CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(C)(=O)=O)cccc2n1Cc1ccccc1 CHEMBL477548 IC50 7.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)O)cc3ccccc3c2n1Cc1ccccc1 CHEMBL514705 IC50 10.0 nM
Cc1ccccc1S(=O)(=O)NC(=O)COc1cccc2c1c(C(=O)C(N)=O)c(CC(C)C)n2Cc1ccccc1 CHEMBL514656 IC50 11.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccccc3Cl)cccc2n1Cc1ccccc1 CHEMBL474874 IC50 14.0 nM
CC(CC(=O)O)c1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)n1 CHEMBL4215835 IC50 14.0 nM
CCc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccccc3)cccc2n1Cc1ccccc1 CHEMBL514692 IC50 15.0 nM
C[C@@H](CC(=O)O)c1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)c1 CHEMBL4210991 IC50 15.0 nM
CCc1c(C(=O)C(N)=O)c2c(OCC(=O)O)cc3ccccc3c2n1Cc1ccccc1 CHEMBL515637 IC50 20.0 nM
CCc1c(C(=O)C(N)=O)c2c(OC(C)C(=O)O)cccc2n1Cc1ccccc1 CHEMBL148649 IC50 22.0 nM
NC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4171084 IC50 26.0 nM
NC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1cccc(CCC(=O)O)n1 CHEMBL4217510 IC50 29.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)C(F)(F)F)cccc2n1Cc1ccccc1 CHEMBL477549 IC50 30.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccccc3)cc3ccccc3c2n1Cc1ccccc1 CHEMBL506485 IC50 30.0 nM
CC(Cc1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)c1)C(=O)O CHEMBL4214052 IC50 32.0 nM
COC(Cc1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)c1)C(=O)O CHEMBL4204172 IC50 39.0 nM
CCc1c(C(=O)C(N)=O)c2c(OCC(=O)O)cccc2n1Cc1ccccc1 CHEMBL148674 IC50 41.0 nM
NC(=O)c1cc2ccc(C(F)(F)F)cc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4176544 IC50 43.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)O)cccc2n1Cc1ccccc1 CHEMBL504813 IC50 50.0 nM
CC(Cc1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)n1)C(=O)O CHEMBL4205511 IC50 65.0 nM
NC(=O)c1cc2ccc(OC(F)F)cc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4160483 IC50 68.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccccc3C(F)(F)F)cccc2n1Cc1ccccc1 CHEMBL477794 IC50 70.0 nM
CCc1c(C(=O)C(N)=O)c2c(OCC(=O)O)cc(C)cc2n1Cc1ccccc1 CHEMBL208315 IC50 75.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OC(C)C(=O)NS(=O)(=O)c3ccccc3)cccc2n1Cc1ccccc1 CHEMBL477156 IC50 80.0 nM
CCc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccccc3)cc3ccccc3c2n1Cc1ccccc1 CHEMBL446349 IC50 90.0 nM
NC(=O)c1cc2ccc(Cl)cc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4172222 IC50 90.0 nM
NC(=O)c1cc2ccc(OCC(F)(F)F)cc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4175583 IC50 93.0 nM
Cc1c(C(=O)C(N)=O)c2c(OCC(=O)O)cccn2c1Cc1ccccc1-c1ccccc1 CHEMBL5172164 IC50 100.0 nM
N#Cc1ccc2cc(C(N)=O)n(-c3cccc(CCC(=O)O)c3)c2c1 CHEMBL4174522 IC50 110.0 nM
NC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1cc(CCC(=O)O)ccn1 CHEMBL4213094 IC50 110.0 nM
CCCCCC/C=C/CC(=O)N[C@H](CSc1ccc(Cc2ccccc2)cc1)CC(=O)O CHEMBL152921 IC50 120.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3cccc(Cl)c3)cccc2n1Cc1ccccc1 CHEMBL477157 IC50 140.0 nM
CC(Cc1ccnc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)c1)C(=O)O CHEMBL4205008 IC50 140.0 nM
NC(=O)c1cc2ccc(C3CC3)cc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4173359 IC50 160.0 nM
CCc1ccc2cc(C(N)=O)n(-c3cccc(CCC(=O)O)c3)c2c1 CHEMBL4175643 IC50 170.0 nM
CCC(Cc1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)n1)C(=O)O CHEMBL4203027 IC50 170.0 nM
Cc1sc2ccccc2c1-c1cc(C(N)=O)n[nH]1 CHEMBL3337976 pIC50 173.78 nM
CCCCCCCCCCCC(=O)c1c(O)c(C(=O)CCCCCCCCCCC)c(O)c(C2CC(c3ccc(O)cc3)Oc3cc(O)ccc32)c1O CHEMBL444450 IC50 200.0 nM
C[C@H](CC(=O)O)c1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)c1 CHEMBL4207266 IC50 200.0 nM
Cc1ccc2cc(C(N)=O)n(-c3cccc(CCC(=O)O)c3)c2c1 CHEMBL4171797 IC50 230.0 nM
NC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1ccnc(CCC(=O)O)c1 CHEMBL4206163 IC50 240.0 nM
NC(=O)c1cc2ccc(F)cc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4161605 IC50 260.0 nM
NC(=O)c1ccc(Cc2ccccc2)cc1-c1cccc(CCC(=O)O)c1 CHEMBL4457557 IC50 280.0 nM
Cc1cc(-c2cc(C(N)=O)n[nH]2)c(C)s1 CHEMBL3337972 pIC50 316.23 nM
Cc1ccc(S(=O)(=O)NC(=O)COc2cccc3c2c(C(=O)C(N)=O)c(CC(C)C)n3Cc2ccccc2)cc1 CHEMBL475071 IC50 320.0 nM
CC(C)(Cc1cccc(-n2c(C(N)=O)cc3ccc(OC(F)(F)F)cc32)n1)C(=O)O CHEMBL4204160 IC50 320.0 nM
COc1cccc(/C=N/Nc2nc3ccccc3[nH]c2=O)c1 CHEMBL5194852 IC50 330.0 nM
Cc1sc(-c2ccccc2)cc1-c1cc(C(N)=O)n[nH]1 CHEMBL3337977 pIC50 346.74 nM
CCCCCC/C=C/CC(=O)N[C@@H](CCC(=O)O)CSc1ccc2ccccc2c1 CHEMBL152402 IC50 380.0 nM
NC(=O)c1cc(-c2cc(Cl)sc2Cl)[nH]n1 CHEMBL3337978 pIC50 398.11 nM
C[C@H](Cc1cccc(-c2cc(Cc3ccccc3)ccc2C(N)=O)c1)C(=O)O CHEMBL4593409 IC50 400.0 nM
NC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1ccc(CCC(=O)O)o1 CHEMBL4207065 IC50 430.0 nM
CCC(Cc1cccc(-c2cc(Cc3ccccc3)ccc2C(N)=O)c1)C(=O)O CHEMBL4533403 IC50 430.0 nM
CC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccc(Cl)cc3)cccc2n1Cc1ccccc1 CHEMBL514846 IC50 540.0 nM
NC(=O)c1ccc(Cc2ccccc2)cc1-c1cccc(CC(C(=O)O)C2CC2)c1 CHEMBL4453126 IC50 580.0 nM
O=c1[nH]c2ccccc2n2c(-c3ccc(O)cc3O)ccc12 CHEMBL5200953 IC50 610.0 nM
COc1ccc2cc(C(N)=O)n(-c3cccc(CCC(=O)O)c3)c2c1 CHEMBL4160502 IC50 620.0 nM
Cc1sccc1-c1cc(C(N)=O)n[nH]1 CHEMBL3337979 pIC50 630.96 nM
CC(Cc1cccc(-c2cc(Cc3ccccc3)ccc2C(N)=O)c1)C(=O)O CHEMBL4451830 IC50 750.0 nM
CCCCCC/C=C/CC(=O)N[C@H](CSc1ccc2ccccc2c1)CC(=O)O CHEMBL152031 IC50 790.0 nM
Cc1cccc2c1cc(C(N)=O)n2-c1cccc(CCC(=O)O)c1 CHEMBL4159939 IC50 830.0 nM
Cc1sc2ccccc2c1-c1cc(C(N)=O)nn1C CHEMBL3337982 pIC50 851.14 nM
Cc1cc(-c2cc(C(N)=O)nn2C)c(C)s1 CHEMBL3337983 pIC50 851.14 nM
CCCCCCCCCCCCCCCCCCOC(COCc1ccc(C#N)cc1)COc1ccc(Cc2noc(=O)[nH]2)cc1 CHEMBL223880 IC50 900.0 nM
NC(=O)c1cc2ccccc2n1-c1cccc(CCC(=O)O)c1 CHEMBL4176269 IC50 990.0 nM
COc1ccc2nc(Oc3ccccc3)cc(CC(N)=O)c2c1 CHEMBL43502 IC50 1000.0 nM
CCCCCCCCCCCCCCOC(COCCCCCCCCCC)COc1ccc(-c2noc(=O)[nH]2)cc1 CHEMBL220842 IC50 1000.0 nM