Cc1ccccc1-c1ccc(-c2ccc3c(c2)c(C)c(CC(C)(C)C(=O)O)n3Cc2ccc(Cl)cc2)cc1F CHEMBL180650 IC50 3.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccc(-c4ccccc4Cl)c(F)c3)cc12 CHEMBL180617 IC50 4.0 nM
COc1ccccc1-c1ccc(-c2ccc3c(c2)c(C)c(CC(C)(C)C(=O)O)n3Cc2ccc(Cl)cc2)cc1F CHEMBL369525 IC50 5.0 nM
CC(=O)c1ccccc1-c1ccc(-c2ccc3c(c2)c(C)c(CC(C)(C)C(=O)O)n3Cc2ccc(Cl)cc2)cc1F CHEMBL368241 IC50 6.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccc(-c4ccccc4)c(F)c3)cc12 CHEMBL182032 IC50 7.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccc(-c4ccccc4F)c(F)c3)cc12 CHEMBL362836 IC50 8.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccc(-c4cccnc4)c(F)c3)cc12 CHEMBL181728 IC50 12.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccc(-c4ccccc4)cc3)cc12 CHEMBL362242 IC50 16.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccc(-c4ccccc4)c(Cl)c3)cc12 CHEMBL362675 IC50 22.0 nM
COc1ncc(-c2cccc(S(=O)(=O)Nc3ccccc3S(N)(=O)=O)c2)cc1Cl CHEMBL3962955 IC50 22.0 nM
Cc1ccc(-c2ccc(-c3ccc4c(c3)c(C)c(CC(C)(C)C(=O)O)n4Cc3ccc(Cl)cc3)cc2F)cc1 CHEMBL183596 IC50 31.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(C#Cc2ccc(C(F)(F)F)cc2)nc1 CHEMBL3986331 IC50 31.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccc(-c4cnccn4)c(F)c3)cc12 CHEMBL181792 IC50 32.0 nM
Cc1cccc(-c2ccc(-c3ccc4c(c3)c(C)c(CC(C)(C)C(=O)O)n4Cc3ccc(Cl)cc3)cc2F)c1 CHEMBL183878 IC50 33.0 nM
COc1cc(Cl)ccc1/C=C/S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3904203 IC50 36.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc(-c2cc3ccccc3o2)cc1 CHEMBL3897379 IC50 40.0 nM
NS(=O)(=O)c1cc(CO)ccc1NS(=O)(=O)CCc1ccc(C#CC2CCCC2)cc1 CHEMBL3961959 IC50 41.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(-c2ccco2)cc1 CHEMBL3943504 IC50 44.0 nM
CC(C)(C)C#Cc1ccc(/C=C/S(=O)(=O)Nc2ccccc2S(N)(=O)=O)cc1 CHEMBL3943346 IC50 55.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(-c2ccco2)cc1 CHEMBL3965498 IC50 57.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(-c2cc3ccccc3o2)cc1 CHEMBL3968523 IC50 74.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(Br)cc1 CHEMBL3966442 IC50 74.0 nM
CC(C)(C)C#Cc1ccc(CCS(=O)(=O)Nc2ccc(CO)cc2S(N)(=O)=O)cc1 CHEMBL3930981 IC50 75.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(Cl)c(Cl)c1 CHEMBL3942994 IC50 77.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1ccc(-c2cc3ccccc3o2)cc1 CHEMBL3898952 IC50 79.0 nM
CC(C)(C)C#Cc1ccc(CCS(=O)(=O)Nc2ccccc2S(N)(=O)=O)cc1 CHEMBL3935976 IC50 81.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1ccc(-c2ccccc2)cc1 CHEMBL3951095 IC50 84.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc2ccccc2c1 CHEMBL3957120 IC50 91.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(C2=CCCC2)cc1 CHEMBL3918947 IC50 97.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(-c2ccc(C(F)(F)F)cc2)cc1 CHEMBL3946465 IC50 100.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(OC(F)F)cc1 CHEMBL3908925 IC50 110.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccccc1OC(F)F CHEMBL3941676 IC50 110.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc(-c2ccco2)cc1 CHEMBL3889985 IC50 120.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(-c2cc3ccccc3o2)cc1 CHEMBL3959989 IC50 130.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(-c2ccccc2)cc1 CHEMBL3907650 IC50 130.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(OC(F)(F)C(F)F)cc1 CHEMBL3975393 IC50 130.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1cc(Cl)ccc1S(N)(=O)=O CHEMBL3903992 IC50 130.0 nM
NS(=O)(=O)c1ccc(Cl)cc1NS(=O)(=O)CCc1ccc(Cl)c(Cl)c1 CHEMBL3951825 IC50 130.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(-c2cc3ccccc3o2)cc1 CHEMBL3906349 IC50 140.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(Br)cc1 CHEMBL3943912 IC50 140.0 nM
NS(=O)(=O)c1cc(Cl)c(F)cc1NS(=O)(=O)CCc1ccc(Cl)c(Cl)c1 CHEMBL3911159 IC50 150.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3cccc(-c4ccccc4)c3)cc12 CHEMBL180846 IC50 160.0 nM
CSc1ccc(/C=C/S(=O)(=O)Nc2cc(F)ccc2S(N)(=O)=O)cc1 CHEMBL3960265 IC50 160.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc(-c2ccccc2)cc1 CHEMBL3891144 IC50 160.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1ccc(-c2ccco2)cc1 CHEMBL3960306 IC50 170.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(-c2ccc(C(F)(F)F)cc2)cc1 CHEMBL3913683 IC50 180.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(-c2ccco2)cc1 CHEMBL3968505 IC50 190.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc2ccccc2c1 CHEMBL3928194 IC50 190.0 nM
COc1ncc(-c2cccc(S(=O)(=O)Nc3ccccc3S(N)(=O)=O)c2)cc1F CHEMBL3923779 IC50 190.0 nM
CSc1ccc(/C=C/S(=O)(=O)Nc2ccc(F)cc2S(N)(=O)=O)cc1 CHEMBL3977611 IC50 220.0 nM
CC(C)(C)c1ccc(CCS(=O)(=O)Nc2ccccc2S(N)(=O)=O)cc1 CHEMBL3926649 IC50 220.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(-c2cccc(OC(F)(F)F)c2)c1 CHEMBL3911878 IC50 220.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(-c2ccc(Cl)c(Cl)c2)c1 CHEMBL3932675 IC50 220.0 nM
CC(C)(O)C#Cc1ccc(/C=C/S(=O)(=O)Nc2ccccc2S(N)(=O)=O)cc1 CHEMBL3906406 IC50 220.0 nM
CC(C)c1ccc2c(c1)c(C(=O)CC(C)(C)C)c(CC(C)(C)C(=O)O)n2Cc1ccc(Cl)cc1 CHEMBL181236 IC50 250.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3958446 IC50 250.0 nM
CC(C)c1ccc2c(c1)c(C(=O)CSC(C)(C)C)c(CC(C)(C)C(=O)O)n2Cc1ccc(Cl)cc1 CHEMBL426054 IC50 260.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(C2Cc3ccccc3O2)cc1 CHEMBL3956630 IC50 270.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc(Cl)c(Cl)c1 CHEMBL3961503 IC50 270.0 nM
COc1ccc(Br)cc1/C=C/S(=O)(=O)Nc1ccc(F)cc1S(N)(=O)=O CHEMBL3948341 IC50 270.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1cccc(C(F)(F)F)c1 CHEMBL3919221 IC50 270.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(C2CCCC2)cc1 CHEMBL3957650 IC50 270.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(C#CC2CCCCC2)nc1 CHEMBL3958405 IC50 270.0 nM
CSc1ccccc1/C=C/S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3926208 IC50 270.0 nM
CC(Cc1ccc(Cl)cc1)S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3920820 IC50 280.0 nM
COc1ccc(Br)cc1/C=C/S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3957007 IC50 280.0 nM
CC(C)c1ccc2c(c1)c(Cc1ccc(C(C)(C)C)cc1)c(CC(C)(C)C(=O)O)n2Cc1ccc(Cl)cc1 CHEMBL360742 IC50 290.0 nM
COc1ccc(Br)cc1/C=C/S(=O)(=O)Nc1cccc(F)c1S(N)(=O)=O CHEMBL3920537 IC50 290.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(Cl)cc1 CHEMBL3962498 IC50 290.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1ccc2ccccc2c1 CHEMBL3950093 IC50 290.0 nM
CN(C)c1ccc(-c2cccc(S(=O)(=O)Nc3ccccc3S(N)(=O)=O)c2)cn1 CHEMBL3890428 IC50 290.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1cc(F)cc(F)c1S(N)(=O)=O CHEMBL3967203 IC50 290.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1ccc(Cl)c(Cl)c1 CHEMBL3891610 IC50 300.0 nM
COc1ccccc1/C=C/S(=O)(=O)Nc1cc(F)ccc1S(N)(=O)=O CHEMBL3964934 IC50 300.0 nM
CC(C)(C)c1ccc(CCS(=O)(=O)Nc2cc(F)ccc2S(N)(=O)=O)cc1 CHEMBL3972879 IC50 300.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(Br)cc1 CHEMBL3891513 IC50 310.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc(Br)cc1 CHEMBL3900511 IC50 310.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)CCc1ccc(Cl)cc1 CHEMBL3922244 IC50 320.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(C(C)(C)C)cc12 CHEMBL182092 IC50 330.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1ccc(CO)cc1S(N)(=O)=O CHEMBL3899058 IC50 330.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc(Cl)cc1 CHEMBL3974448 IC50 350.0 nM
COc1ccccc1/C=C/S(=O)(=O)Nc1ccc(F)cc1S(N)(=O)=O CHEMBL3896616 IC50 360.0 nM
Cc1ccc(NS(=O)(=O)CCc2ccc(C#CC(C)(C)C)cc2)c(S(N)(=O)=O)c1 CHEMBL3934373 IC50 360.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1cc(C#N)ccc1S(N)(=O)=O CHEMBL3956021 IC50 370.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1F CHEMBL3957390 IC50 380.0 nM
CCOc1ccccc1/C=C/S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3932789 IC50 380.0 nM
COc1ccc(Br)cc1/C=C/S(=O)(=O)Nc1cc(F)ccc1S(N)(=O)=O CHEMBL3911599 IC50 420.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccccc1OC(F)(F)F CHEMBL3960258 IC50 420.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(OC(F)(F)C(F)F)cc1 CHEMBL3918599 IC50 420.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1ccc(Cl)cc1 CHEMBL3960671 IC50 430.0 nM
COc1ccccc1/C=C/S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3955177 IC50 430.0 nM
CC(Cc1ccc(Cl)cc1)S(=O)(=O)Nc1cc(F)ccc1S(N)(=O)=O CHEMBL3981844 IC50 450.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(OCc2cnc(Cl)s2)cc1 CHEMBL3936811 IC50 460.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(-c2cccc(Cl)c2Cl)c1 CHEMBL3957896 IC50 480.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc(Cl)cc1 CHEMBL3943328 IC50 490.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)CCc1ccc2ccccc2c1 CHEMBL3979799 IC50 490.0 nM
C/C(=C\c1ccc(Cl)cc1)S(=O)(=O)Nc1cccc(F)c1S(N)(=O)=O CHEMBL3937378 IC50 520.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1ccc(C#N)cc1S(N)(=O)=O CHEMBL3965135 IC50 520.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1cccc(Cl)c1 CHEMBL3899994 IC50 530.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1ccc(C)cc1S(N)(=O)=O CHEMBL3960851 IC50 560.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(Cl)cc1 CHEMBL3965953 IC50 570.0 nM
COc1ccc(-c2cccc(S(=O)(=O)Nc3ccccc3S(N)(=O)=O)c2)cn1 CHEMBL3942873 IC50 570.0 nM
C/C(=C\c1ccc(Cl)cc1)S(=O)(=O)Nc1cc(F)ccc1S(N)(=O)=O CHEMBL3914128 IC50 590.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccccc1Cl CHEMBL3979943 IC50 590.0 nM
Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(-c3ccccc3)cc12 CHEMBL181836 IC50 600.0 nM
C/C(=C\c1ccc(Cl)cc1)S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3926129 IC50 610.0 nM
COc1ccccc1/C=C/S(=O)(=O)Nc1cccc(F)c1S(N)(=O)=O CHEMBL3976177 IC50 620.0 nM
NS(=O)(=O)c1cnccc1NS(=O)(=O)CCc1ccc(-c2cc3ccccc3o2)cc1 CHEMBL3928928 IC50 620.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(-c2cncc(Cl)c2)c1 CHEMBL3979763 IC50 630.0 nM
NS(=O)(=O)c1c(F)cc(F)cc1NS(=O)(=O)CCc1ccc(Cl)c(Cl)c1 CHEMBL3895929 IC50 640.0 nM
CC(C)c1ccc2c(c1)c(Oc1ccccc1)c(CC(C)(C)C(=O)O)n2Cc1ccc(Cl)cc1 CHEMBL182153 IC50 650.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccccc1C(F)(F)F CHEMBL3958782 IC50 650.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)/C=C/c1ccc(C(F)(F)F)cc1 CHEMBL3889743 IC50 650.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl CHEMBL3920921 IC50 650.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(C(F)(F)F)cc1 CHEMBL3985648 IC50 670.0 nM
Cc1ccc(NS(=O)(=O)/C=C/c2ccc(Br)cc2)c(S(N)(=O)=O)c1 CHEMBL3902095 IC50 680.0 nM
CC(C)(C)C#Cc1ccc(CCS(=O)(=O)Nc2ccccc2S(N)(=O)=O)cn1 CHEMBL3909647 IC50 680.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)/C=C/c1ccc(OC(F)F)cc1 CHEMBL3952218 IC50 700.0 nM
C/C(=C\S(=O)(=O)Nc1ccccc1S(N)(=O)=O)c1ccc(Cl)cc1 CHEMBL3890439 IC50 700.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1cc(C)ccc1S(N)(=O)=O CHEMBL3917419 IC50 720.0 nM
COc1ncc(-c2cccc(S(=O)(=O)Nc3ccsc3S(N)(=O)=O)c2)cc1Cl CHEMBL3936192 IC50 740.0 nM
NS(=O)(=O)c1cc(CO)ccc1NS(=O)(=O)CCc1ccc(Cl)cc1 CHEMBL3973991 IC50 750.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)CCc1ccc2ccccc2c1 CHEMBL3934319 IC50 760.0 nM
NS(=O)(=O)c1ccc(F)cc1NS(=O)(=O)CCc1ccc(Cl)cc1 CHEMBL3955098 IC50 800.0 nM
NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(-c2cc(F)cc(F)c2)c1 CHEMBL3972092 IC50 830.0 nM
NS(=O)(=O)c1cc(F)ccc1NS(=O)(=O)/C=C/c1ccc(Br)cc1 CHEMBL3964770 IC50 850.0 nM
NS(=O)(=O)c1c(F)cccc1NS(=O)(=O)/C=C/c1ccc(C(F)(F)F)cc1 CHEMBL3933010 IC50 870.0 nM
NS(=O)(=O)c1cc(Cl)c(F)cc1NS(=O)(=O)CCc1ccc(Cl)cc1 CHEMBL3980697 IC50 870.0 nM
Cc1ccccc1C(=O)c1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(C(C)C)cc12 CHEMBL360114 IC50 900.0 nM
Cc1cc(NC(=O)Nc2ccc(Cl)cc2)ccc1S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3920223 IC50 900.0 nM
CC(C)Oc1ccccc1/C=C/S(=O)(=O)Nc1ccccc1S(N)(=O)=O CHEMBL3950393 IC50 950.0 nM
C/C(=C\c1ccc(Cl)cc1)S(=O)(=O)Nc1ccc(F)cc1S(N)(=O)=O CHEMBL3910817 IC50 1000.0 nM
COc1cc(Cl)ccc1CCS(=O)(=O)Nc1ccc(Cl)cc1S(N)(=O)=O CHEMBL3950804 IC50 1000.0 nM