Cc1ccc(S(=O)(=O)c2ccc(N)cc2C(F)(F)F)cc1-c1cnc(N)nc1 CHEMBL5404826 IC90 21.0 nM
Cc1cc(C(N)=O)cc(S(=O)(=O)c2ccc(C)c(-c3cnc(N)nc3)c2)c1 CHEMBL5403474 IC90 29.0 nM
Cc1ccc(S(=O)(=O)c2ccc3c(c2)CCN3)cc1-c1cnc(N)nc1 CHEMBL5412567 IC90 30.0 nM
CCNc1ccc(S(=O)(=O)c2ccc(C)c(-c3cnc(N)nc3)c2)c(C(F)(F)F)c1 CHEMBL5432144 IC90 31.0 nM
Cc1ccc(NS(=O)(=O)c2ccc3c(c2)CCN3)cc1-c1cnc(N)nc1 CHEMBL5415515 IC90 33.0 nM
Cc1ccc(S(=O)(=O)c2ccc3c(c2)CCN3)cc1-c1cnc2n[nH]cc2c1 CHEMBL5401390 IC90 40.0 nM
Cc1cc2c(cc1-c1cnc(N)nc1)S(=O)(=O)c1ccc(C(N)=O)cc1CC2C CHEMBL5431667 IC90 40.0 nM
Cc1ccc(S(=O)(=O)c2ccc3c(c2)CCNC3=O)cc1-c1cnc(N)nc1 CHEMBL5425702 IC90 40.0 nM
Cc1cc(S(=O)(=O)Nc2ccc(C)c(-c3cnc(N)nc3)c2)ccc1N CHEMBL5394091 IC90 70.0 nM
Nc1ccc(S(=O)(=O)c2cccc(-c3cnc(N)nc3)c2)c(C(F)(F)F)c1 CHEMBL5428765 IC90 131.0 nM
Cc1cc(S(=O)(=O)c2ccc(C)c(-c3cnc(N)nc3)c2)ccc1C(N)=O CHEMBL5403999 IC90 155.0 nM
Cc1ccc(S(=O)(=O)c2ccc3c(c2)CCO3)cc1-c1cnc(N)nc1 CHEMBL5438772 IC90 160.0 nM
Cc1cc(S(=O)(=O)c2ccc(C)c(-c3cnc(N)nc3)c2)ccc1N CHEMBL5405983 IC90 169.0 nM
NC(=O)c1ccc(-c2ccc(-c3ccc4c(c3)COC4=O)s2)cc1 CHEMBL3754633 IC50 180.0 nM
Cc1ccc(S(=O)(=O)c2ccc3c(c2)CNC3=O)cc1-c1cnc(N)nc1 CHEMBL5415901 IC90 199.0 nM
Cc1cc(S(=O)(=O)c2ccc(C)c(-c3cnc(N)nc3)c2)c(C(F)(F)F)cc1N CHEMBL5414566 IC90 203.0 nM
Cc1ccc(S(=O)(=O)c2ccc3[nH]ncc3c2)cc1-c1cnc(N)nc1 CHEMBL5408863 IC90 281.0 nM
O=C1NC(=S)N/C1=C/c1csc(-c2ccc3c(c2)COC3=O)n1 CHEMBL1934375 IC50 340.0 nM
O=C1NC(=S)N/C1=C/c1cc2ccc(-c3ccc4c(c3)COC4=O)cc2s1 CHEMBL1934381 IC50 360.0 nM
O=C1NC(=S)N/C1=C/c1cc2ccc(-c3ccc4c(c3)COC4=O)cc2[nH]1 CHEMBL1934383 IC50 360.0 nM
Cc1ccc(S(=O)(=O)c2ccc3c(c2)CCN3)cc1-c1ccc(N)nc1 CHEMBL5435628 IC90 361.0 nM
O=C1NC(=S)N/C1=C/c1ccc(-c2ccc3c(c2)COC3=O)cn1 CHEMBL1934370 IC50 370.0 nM
O=C1NC(=S)NC(=O)C1=Cc1ccc(-c2ccc3c(c2)COC3=O)s1 CHEMBL1934397 IC50 400.0 nM
O=C1NC(=O)/C(=C\c2ccc(-c3ccc4c(c3)CNC4=O)s2)N1 CHEMBL3103651 IC50 400.0 nM
Cc1ccc(S(=O)(=O)c2ccc3c(c2)CCN3C)cc1-c1cnc(N)nc1 CHEMBL5400754 IC90 406.0 nM
O=C1NC(=S)N/C1=C/c1ccc2cc(-c3ccc4c(c3)COC4=O)ccc2n1 CHEMBL1934386 IC50 470.0 nM
O=C1NC(=S)N/C1=C/c1cc2cc(-c3ccc4c(c3)COC4=O)ccc2s1 CHEMBL1934380 IC50 490.0 nM
Cc1ccc(S(=O)(=O)c2ccc3[nH]ccc3c2)cc1-c1cnc(N)nc1 CHEMBL5403471 IC90 496.0 nM
O=C1NC(=S)N/C1=C/c1cc2cc(-c3ccc4c(c3)COC4=O)ccc2o1 CHEMBL1934382 IC50 510.0 nM
CN1Cc2cc(-c3ccc(/C=C4/NC(=S)NC4=O)s3)ccc2C1=O CHEMBL3103907 IC50 510.0 nM
O=C1NC(=S)N/C1=C/c1ccc(-c2ccc3c(c2)CN(CCCO)C3=O)s1 CHEMBL3103914 IC50 530.0 nM
CCOC(=O)N1Cc2cc(-c3ccc(/C=C4/NC(=S)NC4=O)s3)ccc2C1=O CHEMBL3103917 IC50 550.0 nM
CCN1Cc2cc(-c3ccc(/C=C4/NC(=S)NC4=O)s3)ccc2C1=O CHEMBL3103908 IC50 600.0 nM
O=C1NC(=S)N/C1=C/c1ccc(-c2ccc3c(c2)CNC3=O)cn1 CHEMBL3103655 IC50 630.0 nM
O=C1NC(=S)N/C1=C/c1ccc(-c2ccc3c(c2)C(=O)NCC3)s1 CHEMBL3103647 IC50 640.0 nM
NC(=O)c1ccc(-c2ccc(-c3ccc4c(c3)COC4=O)s2)cc1O CHEMBL3754407 IC50 670.0 nM
CN1Cc2cc(-c3ccc(-c4cncc(NS(=O)(=O)c5ccc(C(=O)O)cc5)c4)s3)ccc2C1=O CHEMBL4169732 IC50 750.0 nM
CN1Cc2cc(-c3ccc(-c4cncc(NS(=O)(=O)c5ccccc5[N+](=O)[O-])c4)s3)ccc2C1=O CHEMBL4174219 IC90 770.0 nM
O=C1NC(=S)N/C1=C/c1ccc(-c2ccc3c(c2)COC3=O)s1 CHEMBL1934364 IC50 780.0 nM
O=C1NC(=S)N/C1=C/c1ccc(-c2ccc3c(c2)CN(CCO)C3=O)s1 CHEMBL3103913 IC50 780.0 nM
COc1ncc(-c2ccc(-c3cnc4c(c3)CN(C)C4=O)s2)cc1NS(=O)(=O)c1ccccc1C(F)(F)F CHEMBL4453871 IC50 780.0 nM
NC(=O)c1cccc(-c2ccc(/C=C3/NC(=S)NC3=O)s2)c1 CHEMBL3102870 IC50 790.0 nM
O=C1NC(=O)C(=Cc2ccc(-c3ccc4c(c3)COC4=O)s2)C(=O)N1 CHEMBL1934396 IC50 800.0 nM
O=C1NC(=S)N/C1=C/c1cc2cc(-c3ccc4c(c3)COC4=O)ccc2[nH]1 CHEMBL1934384 IC50 820.0 nM
O=C1OCc2cc(-c3ccc(-c4ccc(CO)cc4)s3)ccc21 CHEMBL3753587 IC50 900.0 nM
NC(=O)c1ccc(-c2ccc(-c3ccc4c(c3)COC4=O)s2)cn1 CHEMBL3753271 IC50 920.0 nM
CC(=O)N1Cc2cc(-c3ccc(/C=C4/NC(=S)NC4=O)s3)ccc2C1=O CHEMBL3103916 IC50 930.0 nM
Cc1cc2c(c(=S)[nH]1)C(=O)O/C2=C\c1csc2ccccc12 CHEMBL463187 IC50 970.0 nM