CCOC(=O)Sc1nc2cc(-n3nc(C(C)(C)C)sc3=O)c(F)cc2s1 CHEMBL1926835 Ki 40.0 nM
CCCOc1cc(N2CC3=C(CCCC3)C2=O)c(F)cc1Cl CHEMBL2252322 Ki 95.0 nM
C=CCOc1cc(N2CC3=C(CCCC3)C2=O)c(F)cc1Cl CHEMBL2252323 Ki 120.0 nM
CCOc1cc(N2CC3=C(CCCC3)C2=O)c(F)cc1Cl CHEMBL2252320 pKi 199.53 nM
CCOC(=O)Sc1nc2cc(-n3nc(C(C)(C)C)sc3=O)c(Cl)cc2s1 CHEMBL1926845 Ki 200.0 nM
CCOC(=O)CCSc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(Cl)cc2s1 CHEMBL1926967 Ki 250.0 nM
CCCOc1cc(N2CC3=C(CCCC3)C2=O)c(Cl)cc1Cl CHEMBL2252321 Ki 300.0 nM
CCOC(=O)CCSc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(F)cc2s1 CHEMBL1926960 Ki 320.0 nM
CCOC(=O)Sc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(Cl)cc2s1 CHEMBL1926963 Ki 330.0 nM
CCOC(=O)CSc1nc2cc(-n3nc(C(C)(C)C)sc3=O)c(F)cc2s1 CHEMBL1926837 Ki 340.0 nM
CCOC(=O)CCCSc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(F)cc2s1 CHEMBL1926961 Ki 360.0 nM
O=C1C2=C(CCCC2)C(O)N1c1cc(OCc2cccc(Cl)c2)c(Cl)cc1F CHEMBL2252326 pKi 524.81 nM
CCOc1cc(N2CC3=C(CCCC3)C2=O)c(Cl)cc1Cl CHEMBL2252319 Ki 670.0 nM
CC(C)Oc1cc(N2CC3=C(CCCC3)C2=O)c(F)cc1Cl CHEMBL2252347 Ki 690.0 nM
CCCOC(=O)CSc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(F)cc2s1 CHEMBL1926863 Ki 700.0 nM
CCOC(=O)Sc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(F)cc2s1 CHEMBL1926857 Ki 720.0 nM
Cc1nn(-c2cc(NS(C)(=O)=O)c(Cl)cc2Cl)c(=O)n1C(F)F CHEMBL1884669 Ki 720.0 nM
COC(=O)Sc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(F)cc2s1 CHEMBL2230219 Ki 720.0 nM
O=C1C2=C(CCCC2)C(O)N1c1cc(OCc2cccc(F)c2)c(Cl)cc1F CHEMBL2252325 pKi 776.25 nM
CC(C)(C)OC(=O)CSc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(Cl)cc2s1 CHEMBL2230215 pKi 831.76 nM
CCCOC(=O)CSc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(Cl)cc2s1 CHEMBL2230211 pKi 977.24 nM
CCOC(=O)CSc1nc2cc(-n3nc(C(C)(C)C)oc3=O)c(Cl)cc2s1 CHEMBL1926964 pKi 1000.0 nM
