccc(O)cc2O)c2ccc(C(=O)N(C)C)cc2)cc1 CHEMBL4470078 IC50 311.0 nM
Cc1cnc(Cl)nc1-c1ccc(N(Cc2ccccc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL3732469 IC50 350.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(F)cc2)C(=O)c2ccc(O)cc2)cc1 CHEMBL4434941 IC50 390.0 nM
CN(C)C(=O)c1ccc(N(Cc2ccc(C#N)cc2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4561336 IC50 399.0 nM
Cc1nc2[nH]c3c(C4CC4)cccc3c2cc1-c1nnc(CC(C)C)o1 CHEMBL5080906 IC50 462.0 nM
Cc1nc2[nH]c3c(C4CC4)cccc3c2cc1-c1nnc(C(C)C(C)C)o1 CHEMBL5092147 IC50 494.0 nM
Cc1nc2[nH]c3c(C4CC4)cccc3c2cc1-c1nnc(C(C)C)o1 CHEMBL5071248 IC50 592.0 nM
CC(C)(C)OC(=O)N1CC=C(c2cccc3c2C(=O)c2ccccc2C3=O)CC1 CHEMBL4475200 IC50 600.0 nM
O=S(=O)(c1ccc(O)cc1O)N1Cc2cc(O)cc(O)c2C1 CHEMBL4082531 IC50 760.0 nM
CN(C)C(=O)c1ccc(N(CC2CCCCC2)C(=O)c2ccc(O)cc2O)cc1 CHEMBL4579724 IC50 775.0 nM