N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OC[C@@H](O)CO)cc1 CHEMBL212531 IC50 7.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OCCCO)cc1 CHEMBL212431 IC50 7.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OCC(O)CO)cc1 CHEMBL212432 IC50 8.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OC[C@H](O)CO)cc1 CHEMBL209303 IC50 9.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OCCO)cc1 CHEMBL211161 IC50 9.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(CO)cc1 CHEMBL214239 IC50 14.0 nM
COc1ccc(CCCC/N=C(\N)NC(=O)c2nc(Cl)c(N)nc2N)cc1 CHEMBL377986 IC50 15.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1cccc(OCCO)c1 CHEMBL211600 IC50 17.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(O)cc1 CHEMBL210876 IC50 17.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OCCC(=O)O)cc1 CHEMBL379433 IC50 20.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1cccc(O)c1 CHEMBL380011 IC50 20.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(S(=O)(=O)O)cc1 CHEMBL386222 IC50 21.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(N)cc1 CHEMBL212410 IC50 21.0 nM
COC(=O)c1ccc(CCCC/N=C(\N)NC(=O)c2nc(Cl)c(N)nc2N)cc1 CHEMBL379756 IC50 22.0 nM
COc1ccc(OCCC/N=C(\N)NC(=O)c2nc(Cl)c(N)nc2N)cc1 CHEMBL214220 IC50 25.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1cccc(OCC(O)CO)c1 CHEMBL212534 IC50 26.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccccc1OCC(O)CO CHEMBL211658 IC50 28.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccccc1 CHEMBL209659 IC50 29.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccccc1O CHEMBL379066 IC50 30.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccccc1OCCO CHEMBL208889 IC50 31.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCOc1ccc(O)cc1 CHEMBL211946 IC50 32.0 nM
COc1ccc(COCC/N=C(\N)NC(=O)c2nc(Cl)c(N)nc2N)cc1 CHEMBL211773 IC50 41.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(O)c(O)c1 CHEMBL211072 IC50 42.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OCC(=O)O)cc1 CHEMBL209017 IC50 48.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCc1ccccc1 CHEMBL211664 IC50 50.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(C(=O)O)cc1 CHEMBL213175 IC50 51.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCCCc1ccccc1 CHEMBL208620 IC50 58.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCc1ccc(O)cc1 CHEMBL209977 IC50 62.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCCc1ccc(O)cc1 CHEMBL211221 IC50 64.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCc1ccccc1 CHEMBL211611 IC50 66.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCc1ccccc1 CHEMBL212579 IC50 66.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCCc1ccccc1 CHEMBL377239 IC50 68.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCc1ccc(OC2O[C@H](C(=O)O)[C@@H](O)[C@H](O)[C@H]2O)cc1 CHEMBL380393 IC50 73.0 nM
COc1ccc(CCCCC/N=C(\N)NC(=O)c2nc(Cl)c(N)nc2N)cc1 CHEMBL209104 IC50 77.0 nM
CCCCCC/N=C(\N)NC(=O)c1nc(Cl)c(N)nc1N CHEMBL210966 IC50 87.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCc1ccc(O)cc1 CHEMBL211793 IC50 88.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCO CHEMBL377688 IC50 107.0 nM
CCCCCCCC/N=C(\N)NC(=O)c1nc(Cl)c(N)nc1N CHEMBL210981 IC50 108.0 nM
COc1ccc(CCC/N=C(\N)NC(=O)c2nc(Cl)c(N)nc2N)cc1 CHEMBL210967 IC50 124.0 nM
N=C(NC(=O)c1nc(Cl)c(N)nc1N)Nc1ccccc1 CHEMBL211502 IC50 401.0 nM
N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCCCCCCCCc1ccccc1 CHEMBL210866 IC50 477.0 nM
N=C(N)NC(=O)c1nc(Cl)c(N)nc1N CHEMBL945 IC50 776.0 nM