Cc1ccc(-n2sc(=O)n(Cc3ccc(Cl)cc3)c2=O)cc1 CHEMBL2037351 IC50 5.4 nM
Cc1ccc(Cn2sc(=O)n(Cc3ccccc3)c2=O)cc1 CHEMBL2037350 IC50 7.2 nM
Cc1ccc(Cn2c(=O)sn(-c3ccc(C)cc3)c2=O)cc1 CHEMBL2037352 IC50 8.6 nM
COc1ccc(-n2sc(=O)n(Cc3ccc(F)cc3)c2=O)cc1 CHEMBL2037229 IC50 10.9 nM
Cc1ccc(Cn2sc(=O)n(Cc3ccc(F)cc3)c2=O)cc1 CHEMBL2037234 IC50 12.9 nM
O=c1sn(-c2ccc(Cl)cc2)c(=O)n1Cc1ccc(F)cc1 CHEMBL2037228 IC50 13.5 nM
Cc1ccc(-n2sc(=O)n(CC(C)C)c2=O)cc1 CHEMBL2037365 IC50 14.0 nM
Cc1ccc(-n2sc(=O)n(Cc3ccccc3)c2=O)cc1 CHEMBL2037235 IC50 14.4 nM
CCCCn1c(=O)sn(CC)c1=O CHEMBL24773 IC50 14.4 nM
Cc1ccc(-n2sc(=O)n(Cc3cccc(C)c3)c2=O)cc1 CHEMBL2037354 IC50 14.5 nM
CCCCn1sc(=O)n(Cc2ccc(F)cc2)c1=O CHEMBL2035006 IC50 15.6 nM
O=c1sn(-c2ccccc2)c(=O)n1Cc1ccc(F)cc1 CHEMBL2037227 IC50 16.3 nM
Cc1ccc(-n2sc(=O)n(Cc3cccc(Cl)c3)c2=O)cc1 CHEMBL2037353 IC50 17.4 nM
Cc1ccc(-n2sc(=O)n(C)c2=O)cc1 CHEMBL2037358 IC50 18.9 nM
CCCCn1c(=O)sn(-c2ccc(C)cc2)c1=O CHEMBL2037362 IC50 19.7 nM
CCn1sc(=O)n(Cc2ccc(F)cc2)c1=O CHEMBL2037357 IC50 22.3 nM
CCn1sc(=O)n(C)c1=O CHEMBL2037359 IC50 22.3 nM
O=c1sn(-c2ccccc2)c(=O)n1Cc1ccccc1 CHEMBL2037236 IC50 23.5 nM
CCCCn1sc(=O)n(C)c1=O CHEMBL2037360 IC50 23.5 nM
COc1ccc(-n2sc(=O)n(Cc3ccccc3)c2=O)cc1 CHEMBL2037238 IC50 23.9 nM
CCn1sc(=O)n(CC(C)C)c1=O CHEMBL2037366 IC50 26.3 nM
Cn1c(=O)sn(C(C)(C)C)c1=O CHEMBL2037361 IC50 27.8 nM
O=c1sn(-c2ccc(Cl)cc2)c(=O)n1Cc1ccccc1 CHEMBL2037237 IC50 28.7 nM
CC(C)Cn1c(=O)sn(C(C)(C)C)c1=O CHEMBL2037368 IC50 29.1 nM
CCCCn1sc(=O)n(CCCC)c1=O CHEMBL2037363 IC50 29.8 nM
Cc1ccc(-n2sc(=O)n(Cc3ccc(F)cc3)c2=O)cc1 CHEMBL1917204 IC50 30.0 nM
O=c1sn(-c2cccc(Cl)c2)c(=O)n1Cc1ccccc1 CHEMBL2037349 IC50 32.5 nM
Cc1ccc(-n2sc(=O)n(Cc3ccc(Cl)c(Cl)c3)c2=O)cc1 CHEMBL2037356 IC50 34.2 nM
O=c1sn(-c2ccc(Cl)c(Cl)c2)c(=O)n1Cc1ccc(F)cc1 CHEMBL2037230 IC50 35.7 nM
Cc1cccc(-n2sc(=O)n(Cc3ccccc3)c2=O)c1 CHEMBL2037348 IC50 38.2 nM
CCCCn1sc(=O)n(CC(C)C)c1=O CHEMBL2037367 IC50 38.6 nM
O=c1sn(-c2cccc(Cl)c2)c(=O)n1Cc1ccc(F)cc1 CHEMBL2037233 IC50 52.3 nM
CCCCn1c(=O)sn(C(C)(C)C)c1=O CHEMBL2037364 IC50 53.6 nM
CCn1sc(=O)n(CCOC)c1=O CHEMBL2037369 IC50 54.3 nM
O=c1sn(-c2cccc(C(F)(F)F)c2)c(=O)n1Cc1ccccc1 CHEMBL2037347 IC50 57.4 nM
O=c1sn(-c2cccc(C(F)(F)F)c2)c(=O)n1Cc1ccc(F)cc1 CHEMBL2037231 IC50 79.3 nM
O=c1sn(-c2ccc(Cl)c(Cl)c2)c(=O)n1Cc1ccccc1 CHEMBL2037346 IC50 88.9 nM
Cc1cccc(-n2sc(=O)n(Cc3ccc(F)cc3)c2=O)c1 CHEMBL2037232 IC50 121.0 nM
COc1ccc(Cn2c(=O)sn(-c3ccc(C)cc3)c2=O)cc1 CHEMBL2037355 IC50 176.0 nM