C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)F CHEMBL42314 IC50 0.0 nM
CC(/C=C/[C@@H]1C[C@]1(C)c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL75133 EC50 0.2 nM
CC1=C(/C=C/C(C)=C/C=C/C(C)=C/C(=O)O)C(C)(C)CCC1 CHEMBL38 Ki 0.4 nM
CCN(c1ccc(C(=O)O)cc1)c1ccc(C(C)C)c(OCC(C)C)c1 CHEMBL5289973 EC50 0.58 nM
O=C(O)[C@@H]1C[C@H]1c1nc(-c2ccccc2)c(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)o1 CHEMBL5404648 EC50 0.7 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(-c2ccc(F)cc2)cc(C(C)C)c1OCC(F)F CHEMBL133915 Ki 0.8 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(-c2cccs2)cc(C(C)C)c1OCC(F)F CHEMBL130374 Ki 0.8 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(/C=C4\SC(=O)NC4=O)ccc3OC(F)(F)F)cc21 CHEMBL248415 EC50 0.9 nM
CCCCOc1c(/C(C)=C(F)\C=C\C(C)=C\C(=O)O)cc(C(C)C)cc1C(C)C CHEMBL131826 Efficacy 1.0 nM
CC(/C=C/C(F)=C(/C)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)(F)F)=C\C(=O)O CHEMBL335242 Efficacy 1.0 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(-c2cccc(F)c2)cc(C(C)C)c1OCC(F)F CHEMBL130232 Ki 1.0 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(-c2ccccc2F)cc(C(C)C)c1OCC(F)F CHEMBL422088 Efficacy 1.0 nM
CCCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(F)(F)C(F)(F)F)cc1C(C)C CHEMBL424269 Efficacy 1.0 nM
COc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)C)cc1C(C)C CHEMBL90824 Ki 1.0 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(C(C)C)cc(C(C)C)c1OCCF CHEMBL92430 Ki 1.0 nM
COc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL329334 Ki 1.0 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(C(C)C)cc(C(C)C)c1OCC(F)F CHEMBL88931 IC50 1.0 nM
Cc1cc2c(cc1-c1cc(CCC(=O)O)ccc1OC(F)(F)F)N(CC(F)(F)F)C(=O)CC2(C)C CHEMBL247220 EC50 1.4 nM
CC(/C=C/C1CC1(C)c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL69091 Kd 1.5 nM
CC1=C(/C=C/C(C)=C\C=C\C(C)=C\C(=O)O)C(C)(C)CCC1 CHEMBL705 EC50 1.5 nM
C/C(=C\C(=O)O)c1ccc2[nH]cc(-c3cc(C(C)(C)C)cc(C(C)(C)C)c3OCC(F)F)c2c1 CHEMBL430651 Ki 1.6 nM
CCCOc1c(-c2c[nH]c3ccc(/C(C)=C/C(=O)O)cc23)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL92447 Ki 1.6 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(/C=C/C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL246821 EC50 1.8 nM
Cc1cc2c(cc1-c1cc(/C=C/C(=O)O)ccc1OC(F)(F)F)N(CC(F)(F)F)C(=O)CC2(C)C CHEMBL247005 EC50 1.8 nM
CC(/C=C/C(F)=C(/C)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)F)=C\C(=O)O CHEMBL111217 Efficacy 2.0 nM
CCC(C)(C)c1cc(/C(C)=C(F)\C=C\C(C)=C\C(=O)O)c(OCC(F)F)c(C(C)(C)CC)c1 CHEMBL130231 Efficacy 2.0 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(-c2cc(F)cc(F)c2)cc(C(C)C)c1OCC(F)F CHEMBL337393 Efficacy 2.0 nM
COc1cc2c(cc1/C(C)=C\C=C\C(C)=C\C(=O)O)C(C)(C)CCC2(C)C CHEMBL111589 Ki 2.0 nM
CCCOc1cc2c(cc1/C(C)=C\C=C\C(C)=C\C(=O)O)C(C)(C)CCC2(C)C CHEMBL109581 EC50 2.0 nM
CCC(C)(C)c1cc(/C(C)=C\C=C\C(C)=C\C(=O)O)c(OC)c(C(C)(C)CC)c1 CHEMBL91185 Ki 2.0 nM
CCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)C)cc1C(C)C CHEMBL88740 Ki 2.0 nM
CCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)(C)CC)cc1C(C)(C)CC CHEMBL315986 Ki 2.0 nM
CC(/C=C/CC1(c2ccc3c(c2)C(C)(C)CCC3(C)C)CC1)=C\C(=O)O CHEMBL89331 Kd 2.0 nM
CCCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(/C=C/C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL246629 EC50 2.1 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc([C@@H]4C[C@H]4C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL247401 EC50 2.3 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCCCF CHEMBL92243 Ki 2.7 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL1023 EC50 2.7 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(-c2ccco2)cc(C(C)C)c1OCC(F)F CHEMBL130317 Ki 3.0 nM
CCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(F)(F)C(F)(F)F)cc1C(C)C CHEMBL132568 Efficacy 3.0 nM
Cc1cc2c(cc1C1(c3ccc(C(=O)O)cn3)CC1)C(C)(C)CCC2(C)C CHEMBL288436 Kd 3.0 nM
C/C(=C\C(=O)O)c1cc2c(-c3cc(C(C)(C)C)cc(C(C)(C)C)c3OCC(F)(F)F)cccc2s1 CHEMBL41260 Ki 3.0 nM
C/C(=C\C(=O)O)c1cc2c(-c3cc(C(C)(C)C)cc(C(C)(C)C)c3OCCCF)cccc2s1 CHEMBL41146 Ki 3.0 nM
CCC(C)/C=C/CC(=C/C(=O)O)/C=C/C1=C(C)CCCC1(C)C CHEMBL75548 Kd 3.0 nM
CCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)C)cc1C(C)C CHEMBL91779 Ki 3.0 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(C(C)C)cc(C(C)C)c1OCC(F)(F)F CHEMBL423503 Ki 3.0 nM
CC(/C=C/CC1(c2cc(C(C)(C)C)cc(C(C)(C)C)c2)CC1)=C\C(=O)O CHEMBL89581 Kd 3.0 nM
CC(/C=C/C1(c2ccc3c(c2)C(C)(C)CCC3(C)C)CC1)=C\C(=O)O CHEMBL93518 Ki 3.0 nM
CC1(C)CCC(C)(C)c2cc(C3CCCc4oc(/C=C/C(=O)O)cc43)ccc21 CHEMBL62880 EC50 3.0 nM
CC(/C=C/[C@]12CCC[C@@]1(c1ccc3c(c1)C(C)(C)CCC3(C)C)C2)=C\C(=O)O CHEMBL310047 Ki 3.0 nM
CC(/C=C/[C@H]1CCC[C@@H]1c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL80236 Ki 3.0 nM
CC1(C)CCC(C)(C)c2cc(N(CC3CC3)c3ncc(C(=O)O)cn3)ccc21 CHEMBL114640 EC50 3.0 nM
CCCCOc1c(-c2c[nH]c3ccc(/C(C)=C/C(=O)O)cc23)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL93246 Ki 3.2 nM
CCCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL110195 EC50 3.3 nM
C/C(=C/C=C/C(C)=C(\F)C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)F CHEMBL325592 EC50 3.4 nM
Cc1cc2c(cc1-c1cc(CCC(=O)O)ccc1OC(F)(F)F)N(C(C)C)C(=O)CC2(C)C CHEMBL399461 EC50 3.4 nM
CCCC1=C(CCC(C)C)/C(=C/C(C)=C\C=C\C(C)=C\C(=O)O)CCC1 CHEMBL5200645 Kd 3.6 nM
CCN(c1ccc2c(c1)C(C)(C)CCC2(C)C)c1ccc(C(=O)O)cn1 CHEMBL1221641 EC50 3.8 nM
CCOc1cc2c(cc1/C(C)=C\C=C\C(C)=C\C(=O)O)C(C)(C)CCC2(C)C CHEMBL109847 Ki 4.0 nM
C/C(=C\c1ncc(C(=O)O)s1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL328481 EC50 4.0 nM
CC(/C=C/[C@H]1C[C@@]1(C)c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL308377 EC50 4.0 nM
CCCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)C)cc1C(C)C CHEMBL414218 Ki 4.0 nM
CC(/C=C/C1(c2cc3c(cc2C)C(C)(C)CCC3(C)C)CC1)=C\C(=O)O CHEMBL92284 Ki 4.0 nM
CC1(C)CCC(C)(C)c2cc(C3CCCc4oc(/C=C5/SC(=O)NC5=O)cc43)ccc21 CHEMBL305115 EC50 4.0 nM
CC(/C=C/[C@@]1(C)CCC[C@@H]1c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL312395 Ki 4.0 nM
CC(/C=C/[C@]1(C)CCC[C@@H]1c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL75814 Ki 4.0 nM
CC1=C(/C=C\C(C)=C/C=C/C(C)=C/C(=O)O)C(C)(C)CCC1 CHEMBL4582509 EC50 4.0 nM
CCC(C)C1=C(CCC(C)C)/C(=C/C(C)=C\C=C\C(C)=C\C(=O)O)CCC1 CHEMBL5169878 Kd 4.1 nM
CC(/C=C/C=C(\C)c1cc(C(C)(C)C)cc(C(C)(C)C)c1)=C\C(=O)O CHEMBL89241 Ki 4.6 nM
CCCCC1=C(CCC(C)C)/C(=C/C(C)=C\C=C\C(C)=C\C(=O)O)CCC1 CHEMBL5190999 Kd 4.7 nM
C/C(=C/C=C(F)/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)F CHEMBL326673 Ki 4.8 nM
CCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)C)cc1C(F)(F)C(F)(F)F CHEMBL131122 Efficacy 5.0 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(C(C)C)cc(-c2ccccc2)c1OCC(F)F CHEMBL424639 Efficacy 5.0 nM
CC1(C)CCC(C)(C)c2cc(C(=C3CC3)c3ccc(C(=O)O)cc3)ccc21 CHEMBL280140 AC50 5.0 nM
CCCCCCCOc1c(-c2cccc3sc(/C(C)=C/C(=O)O)cc23)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL291034 Ki 5.0 nM
CO/N=C(\c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL423465 EC50 5.0 nM
CCO/N=C(\c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL166201 EC50 5.0 nM
CC(/C=C/C1=C(c2cc3c(cc2C)C(C)(C)CCC3(C)C)CCC1)=C\C(=O)O CHEMBL312737 Ki 5.0 nM
Cc1cc2c(cc1-c1cc(C3CC3C(=O)O)ccc1OC(F)(F)F)N(C(C)C)C(=O)CC2(C)C CHEMBL399326 EC50 5.0 nM
O=C(O)C1CC1c1nc(-c2ccccc2)c(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)o1 CHEMBL5465166 EC50 5.0 nM
CCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(F)(F)C(F)(F)F)cc1C(C)C CHEMBL133896 IC50 5.3 nM
CCN(c1ccc(C(=O)O)cn1)c1cc(OCC(C)C)c(C(C)C)cc1/C=C/c1ccccc1 CHEMBL2029403 pA2 5.495 nM
C=C(c1ccc(C(=O)O)cn1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL109117 EC50 6.0 nM
CCOc1c(-c2cccc3sc(/C(C)=C/C(=O)O)cc23)cc(C(C)C)cc1C(C)C CHEMBL41890 Ki 6.0 nM
CC(/C=C/CC1(c2cc(C(C)(C)C)cc3c2CCC3(C)C)CC1)=C\C(=O)O CHEMBL88216 Kd 6.0 nM
C=CCO/N=C(\c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL166244 EC50 6.0 nM
CCCO/N=C(\c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL165734 Ki 6.0 nM
Cc1cc2c(cc1/C(=N/O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL162334 Ki 6.0 nM
CCCOc1cc2c(cc1C(=C1CC1)c1ccc(C(=O)O)cn1)C(C)(C)CCC2(C)C CHEMBL366112 IC50 6.0 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)O[C@@H]1CCC[C@]31c1ccc(C(=O)O)cc1 CHEMBL3781132 pEC50 6.31 nM
CCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL92050 EC50 6.4 nM
CCCCCCOc1cc2c(cc1-n1c(C(F)(F)F)nc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL5093229 pA2 6.761 nM
CC1=C(/C=C/c2occc2/C=C/C(C)=C/C(=O)O)C(C)(C)CCC1 CHEMBL347411 Kd 7.0 nM
C/C(=C\C(=O)O)c1cc2c(-c3cc(C(C)(C)C)cc(C(C)(C)C)c3OCCC(F)F)cccc2s1 CHEMBL43238 Ki 7.0 nM
C/C(=C\C(=O)O)c1cc2c(-c3cc(C(C)(C)C)cc(C(C)(C)C)c3C)cccc2s1 CHEMBL44420 Ki 7.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(CCC(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL246825 EC50 7.2 nM
CCCCOc1c(-c2c[nH]c3ccc(/C(C)=C/C(=O)O)cc23)cc(C(C)C)cc1C(C)C CHEMBL92798 Ki 7.4 nM
C/C(=C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)(F)F CHEMBL92487 IC50 8.0 nM
CCCN(C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc2c1CCC2(C)C CHEMBL208316 Ki 8.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCc2ccc(C)cc21 CHEMBL3289659 Kd 8.0 nM
C/C(=C/C(F)=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)F CHEMBL110921 Ki 8.2 nM
CCCCCOc1cc2c(cc1-n1c(C(F)(F)F)nc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL5088616 pA2 8.71 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCC(C(C)C)=C1CCC(C)C CHEMBL3622724 Kd 9.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCCc2ccccc21 CHEMBL3622719 Kd 9.0 nM
C/C(=C\C(=O)O)c1cc2c(o1)CCCC2c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL2113737 EC50 10.0 nM
CCCCOc1cc2c(cc1C(=C1CC1)c1ccc(C(=O)O)cn1)C(C)(C)CCC2(C)C CHEMBL184497 IC50 10.0 nM
Cc1cc2c(cc1-c1cc([C@@H]3C[C@H]3C(=O)O)ccc1OC(F)(F)F)N(C(C)C)C(=O)CC2(C)C CHEMBL247402 EC50 10.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCc2cccc(C)c21 CHEMBL3289660 Kd 10.0 nM
C/C(=C\c1ccc(C(=O)O)s1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL91718 EC50 11.0 nM
CCCCOc1c(-c2cccc3cc(/C(C)=C(\F)C(=O)O)oc23)cc(C(C)C)cc1C(C)C CHEMBL290246 IC50 11.0 nM
Cc1cc2c(cc1/C(=N/OCC#N)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL164902 Ki 11.0 nM
C/C(=C\C(=O)O)c1cc2c(-c3cc(C(C)(C)C)cc(C(C)(C)C)c3OCC(F)F)cccc2s1 CHEMBL290761 Ki 12.0 nM
CC1(C)CCC(C)(C)c2cc(/C(=N/O)c3ccc(C(=O)O)cc3)c(Br)cc21 CHEMBL348797 Ki 12.0 nM
Cc1cc2c(cc1Cc1ccc(C(=O)O)c(F)c1)C(C)(C)CCC2(C)C CHEMBL583996 Ki 12.0 nM
CCN(c1ccc(C(C)C)c(OCC(C)CF)c1)c1ccc(C(=O)O)cn1 CHEMBL3425764 EC50 12.0 nM
CC1=C(/C=C\C(C)=C\C=C\C(C)=C\C(=O)O)C(C)(C)CCC1 CHEMBL44478 EC50 13.0 nM
CCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)(C)CC)cc1C(C)(C)CC CHEMBL90254 IC50 13.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CC[C@H](C)c2ccccc21 CHEMBL3098858 Kd 13.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCC(CCC(C)C)=C1CCC(C)C CHEMBL5197860 Kd 13.0 nM
CCCOc1c(-c2cccc3sc(/C(C)=C/C(=O)O)cc23)cc(C(C)C)cc1C(C)C CHEMBL41742 Ki 14.0 nM
CCCOc1c(/C(C)=C\C=C\C(C)=C\C(=O)O)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL420249 Ki 14.0 nM
CCC1=C(CCC(C)C)/C(=C/C(C)=C\C=C\C(C)=C\C(=O)O)CCC1 CHEMBL3622722 Kd 14.0 nM
CC(/C=C/[C@@H]1CCC[C@@H]1c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL311113 Ki 15.0 nM
Cc1cc2c(cc1-n1c(C(F)(F)F)nc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL2332887 EC50 15.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCc2cc(C)ccc21 CHEMBL3289658 Kd 15.0 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)O[C@@H]1CCCC[C@]31c1ccc(C(=O)O)cc1 CHEMBL3780763 pEC50 15.85 nM
CCC1=C(C(C)C)/C(=C/C(C)=C\C=C\C(C)=C\C(=O)O)CCC1 CHEMBL2114968 Kd 16.0 nM
C/C=C(\C)CC(=C/C(=O)O)/C=C(C)/C=C1\CCCC(CC)=C1C(C)C CHEMBL72988 Kd 16.0 nM
CCC(C)(C)c1cc(/C(C)=C\C=C\C(C)=C\C(=O)O)c(OCC(F)F)c(C(C)(C)CC)c1 CHEMBL313647 IC50 16.0 nM
CC(/C=C/CC1(c2cc3c(cc2C)C(C)(C)CCC3(C)C)CC1)=C\C(=O)O CHEMBL89058 Kd 16.0 nM
CCCOc1cc2c(cc1/C(C)=C/C=C/C(C)=C/C(=O)O)C(C)(C)CCC2(C)C CHEMBL5273291 EC50 16.0 nM
O=C(O)[C@H]1C[C@@H]1c1nc(-c2ccccc2)c(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)o1 CHEMBL5412777 EC50 16.0 nM
Cc1cc2c(cc1-c1cc(/C=C/C(=O)O)ccc1OC(F)(F)F)N(C(C)C)C(=O)CC2(C)C CHEMBL428930 EC50 16.3 nM
CCCN(C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1 CHEMBL379057 Ki 17.0 nM
CCCN(C/C=C/C(C)=C/C(=O)O)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL205532 Ki 18.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCc2c(C)cccc21 CHEMBL3289657 Kd 18.0 nM
Cc1cc2c(cc1-c1cc(/C=C/C(=O)O)ccc1OCC(F)(F)F)N(C(C)C)C(=O)CC2(C)C CHEMBL247819 EC50 18.3 nM
C[C@H](NC(=O)[C@H](Cc1ccccc1)NP(=O)(O)O)C(=O)NCC(N)=O CHEMBL2372524 Ki 19.0 nM
CCN(c1ccc(C(C)C)c(OCC(C)C)c1)c1ccc(C(=O)O)cn1 CHEMBL1688383 EC50 19.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCC(C2CC2)=C1CCC(C)C CHEMBL3622723 EC50 19.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(C4CC4C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL246824 EC50 19.2 nM
C=C(c1ccc(C(=O)NO)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL2398772 EC50 19.5 nM
CC(C)c1cccc(-c2cc(/C=C/C(=O)O)ccc2O)c1 CHEMBL5266566 pEC50 19.95 nM
CC1(C)CCC(C)(C)c2cc(C3CCCc4sc(/C=C/C(=O)O)cc43)ccc21 CHEMBL62537 EC50 20.0 nM
COc1cc2c(cc1C1CCCc3oc(/C=C/C(=O)O)cc31)C(C)(C)CCC2(C)C CHEMBL294346 Ki 20.0 nM
CC(/C=C/C1=C(c2ccc3c(c2)C(C)(C)CCC3(C)C)CCC1)=C\C(=O)O CHEMBL79234 Ki 20.0 nM
CC(/C=C/C1(c2cc3c(cc2C)C(C)(C)CCC3(C)C)OCCO1)=C\C(=O)O CHEMBL111911 EC50 21.0 nM
Cc1cc2c(cc1/C(=N/OCC(C)C)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL351943 Ki 21.0 nM
Cc1cc2c(cc1C(=C1CC1)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL277626 IC50 21.0 nM
CCCCN(C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc2c1CCC2(C)C CHEMBL204725 Ki 21.0 nM
CC(/C=C/[C@@H]1CCCN1c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL378926 Ki 21.0 nM
CC(C)=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL25244 AC50 22.0 nM
CCOc1c(-c2cccc3cc(/C(C)=C/C(=O)O)oc23)cc(C(C)C)cc1C(C)C CHEMBL289057 Ki 22.0 nM
C/C(=C(/F)C(=O)O)c1cc2cccc(-c3cc(C(C)C)cc(C(C)C)c3OCC(F)F)c2o1 CHEMBL41422 IC50 22.0 nM
CN1Cc2oc(/C=C/C(=O)O)cc2C(c2ccc3c(c2)C(C)(C)CCC3(C)C)C1 CHEMBL2113736 EC50 22.0 nM
Cc1cc2c(cc1-c1cc3cc(C(=O)O)c(=O)oc3cc1O)C(C)(C)CCC2(C)C CHEMBL4449685 EC50 22.0 nM
C/C(=C\c1nc(-c2ccccc2)c(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)o1)C(=O)O CHEMBL5407623 EC50 22.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCC(C)c2ccccc21 CHEMBL3098772 Kd 23.0 nM
Cc1cc2c(cc1-c1cc(/C=C/C(=O)O)ccc1OC(F)(F)F)N(C)C(=O)CC2(C)C CHEMBL247836 EC50 24.3 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CC[C@@H](C)c2ccccc21 CHEMBL3098773 Kd 25.0 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)OC1CCCC31c1ccc(C(=O)O)cc1 CHEMBL3779935 pEC50 25.12 nM
CC1=C(/C=C/c2ccccc2/C=C/C(C)=C/C(=O)O)C(C)(C)CCC1 CHEMBL157333 Kd 26.0 nM
Cc1cc2c(cc1C1(c3ccc(C(=O)O)cc3)CC1)C(C)(C)CCC2(C)C CHEMBL106896 EC50 26.0 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1Cl)C(C)(C)CCC2(C)C CHEMBL101609 Kd 27.0 nM
Cc1cc2c(cc1-n1c(C(F)(F)F)nc3cc(C(=O)O)cnc31)C(C)(C)CCC2(C)C CHEMBL4465555 EC50 27.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(/C=C(\C)C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL248016 EC50 27.9 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1Br)C(C)(C)CCC2(C)C CHEMBL101661 Kd 28.0 nM
Cc1cc2c(cc1C1CCCc3oc(/C=C/C(=O)O)cc31)C(C)(C)CCC2(C)C CHEMBL432140 EC50 29.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCc2ccccc21 CHEMBL3098771 Kd 29.0 nM
Cc1cc2c(cc1C1(c3ccc(C(=O)O)cc3)OCCO1)C(C)(C)CCC2(C)C CHEMBL5280414 EC50 29.0 nM
COc1c(-c2csc3ccc(/C(C)=C/C(=O)O)cc23)cc(C(C)C)cc1C(C)C CHEMBL314745 Ki 29.6 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1CC)C(C)(C)CCC2(C)C CHEMBL100623 Kd 31.0 nM
CCN(C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1 CHEMBL205634 Ki 31.0 nM
C/C(=C\c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL32505 IC50 32.0 nM
CCN(c1ccc(C(=O)O)cc1)c1ccc(C(C)C)c(OC(C)C)c1 CHEMBL5279494 EC50 32.0 nM
CC1=C(C(C)C)/C(=C/C(C)=C\C=C\C(C)=C\C(=O)O)CCC1 CHEMBL2111790 Kd 33.0 nM
CC1(C)CCC(C)(C)c2cc(C3(c4ccc(C(=O)O)cc4)OCCO3)ccc21 CHEMBL112715 EC50 34.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCC(C2CC2)=C1C(C)C CHEMBL3622720 Kd 34.0 nM
O=C(O)/C=C/c1nc(-c2ccccc2)c(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)o1 CHEMBL5436895 EC50 35.0 nM
Cc1cc2c(cc1-c1cc(CCC(=O)O)ccc1OCC(F)(F)F)N(C(C)C)C(=O)CC2(C)C CHEMBL410399 EC50 36.5 nM
CC(/C=C/CN(C)c1cc(C(C)(C)C)cc(C(C)(C)C)c1)=C\C(=O)O CHEMBL208213 Ki 37.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(C(C)CC(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL247000 EC50 37.7 nM
CCOc1c(/C(=C\C=C\C(C)=C\C(=O)O)C(F)(F)F)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL107555 EC50 38.0 nM
C=C1C[C@H](c2ccc3c(c2)C(C)(C)CCC3(C)C)[C@@H](/C=C/C(C)=C/C(=O)O)C1 CHEMBL312233 Ki 38.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(/C=C\C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL246823 EC50 39.1 nM
O=C(/C=C/c1ccccc1)Nc1cc(-c2ccnc(N3CCC(CO)CC3)c2)ccn1 CHEMBL5438255 Kd 39.39 nM
CCCOc1cc2c(cc1C1CCCc3oc(/C=C/C(=O)O)cc31)C(C)(C)CCC2(C)C CHEMBL64771 EC50 40.0 nM
CC(/C=C/CC1(c2ccc3c(c2)C(C)(C)CCC3(C)C)CCCC1)=C\C(=O)O CHEMBL90674 Kd 41.0 nM
CC1(C)CCC(C)(C)c2cc(C3CCCc4oc(/C=C/C(=O)O)nc43)ccc21 CHEMBL64222 EC50 42.0 nM
CCN(C/C=C/C(C)=C/C(=O)O)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL427391 Ki 42.0 nM
CCCOc1c(-c2cccc3cc(/C(C)=C/C(=O)O)oc23)cc(C(C)C)cc1C(C)C CHEMBL41675 Ki 44.0 nM
Cc1cc2c(cc1-c1cc(CCC(=O)O)ccc1OC(F)(F)F)N(C)C(=O)CC2(C)C CHEMBL248236 EC50 45.9 nM
Cc1cc2c(cc1/C(=N\O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL3350249 EC50 46.0 nM
C/C(=C\C(=O)O)c1cc2cccc(-c3cc(C(C)C)cc(C(C)C)c3OCCCF)c2o1 CHEMBL290399 Ki 47.0 nM
CCCN(C/C=C/C(C)=C/C(=O)O)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL205600 Ki 47.0 nM
CCN(c1ccc(C(=O)O)cn1)c1cc(OCC(C)C)c(C(C)C)cc1NC(=O)c1ccccc1 CHEMBL4778155 pA2 47.86 nM
O=C(O)CCc1nc(-c2ccccc2)c(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)o1 CHEMBL4855847 EC50 50.0 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)OC1CCCCC31c1ccc(C(=O)O)c(F)c1 CHEMBL3781998 pEC50 50.12 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)OC1CCCCC31c1ccc(C(=O)O)cc1 CHEMBL3780004 pEC50 50.12 nM
Cc1cc2c(cc1C1(c3ccc(C(=O)O)cc3)CO1)C(C)(C)CCC2(C)C CHEMBL106817 EC50 51.0 nM
CC(/C=C/C1(c2ccc3c(c2)C(C)(C)CCC3(C)C)CCCC1)=C\C(=O)O CHEMBL93848 EC50 51.0 nM
Cc1cc2c(cc1Sc1ccc(C(=O)O)cn1)C(C)(C)CCC2(C)C CHEMBL116886 EC50 54.0 nM
C/C=C(/c1ccc(C(=O)O)cc1)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL115050 EC50 55.0 nM
CC1(C)CCC(C)(C)c2cc(C3(c4ccc(C(=O)O)cc4)CC3)ccc21 CHEMBL326855 EC50 55.0 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1C(C)C)C(C)(C)CCC2(C)C CHEMBL99325 Kd 55.0 nM
C/C(=C\c1ncc(C(=O)O)n1S(=O)(=O)N(C)C)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL433178 EC50 59.0 nM
O=C(O)CCc1nc(-c2ccccc2)c(-c2cc(Cl)cc(Cl)c2)o1 CHEMBL4874191 EC50 60.0 nM
CCN1C(=O)C(C)(C)Oc2cc(C)c(-c3cc(/C(C)=C/C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL248191 EC50 61.2 nM
CC(/C=C/CN(CC1CC1)c1cc(C(C)(C)C)cc2c1CCC2(C)C)=C\C(=O)O CHEMBL377178 Ki 63.0 nM
CCCCCCOc1cc2c(cc1N(C)c1ncc(C(=O)O)cn1)C(C)(C)CCC2(C)C CHEMBL115097 pA2 63.1 nM
C=C1C[C@@H](/C=C/C(C)=C/C(=O)O)[C@@H](c2ccc3c(c2)C(C)(C)CCC3(C)C)C1 CHEMBL80424 Ki 66.0 nM
CCN(c1ccc(C(C)C)c(OC(C)C)c1)c1ccc(C(=O)O)cn1 CHEMBL1688382 EC50 66.0 nM
CC(/C=C/CN(c1cc(C(C)(C)C)cc2c1CCC2(C)C)C(C)C)=C\C(=O)O CHEMBL205694 Ki 67.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(/C=C/C(=O)O)ccc3OCC(F)(F)F)cc21 CHEMBL400557 EC50 67.3 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1F)C(C)(C)CCC2(C)C CHEMBL330593 Kd 69.0 nM
CCOc1c(-c2[nH]nc3ccc(/C(C)=C/C(=O)O)cc23)cc(C(C)C)cc1C(C)C CHEMBL91979 Ki 69.2 nM
O=C(O)CCc1nc(-c2ccccc2)c(-c2cccc(C(F)(F)F)c2)o1 CHEMBL4876667 EC50 70.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(CCC(=O)O)ccc3OCC(F)(F)F)cc21 CHEMBL400894 EC50 70.2 nM
CC(/C=C/C1CC1(C)c1cc2c(cc1C)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL308883 Kd 71.0 nM
CC1(C)CCC(C)(C)c2cc(C3(c4ccc(C(=O)O)cc4)OCCS3)ccc21 CHEMBL113975 EC50 74.0 nM
CCCN1c2ccc(NS(=O)(=O)c3cccc(C(F)(F)F)c3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL238009 IC50 76.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCC(c2ccccc2)=C1CCC(C)C CHEMBL3622725 EC50 80.0 nM
O=C(O)Cc1ccc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 CHEMBL4451817 EC50 80.0 nM
Cc1cc2c(cc1Cc1ccc(C(=O)O)c([N+](=O)[O-])c1)C(C)(C)CCC2(C)C CHEMBL583410 Ki 81.0 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1OC)C(C)(C)CCC2(C)C CHEMBL101212 EC50 83.0 nM
Cc1cc2c(cc1-n1ccc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL2332890 EC50 83.0 nM
CC(C)=C(c1ccc(C(=O)O)cc1)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL24966 EC50 86.0 nM
CCCCO/N=C(\c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL162005 EC50 86.0 nM
CCOCCOc1cc2c(cc1-n1c(C(F)(F)F)nc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL4777069 pA2 87.1 nM
C/C(=C\c1nc(C(=O)O)c[nH]1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL329802 EC50 89.0 nM
CN(c1cc(C(F)(F)F)nc(OCCC(=O)O)n1)c1cccc2c1CCC2 CHEMBL4558880 EC50 93.0 nM
CCN1c2ccc(NS(=O)(=O)c3cccc(C(F)(F)F)c3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL393650 IC50 95.0 nM
O=C(O)c1ccc(COc2ccccc2-c2ccccc2)cc1 CHEMBL4455253 Kd 95.0 nM
CCn1c(=O)c2c(c3cc(-c4cc(/C=C/C(=O)O)ccc4OC(F)(F)F)ccc31)CCC2 CHEMBL247012 EC50 96.6 nM
CC1(C)CCC(C)(C)c2cc(C3CCCc4sc(CCC(=O)O)cc43)ccc21 CHEMBL60090 EC50 97.0 nM
Cc1cc2c(cc1C1=NOC(c3ccc(C(=O)O)cc3)C1)C(C)(C)CCC2(C)C CHEMBL25337 AC50 100.0 nM
CCN(C/C=C/C(C)=C/C(=O)O)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL378553 Ki 103.0 nM
CC(/C=C/[C@H]1CCCN1c1ccc2c(c1)C(C)(C)CCC2(C)C)=C\C(=O)O CHEMBL208503 Ki 103.0 nM
C/C(=C\c1ccc(C(=O)O)cn1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL92926 EC50 105.0 nM
CC1(C)CCC(C)(C)c2cc(C(=O)c3ccc(C(=O)O)cc3)c(Br)cc21 CHEMBL101712 Kd 105.0 nM
Cc1oc(/C=C/C(=O)O)cc1Cc1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL62258 EC50 106.0 nM
Cc1cc2c(cc1C(C)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL105979 Kd 110.0 nM
C=C(C)COc1cc(N(CC)c2ccc(C(=O)O)cn2)ccc1C(C)C CHEMBL1688385 EC50 110.0 nM
C/C(=C\c1csc(C(=O)O)c1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL316336 EC50 112.0 nM
CC(C)c1cc2c(cc1C(=O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL101666 Kd 113.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(C4CC4C(=O)O)ccc3OCC(F)(F)F)cc21 CHEMBL246210 EC50 115.8 nM
CCN(c1ccc(C(=O)O)cn1)c1cc(OCC(C)C)c(C(C)C)cc1NC(=O)c1cc2cc3c4c(c2oc1=O)CCCN4CCC3 CHEMBL4788526 pA2 117.49 nM
CC1=C(C)/C(=C/C(C)=C\C=C\C(C)=C\C(=O)O)CCC1 CHEMBL2111792 Kd 120.0 nM
CCCOc1cc2c(cc1C(=C1CC1)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL187021 IC50 120.0 nM
CC(/C=C/CN(Cc1ccccc1)c1cc(C(C)(C)C)cc(C(C)(C)C)c1)=C\C(=O)O CHEMBL208529 Ki 121.0 nM
CCCCCCCCN(C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1 CHEMBL205894 Ki 122.0 nM
CC(=C/C=C/C(C)=C/C(=O)O)/C=C1\CCCC(c2ccccc2)=C1C(C)C CHEMBL3622721 Kd 125.0 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)O[C@H]1CCCCC[C@@]31c1ccc(C(=O)O)cc1 CHEMBL3781771 pEC50 125.89 nM
CC1(C)CCC(C)(C)c2cc(C(=O)c3ccc(C(=O)O)cc3)c(Cl)cc21 CHEMBL102039 Kd 130.0 nM
CN1c2ccc(S(=O)(=O)c3ccc(OC(F)(F)F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL395801 IC50 130.0 nM
CCCN1c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL397150 IC50 130.0 nM
O=C(O)CCc1nc(-c2cc(Cl)cc(Cl)c2)c(-c2ccccc2)o1 CHEMBL4446467 EC50 130.0 nM
C/C(=C\C(=O)O)c1ccc2scc(-c3cc(C(C)C)cc(C(C)C)c3O)c2c1 CHEMBL93571 Ki 131.0 nM
Cc1ccc(-c2ccc(C(=O)O)cc2)cc1-c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL27226 AC50 135.0 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1CCC)C(C)(C)CCC2(C)C CHEMBL101302 Kd 137.0 nM
Cc1cc2c(cc1C(=O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL98172 Kd 138.0 nM
CC1(C)CCC(C)(C)c2cc(Cc3coc(/C=C/C(=O)O)c3)ccc21 CHEMBL63048 Ki 138.0 nM
CCCCS(=O)(=O)Nc1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2CCC)C(C)(C)CCC3(C)C CHEMBL236697 IC50 140.0 nM
Cc1cc2c(cc1-n1nnc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL2146901 EC50 143.0 nM
Cc1cc2c(cc1-c1cc(C3CC3C(=O)O)ccc1OCC(F)(F)F)N(C)C(=O)CC2(C)C CHEMBL247400 EC50 144.0 nM
C=C(c1ccc(C(=O)O)cc1)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL96184 Kd 150.0 nM
Cc1cc2c(cc1-n1c(N)nc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL2332886 EC50 155.0 nM
CCN(c1ccc(C(C)C)c(OCC=C(C)C)c1)c1ccc(C(=O)O)cn1 CHEMBL1688386 EC50 160.0 nM
CCN(c1ccc(C(C)C)c(OCC(F)(F)F)c1)c1ccc(C(=O)O)cn1 CHEMBL1688387 EC50 160.0 nM
CCCCCOc1cc(N(CC)c2ccc(C(=O)O)cn2)ccc1C(C)C CHEMBL1688390 EC50 160.0 nM
CCN(c1ccc(C(C)C)c(OCc2ccccc2)c1)c1ccc(C(=O)O)cn1 CHEMBL1688392 EC50 160.0 nM
CC(C)(C)c1ccccc1OCc1ccc(C(=O)O)cc1 CHEMBL4570663 EC50 160.0 nM
C/C(=C\C(=O)O)c1cc2cccc(-c3cc(C(C)C)cc(C(C)C)c3OCC(F)F)c2o1 CHEMBL265051 Ki 161.0 nM
Cc1cc2c(cc1Cc1ccc(C(=O)O)cc1F)C(C)(C)CCC2(C)C CHEMBL575324 Ki 161.0 nM
CCN(c1ccc(OCC(C)C)c(C(C)C)c1)c1ccc(C(=O)O)cn1 CHEMBL3425765 EC50 169.0 nM
CC1(C)CCC(C)(C)c2cc(C3(c4ccc(C(=O)O)cc4)SCCS3)ccc21 CHEMBL323626 EC50 170.0 nM
COc1ccc(S(=O)(=O)c2ccc3c(c2)N=C(c2ccc(C(=O)O)cc2)c2cc4c(cc2N3C)C(C)(C)CCC4(C)C)cc1 CHEMBL409214 IC50 170.0 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)CCC1(CCc2cc(C(=O)O)ccc2O1)O3 CHEMBL5172069 EC50 170.0 nM
CCN1C(=O)C(C)(C)Oc2cc(C)c(-c3cc(/C=C/C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL247856 EC50 173.1 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)C(C)C2(C)C CHEMBL106837 Kd 176.0 nM
CCCCOc1cc(N(CC)c2ccc(C(=O)O)cn2)ccc1C(C)C CHEMBL1688389 EC50 180.0 nM
O=C(O)CCc1nc(-c2ccc(Cl)cc2)c(-c2cc(Cl)cc(Cl)c2)o1 CHEMBL4879068 EC50 180.0 nM
CCCCNS(=O)(=O)c1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2C)C(C)(C)CCC3(C)C CHEMBL427694 IC50 190.0 nM
CN1c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL235204 IC50 190.0 nM
CCc1cc2c(cc1C(=O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL97910 Kd 195.0 nM
C/C(=C\C(=O)O)c1cc2cccc(-c3cc(C(C)C)cc(C(C)C)c3OCC(F)(F)F)c2o1 CHEMBL39206 Ki 198.0 nM
Cc1cc2c(cc1-c1cc([C@H]3C[C@@H]3C(=O)O)ccc1OC(F)(F)F)N(C(C)C)C(=O)CC2(C)C CHEMBL248414 EC50 198.0 nM
CC(C)=C(/C=C/C(C)=C/C(=O)O)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL115164 EC50 200.0 nM
CCCCS(=O)(=O)Nc1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2CC)C(C)(C)CCC3(C)C CHEMBL396661 IC50 200.0 nM
Cc1cc(COc2ccc(C)c3c2CCC3)ccc1CCC(=O)O CHEMBL5415488 Kd 200.0 nM
C/C(=C\c1cc(C(=O)O)cs1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL93628 EC50 201.0 nM
CCN(c1ccc2c(c1)C(C)(C)CCC2(C)C)c1ccc(-c2nnn[nH]2)cn1 CHEMBL1221640 EC50 205.0 nM
COc1ccc(C2CC2C(=O)O)cc1-c1cc2c(cc1C)C(C)(C)CC(=O)N2C(C)C CHEMBL246211 EC50 207.5 nM
C/C(=C\c1ncc(C(=O)O)s1)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL93577 EC50 210.0 nM
Cc1cc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)ccc1CC(=O)O CHEMBL4476449 EC50 210.0 nM
C=C(/C=C/C=C/C(=O)O)c1cc(C(C)(C)C)cc2c1CCC2(C)C CHEMBL90113 Kd 220.0 nM
CCN1c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL397149 IC50 220.0 nM
CCCCCOc1cc2c(cc1-c1cc(CCC(=O)O)ccc1O)C(C)(C)CCC2(C)C CHEMBL5278384 EC50 240.0 nM
CCCS(=O)(=O)Nc1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2C)C(C)(C)CCC3(C)C CHEMBL391903 IC50 250.0 nM
O=C(O)CCCc1cc(-c2cc(Cl)cc(Cl)c2)n(-c2ccccc2)n1 CHEMBL4862605 EC50 250.0 nM
CO/N=C(/c1ccc(C(=O)O)cc1)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL164557 EC50 253.0 nM
CC(C)=CCN(C/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc2c1CCC2(C)C CHEMBL204789 Ki 254.0 nM
CCCN(C/C=C/C(C)=C/C(=O)O)c1cc2c(cc1OC)C(C)(C)CCC2(C)C CHEMBL204773 Ki 257.0 nM
CCCc1cc2c(cc1C(=O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL98142 Kd 269.0 nM
CCCCOc1cc2c(cc1C(=C1CC1)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL188581 IC50 270.0 nM
CCOc1c(-c2cccc3cc(/C(C)=C/C(=O)O)sc23)cc(C(C)C)cc1C(C)C CHEMBL417520 Ki 271.0 nM
C/C(=C\c1ccc(C(=O)O)cc1)c1cc2c(cc1Cl)C(C)(C)CCC2(C)C CHEMBL36464 EC50 275.0 nM
Cc1cc2c(cc1-n1nnc3cc(C(=O)O)cnc31)C(C)(C)CCC2(C)C CHEMBL4546707 EC50 275.0 nM
Cc1cc2c(cc1Sc1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL118693 EC50 280.0 nM
CCCCCCOc1cc(N(CC)c2ccc(C(=O)O)cn2)ccc1C(C)C CHEMBL1688391 EC50 280.0 nM
CN1c2ccc([N+](=O)[O-])cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL326525 IC50 290.0 nM
CCN(c1ccc(C(C)C)c(OCC2CC2)c1)c1ccc(C(=O)O)cn1 CHEMBL1688384 EC50 290.0 nM
C/C(=C\c1ccc(C(=O)O)cc1)c1cc2c(cc1Br)C(C)(C)CCC2(C)C CHEMBL284167 EC50 298.0 nM
CC(c1ccc(C(=O)O)cc1)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL115763 EC50 300.0 nM
C/C(=C\c1ccc(C(=O)O)cc1)c1cc2c(cc1C(C)C)C(C)(C)CCC2(C)C CHEMBL424636 EC50 300.0 nM
Cc1cc(C)cc(-c2oc(CCC(=O)O)nc2-c2ccccc2)c1 CHEMBL4855868 EC50 300.0 nM
CC(C)(C)c1cc(-c2oc(CCC(=O)O)nc2-c2ccccc2)cc(C(C)(C)C)c1 CHEMBL4854458 EC50 300.0 nM
O=C(O)CCc1cc(-c2cc(Cl)cc(Cl)c2)n(-c2ccc(Cl)cc2)n1 CHEMBL4849999 EC50 300.0 nM
CCc1cc2c(cc1/C(C)=C/c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL284937 IC50 320.0 nM
CCN1c2ccc(C#N)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL244832 IC50 320.0 nM
C=C(c1ccc(C(=O)O)s1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL111983 EC50 330.0 nM
CCN(c1ccc(C(C)C)c(OCCc2ccccc2)c1)c1ccc(C(=O)O)cn1 CHEMBL1688393 EC50 330.0 nM
CCCS(=O)(=O)Nc1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2CC)C(C)(C)CCC3(C)C CHEMBL391309 IC50 340.0 nM
Cc1cc2c(cc1/C(=N/OCCN)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL162876 EC50 350.0 nM
O=C(O)CSc1nc(Cl)cc(Nc2cccc3c2CCCC3)n1 CHEMBL4575123 Kd 350.0 nM
COc1ccc(CCC(=O)O)cc1-c1cc2c(cc1C)C(C)(C)CC(=O)N2C(C)C CHEMBL428406 EC50 361.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc([C@H]4C[C@@H]4C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL399327 EC50 361.0 nM
Cc1cc2c(cc1-n1c(C)nc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL2146900 EC50 367.0 nM
CCCCS(=O)(=O)Nc1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2C)C(C)(C)CCC3(C)C CHEMBL391112 IC50 370.0 nM
CC1=CC(C)=[N+]2C1=C(c1ccc(C(=O)NCCOCCOc3cc4c(cc3-n3c(C(F)(F)F)nc5cc(C(=O)O)ccc53)C(C)(C)CCC4(C)C)cc1)c1c(C)cc(C)n1[B-]2(F)F CHEMBL4763024 Kd 375.0 nM
CC(C)=C(/C=C/C(C)=C/C(=O)O)c1ccc2c(c1)C(C)(C)CCC2(C)C CHEMBL414233 EC50 380.0 nM
CO/N=C(/c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL2110181 EC50 384.0 nM
CN1c2ccc(Sc3ccc(OC(F)(F)F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL395564 IC50 390.0 nM
C/C(=C\C(=O)O)c1ccc2scc(-c3cc(C(C)C)cc(C(C)C)c3OCCCF)c2c1 CHEMBL264746 Ki 394.7 nM
CN1c2ccc(NS(=O)(=O)/C=C/c3ccccc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL236698 IC50 400.0 nM
CN1c2ccc(S(=O)(=O)Cc3ccc(Cl)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL397281 IC50 420.0 nM
Cc1ccc(-c2ccc(C(=O)O)cc2)cc1-c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL25088 AC50 430.0 nM
CN1c2ccc(C#N)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL244621 IC50 430.0 nM
Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)N=C(c2ccc(C(=O)O)cc2)c2cc4c(cc2N3C)C(C)(C)CCC4(C)C)cc1 CHEMBL437956 IC50 430.0 nM
O=C(O)CCc1cc(-c2cc(Cl)cc(Cl)c2)n(-c2ccc(F)cc2)n1 CHEMBL4849776 EC50 430.0 nM
O=C(O)CCc1cc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)n(-c2ccc(Cl)cc2)n1 CHEMBL4855407 EC50 440.0 nM
CN1c2ccc(S(=O)(=O)N3CCOCC3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL244565 IC50 450.0 nM
CN1c2ccc(S(=O)(=O)N3CCCC3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL397512 IC50 450.0 nM
CCCS(=O)(=O)c1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2C)C(C)(C)CCC3(C)C CHEMBL245242 IC50 450.0 nM
CCCOc1cc(N(CC)c2ccc(C(=O)O)cn2)ccc1C(C)C CHEMBL1688388 EC50 450.0 nM
CCN(c1ccc(OCC(C)CF)c(C(C)C)c1)c1ccc(C(=O)O)cn1 CHEMBL3425828 EC50 450.0 nM
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1O)C(C)(C)CCC2(C)C CHEMBL328419 EC50 455.0 nM
Cc1cc2c(cc1Cc1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL432587 EC50 460.0 nM
CN1c2ccc(S(=O)(=O)Nc3ccc(OC(F)(F)F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL397511 IC50 460.0 nM
COc1ccc(S(=O)(=O)Nc2ccc3c(c2)N=C(c2ccc(C(=O)O)cc2)c2cc4c(cc2N3C)C(C)(C)CCC4(C)C)cc1 CHEMBL397151 IC50 470.0 nM
CC(C)(C)c1cc(-c2ccc(CC(=O)O)cc2)cc(C(C)(C)C)c1 CHEMBL4578667 EC50 470.0 nM
CN1c2ccc(NS(=O)(=O)c3cccc(C(F)(F)F)c3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL393451 IC50 480.0 nM
O=C(O)CCCc1nc(-c2ccccc2)c(-c2cc(Cl)cc(Cl)c2)o1 CHEMBL4868343 EC50 480.0 nM
Cc1cc2c(cc1/C(=N/OC(C)(C)C)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL162827 Ki 484.0 nM
Cc1cc(=O)oc2c(/C=N/NC(=O)CSc3nc4ccccc4s3)c(O)ccc12 CHEMBL3319093 Kd 488.0 nM
CCCCc1cc2c(cc1C(=C1CC1)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL188638 IC50 500.0 nM
CCN1c2ccc(C#N)cc2N=C(c2ccc(C(=O)O)c(F)c2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL398163 IC50 500.0 nM
O=C(O)CCc1nc(-c2ccccc2)c(-c2cccc(Cl)c2)o1 CHEMBL4875485 EC50 500.0 nM
Cc1cccc(-c2oc(CCC(=O)O)nc2-c2ccccc2)c1 CHEMBL4859732 EC50 500.0 nM
Cc1cc(COc2cccc3c2CCC3)ccc1CCC(=O)O CHEMBL5430265 EC50 500.0 nM
CN1c2ccc(NS(=O)(=O)c3ccccc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL396658 IC50 510.0 nM
O=C(O)CCc1nc(-c2ccccc2)c(-c2ccc(Cl)c(Cl)c2)o1 CHEMBL4852349 EC50 510.0 nM
Cc1cc2c(cc1Oc1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL105805 Kd 520.0 nM
CN1c2ccc(C#N)cc2N=C(c2ccc(C(=O)O)c(F)c2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL396200 IC50 520.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(CCCC(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL247849 EC50 527.0 nM
CC(/C=C/CNc1cc(C(C)(C)C)cc(C(C)(C)C)c1)=C\C(=O)O CHEMBL208349 Ki 529.0 nM
CCN1c2ccc(C#N)cc2N=C(c2ccc(C(=O)O)cc2F)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL242274 IC50 530.0 nM
CC1(C)CCC(C)(C)c2cc(C3(c4ccc(C(=O)O)cc4)SCCCS3)ccc21 CHEMBL113864 EC50 540.0 nM
CCCN1c2ccc(NS(=O)(=O)CCC)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL237762 IC50 550.0 nM
C/C(=C\c1ccc(C(=O)O)o1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL96829 EC50 592.0 nM
O=C(O)CCc1ccc(COc2cccc3c2CCC3)cc1 CHEMBL5415478 EC50 600.0 nM
CCO/N=C(/c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C CHEMBL2110180 Ki 620.0 nM
O=C(O)CCc1nc(-c2ccc(Cl)c(Cl)c2)c(-c2ccccc2)o1 CHEMBL4471300 EC50 620.0 nM
CC1(C)CCC(C)(C)c2cc(-n3c(C(F)(F)F)nc4cc(C(=O)O)ccc43)c(OCCOCCNc3ccc([N+](=O)[O-])c4nonc34)cc21 CHEMBL4798235 Kd 629.0 nM
Cc1cc2c(cc1-n1cnc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL2332885 EC50 633.0 nM
CCCN(C(=O)/C=C/C(C)=C/C(=O)O)c1cc(C(C)(C)C)cc(C(C)(C)C)c1 CHEMBL206005 Ki 644.0 nM
CCOc1c(-c2noc3ccc(/C(C)=C/C(=O)O)cc23)cc(C(C)C)cc1C(C)C CHEMBL328507 Ki 648.0 nM
Cc1cc2c(cc1C(C)(C)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL110629 EC50 650.0 nM
CN1c2ccc(SCc3ccc(Cl)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL438857 IC50 670.0 nM
O=C(O)CCc1nc(-c2ccccc2)c(-c2cc(F)cc(F)c2)o1 CHEMBL4865656 EC50 680.0 nM
O=C(O)CCc1cc(-c2cc(Cl)cc(Cl)c2)n(-c2ccccc2)n1 CHEMBL4873606 EC50 700.0 nM
CCCCCCOc1cc2c(cc1-n1nnc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL5081924 Kd 705.0 nM
CC1(C)CCC(C)(C)c2cc(C(=O)c3ccc(C(=O)O)cc3)c(F)cc21 CHEMBL419166 Kd 706.0 nM
Cc1cc2c(cc1/C(=N/OCC(=O)O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL348794 EC50 713.0 nM
COc1ccc(Sc2ccc3c(c2)N=C(c2ccc(C(=O)O)cc2)c2cc4c(cc2N3C)C(C)(C)CCC4(C)C)cc1 CHEMBL395563 IC50 720.0 nM
CCN1c2ccc(NC(=O)Cc3ccc(F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL237800 IC50 720.0 nM
CCCCOc1c(-c2cn(C)c3ccc(/C(C)=C/C(=O)O)cc23)cc(C(C)C)cc1C(C)C CHEMBL421748 Ki 740.0 nM
Cc1ccc(OCc2ccc(CCC(=O)O)cc2)c2c1CCC2 CHEMBL5398107 EC50 740.0 nM
CC1(C)CCC(C)(C)c2cc(C3(c4ccc(C(=O)O)cc4)OCCCO3)ccc21 CHEMBL113865 EC50 750.0 nM
CCN1C(=O)CC(C)(C)c2cc(C)c(-c3cc(CC(C)C(=O)O)ccc3OC(F)(F)F)cc21 CHEMBL246827 EC50 760.0 nM
CCCCCOc1cc2c(cc1-n1nnc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C CHEMBL5088399 Kd 764.0 nM
CC1(C)CCC(C)(C)c2cc(Sc3ccc(C(=O)O)cc3)ccc21 CHEMBL119781 EC50 770.0 nM
CC(C)=CCc1cc([C@@H]2CC(=O)c3ccc(O)c(CC=C(C)C)c3O2)cc2c1OC(C(C)(C)O)C2 CHEMBL3314592 EC50 770.0 nM
COc1ccc(CS(=O)(=O)c2ccc3c(c2)N=C(c2ccc(C(=O)O)cc2)c2cc4c(cc2N3C)C(C)(C)CCC4(C)C)cc1 CHEMBL436628 IC50 780.0 nM
CC(C)=CCc1cc([C@@H]2CC(=O)c3ccc(O)c(CC=C(C)C)c3O2)cc2c1OC(C)(C)C(O)C2 CHEMBL3314593 EC50 780.0 nM
CCN1c2ccc(C(C)=O)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL394622 IC50 790.0 nM
O=C(O)c1ccc(COc2cccc3c2CCC3)cc1F CHEMBL5417534 EC50 800.0 nM
CCCCOc1c(/C(C)=C\C=C\C(=C\C(=O)O)C(F)(F)F)cc(C(C)(C)C)cc1C(C)(C)C CHEMBL107554 EC50 805.8 nM
CC1(C)CCC(C)(C)c2cc(C(=O)c3ccc(C(=O)O)cc3)c(O)cc21 CHEMBL100986 Kd 818.0 nM
CCN(c1ccc(C(C)C)c(OCCCc2ccccc2)c1)c1ccc(C(=O)O)cn1 CHEMBL1688394 EC50 820.0 nM
CCOc1cc2c(cc1C(=O)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C CHEMBL3714906 Ki 824.0 nM
CCS(=O)(=O)Nc1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2C)C(C)(C)CCC3(C)C CHEMBL428204 IC50 840.0 nM
CN1c2ccc(NS(=O)(=O)c3cccc4ccccc34)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL391572 IC50 850.0 nM
CN1c2ccc(NC(=O)Cc3ccc(F)cc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL394103 IC50 880.0 nM
O=C(O)CCOc1nc(Nc2cccc3c2CCC3)cc(C(F)(F)F)n1 CHEMBL4518775 Kd 880.0 nM
CC(=O)c1ccc2c(c1)N=C(c1ccc(C(=O)O)cc1)c1cc3c(cc1N2C)C(C)(C)CCC3(C)C CHEMBL397034 IC50 890.0 nM
CC1(C)CCC(C)(C)c2cc3c(cc21)Sc1ccccc1N=C3c1ccc(C(=O)O)cc1 CHEMBL337859 Ki 900.0 nM
CN1c2ccc(NC(=O)c3ccccc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL236490 IC50 900.0 nM
CCN(CC)c1ccc(/C=N/NC(=O)CSc2nc3c(o2)=C=C=CC=3)c(O)c1 CHEMBL3828515 Kd 910.0 nM
N[C@@H](Cc1cc(I)c(Oc2cc(I)c(O)c(I)c2)c(I)c1)C(=O)O CHEMBL1624 Kd 930.0 nM
C/C(=C\c1nc(-c2ccccc2)c(-c2ccccc2)o1)C(=O)O CHEMBL5399947 EC50 930.0 nM
CN1c2ccc(NC(=O)Cc3ccccc3)cc2N=C(c2ccc(C(=O)O)cc2)c2cc3c(cc21)C(C)(C)CCC3(C)C CHEMBL392858 IC50 970.0 nM
Cc1c2c(n(-c3ccc(CC(=O)O)cc3)c1C)CCC(F)(F)C2 CHEMBL4171515 EC50 970.0 nM