CC1(C)Cc2c(sc(NC(=S)NC(=O)c3ccccc3)c2C(=O)O)CO1 CHEMBL1328505 EC50 22.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)c3cccs3)c2C(=O)O)CO1 CHEMBL4097338 EC50 25.0 nM
Nc1nc2c(ncn2[C@@H]2O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2O)c(=O)[nH]1 CHEMBL384759 Kd 25.83 nM
O=C(NC(=S)Nc1sc2c(c1C(=O)O)CC1(CCCC1)OC2)c1ccccc1 CHEMBL4098837 EC50 33.0 nM
CCC1(C)Cc2c(sc(NC(=S)NC(=O)c3ccccc3)c2C(=O)O)CO1 CHEMBL4080794 EC50 35.0 nM
CC1(C)CCc2sc(NC(=S)NC(=O)c3ccccc3)c(C(=O)O)c2C1 CHEMBL4091094 EC50 63.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)c3ccco3)c2C(=O)O)CO1 CHEMBL4068483 EC50 74.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)c3ccc(F)cc3)c2C(=O)O)CO1 CHEMBL4069652 EC50 77.0 nM
Nc1nc2c(ncn2[C@@H]2O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2O)c(=O)[nH]1 CHEMBL1233147 Kd 78.14 nM
Cc1ccc(C(=O)NC(=S)Nc2sc3c(c2C(=O)O)CC(C)(C)OC3)cc1 CHEMBL4089622 EC50 97.0 nM
O=C(NC(=S)Nc1sc2c(c1C(=O)O)CCOC2)c1ccccc1 CHEMBL4065916 EC50 110.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)c3ccccc3F)c2C(=O)O)CO1 CHEMBL4072366 EC50 140.0 nM
COc1ccc(C(=O)NC(=S)Nc2sc3c(c2C(=O)O)CC(C)(C)OC3)cc1 CHEMBL4099312 EC50 140.0 nM
CC1Cc2c(sc(NC(=S)NC(=O)c3ccccc3)c2C(=O)O)CO1 CHEMBL4087327 EC50 140.0 nM
COc1cccc(C(=O)NC(=S)Nc2sc3c(c2C(=O)O)CC(C)(C)OC3)c1 CHEMBL4060979 EC50 150.0 nM
CC(C)(C)C1Cc2c(sc(NC(=S)NC(=O)c3ccccc3)c2C(=O)O)CO1 CHEMBL4070133 EC50 220.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)c3ccc(Br)cc3)c2C(=O)O)CO1 CHEMBL4072864 EC50 270.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)c3cccc(F)c3)c2C(=O)O)CO1 CHEMBL4097914 EC50 290.0 nM
Cc1cccc(C(=O)NC(=S)Nc2sc3c(c2C(=O)O)CC(C)(C)OC3)c1 CHEMBL4064268 EC50 360.0 nM
Cc1ccccc1C(=O)NC(=S)Nc1sc2c(c1C(=O)O)CC(C)(C)OC2 CHEMBL4092004 EC50 410.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)c3ccccc3Br)c2C(=O)O)CO1 CHEMBL4095262 EC50 430.0 nM
CC1(C)Cc2c(sc(NC(=S)NC(=O)C3CCCCC3)c2C(=O)O)CO1 CHEMBL4079309 EC50 460.0 nM
CC1(C)Cc2c(sc(NC(=O)NC(=O)c3ccccc3)c2C(=O)O)CO1 CHEMBL4105037 EC50 830.0 nM