O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2cc(Oc3ccccc3)ccc2F)N1CC1CC1 CHEMBL5413526 IC50 50.0 nM
CCCCCCc1ccc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)cc1 CHEMBL5399303 IC50 54.0 nM
O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2ccc(Oc3ccc(Cl)cc3)cc2)N1CC1CC1 CHEMBL5410458 IC50 60.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(F)c(OC(F)(F)F)c2)cc1 CHEMBL5422228 IC50 73.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Cl)c(C2CC2)c1 CHEMBL5402465 IC50 92.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1cccc(Oc2ccc(F)cc2)c1 CHEMBL5415049 IC50 98.0 nM
Cc1cc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)cc(C)c1Cl CHEMBL5438925 IC50 100.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cc(F)cc4[nH]c(=O)oc34)c2C1c1cccc(Oc2ccc(F)cc2)c1 CHEMBL5420148 IC50 100.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Sc2ccc(OC(F)(F)F)cc2)cc1 CHEMBL5418974 IC50 110.0 nM
CCc1cc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)ccc1Cl CHEMBL5400683 IC50 120.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(C(F)(F)F)cc2)cc1 CHEMBL5411892 IC50 120.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)cc2Cl)cc1 CHEMBL5407874 IC50 120.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1cccc(Oc2ccc(C(F)(F)F)cc2C(F)(F)F)c1 CHEMBL5421014 IC50 120.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(Cl)cc2)cc1 CHEMBL5425260 IC50 130.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(Cl)cc2)cc1F CHEMBL5422282 IC50 130.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1Cl CHEMBL5415916 IC50 130.0 nM
Cc1cc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)ccc1OCCCC(F)(F)F CHEMBL5428926 IC50 140.0 nM
CCCCc1cccc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)c1 CHEMBL5408562 IC50 140.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2cc(Cl)cc(C(F)(F)F)c2)cc1 CHEMBL5398843 IC50 140.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(Cl)c(Cl)c2)cc1 CHEMBL5411035 IC50 140.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc3onc(C(F)(F)F)c3c2)cc1 CHEMBL5415508 IC50 140.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Cl)cc1 CHEMBL5429708 IC50 150.0 nM
Cc1cc(OC(F)(F)F)ccc1Oc1ccc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)cc1 CHEMBL5397090 IC50 150.0 nM
Cc1cc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)c(F)cc1Oc1ccc(OC(F)(F)F)cc1 CHEMBL5398412 IC50 150.0 nM
Cc1cc(Oc2ccc(C3c4c(-c5cccc6[nH]c(=O)oc56)n[nH]c4C(=O)N3CC(C)(F)F)cc2)ccc1OC(F)(F)F CHEMBL5426513 IC50 160.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1cccc(Oc2ccc(OC(F)(F)F)cc2)c1 CHEMBL5422254 IC50 160.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2cc(Cl)cc(OC(F)(F)F)c2)cc1 CHEMBL5411302 IC50 170.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2cccc(Cl)c2OC(F)(F)F)cc1 CHEMBL5439463 IC50 170.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(Cl)cc2)c(Cl)c1 CHEMBL5410235 IC50 170.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(CC(F)(F)F)cc2)cc1 CHEMBL5398791 IC50 170.0 nM
O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2cc(Oc3ccccc3)ccc2F)N1CC(F)(F)F CHEMBL5437469 IC50 180.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(C(F)(F)F)cc2C(F)(F)F)cc1 CHEMBL5405342 IC50 180.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(SC(F)(F)F)cc2)cc1 CHEMBL5408029 IC50 180.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)c(Cl)c2)cc1F CHEMBL5422061 IC50 180.0 nM
Cc1cc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)ccc1Oc1ccc(OC(F)(F)F)cc1 CHEMBL5416880 IC50 180.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(C(F)(F)c2ccccc2)cc1 CHEMBL5394161 IC50 180.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)c(F)c2)cc1 CHEMBL5397515 IC50 190.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1cc(Oc2ccc(F)cc2)cc(C(F)(F)F)c1 CHEMBL5424317 IC50 190.0 nM
Cc1cc(Oc2ccc(OC(F)(F)F)c(Cl)c2)ccc1C1c2c(-c3cccc4[nH]c(=O)oc34)n[nH]c2C(=O)N1CC(C)(F)F CHEMBL5415979 IC50 200.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 CHEMBL5303480 IC50 200.0 nM
Cc1cc(Oc2ccc(C3c4c(-c5cccc6[nH]c(=O)oc56)n[nH]c4C(=O)N3CC(C)(F)F)cc2)cc(C(F)(F)F)c1 CHEMBL5432794 IC50 200.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1F CHEMBL5397308 IC50 210.0 nM
Cc1cc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)ccc1Oc1ccc(OC(F)(F)F)c(Cl)c1 CHEMBL5423868 IC50 230.0 nM
O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2ccc(-c3ccccc3F)cc2)N1CC1CC1 CHEMBL5409665 IC50 240.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc3c(c2)OC(F)(F)C(F)(F)O3)cc1 CHEMBL5401071 IC50 240.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cc(F)cc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(Cl)cc2)cc1 CHEMBL5406702 IC50 240.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(C(F)(F)F)c(C(F)(F)F)c2)cc1 CHEMBL5418646 IC50 250.0 nM
C[C@@H](Oc1ccc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)cc1)c1ccccc1 CHEMBL5423038 IC50 250.0 nM
COC(c1ccccc1)c1ccc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)cc1 CHEMBL5433712 IC50 250.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)sc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1 CHEMBL5427315 IC50 250.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1 CHEMBL5416353 IC50 260.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)cc2)c(OCCCC(F)(F)F)c1 CHEMBL5421968 IC50 280.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1F CHEMBL5423904 IC50 290.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)[nH]c34)c2C1c1ccc(Oc2ccc(Cl)cc2)cc1 CHEMBL5420756 IC50 300.0 nM
O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2cccc(Oc3ccc(Cl)cn3)c2)N1CC1CC1 CHEMBL5406964 IC50 310.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)c(Cl)c2)c(OC(F)(F)F)c1 CHEMBL5427616 IC50 330.0 nM
CC(=O)Nc1cccc(-c2n[nH]c3c2C(c2cc(Oc4ccccc4)ccc2F)N(CC(F)(F)F)C3=O)c1 CHEMBL5439213 IC50 340.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(OC(F)(F)F)cc1 CHEMBL5422619 IC50 340.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)c(Cl)c2)cc1 CHEMBL5406141 IC50 340.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(OCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 CHEMBL5410181 IC50 340.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2cc(Cl)c(OC(F)(F)F)c(Cl)c2)cc1 CHEMBL5406855 IC50 360.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(S(=O)(=O)C(F)(F)F)cc2)cc1 CHEMBL5414041 IC50 360.0 nM
O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2cccc(OC3CCC3)c2)N1CC1CC1 CHEMBL5403205 IC50 370.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)c(Cl)c2)c(C(F)(F)F)c1 CHEMBL5424109 IC50 390.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc(NC=O)c3)c2C1c1ccc(Cl)cc1 CHEMBL5432741 IC50 420.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)c(C(F)(F)F)c2)cc1 CHEMBL5431685 IC50 430.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1cnc(Oc2ccc(Cl)c(Cl)c2)s1 CHEMBL5393837 IC50 430.0 nM
O=C1c2[nH]nc(-c3ccc(F)c4[nH]c(=O)oc34)c2C(c2cc(Oc3ccccc3)ccc2F)N1CC(F)(F)F CHEMBL5438690 IC50 460.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2cc(C(F)(F)F)cc(Cl)n2)cc1 CHEMBL5436462 IC50 500.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(Cl)cc2)cn1 CHEMBL5413159 IC50 510.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2ccc(OC(F)(F)F)c(Cl)c2)c(OCCCC(F)(F)F)c1 CHEMBL5403365 IC50 530.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Oc2nc(C(F)(F)F)cs2)cc1 CHEMBL5394071 IC50 540.0 nM
CCC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(F)cc1 CHEMBL5394551 IC50 570.0 nM
Cc1cc(C2c3c(-c4cccc5[nH]c(=O)oc45)n[nH]c3C(=O)N2CC(C)(F)F)c(F)cc1Oc1cc(C(F)(F)F)cc(C(F)(F)F)c1 CHEMBL5429973 IC50 600.0 nM
O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2cccc(Oc3ccccc3)c2)N1Cc1ncco1 CHEMBL5418458 IC50 620.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(CN2CCC(F)(F)CC2)cc1 CHEMBL5434523 IC50 650.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(Cl)cc1Oc1ccccc1 CHEMBL5417908 IC50 660.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1cccc(Nc2ccccc2)c1 CHEMBL5411470 IC50 760.0 nM
O=C1c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C(c2ccc(Oc3ccccc3)nc2)N1CC1CC1 CHEMBL5416242 IC50 770.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc2c(cnn2-c2ccccc2)c1 CHEMBL5412308 IC50 780.0 nM
O=C1c2[nH]nc(-c3cc(Oc4ccccc4)cc4[nH]c(=O)oc34)c2C(c2ccc(F)cc2)N1CC(F)(F)F CHEMBL5408184 IC50 830.0 nM
CCN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1ccc(F)cc1 CHEMBL5396446 IC50 920.0 nM
CC(F)(F)CN1C(=O)c2[nH]nc(-c3cccc4[nH]c(=O)oc34)c2C1c1cnc(C(F)(F)F)s1 CHEMBL5424593 IC50 1000.0 nM