Cc1ccc(F)c2cc(C(=O)Nc3cc(F)cc(N4CCC(N(C)C)CC4)c3)[nH]c12 CHEMBL5078908 IC50 3.0 nM
CC(=O)N1CC[C@H]2[C@@H]1CCN2[C@H]1CCC[C@@H](NC(=O)c2cc3c(F)ccc(C)c3[nH]2)C1 CHEMBL5178972 IC50 5.0 nM
CC(=O)N(C)C1CCN(c2cc(F)cc(NC(=O)c3cc4c(F)ccc(C)c4[nH]3)c2)C1 CHEMBL5073608 IC50 7.0 nM
Cc1ccc(F)c2cc(C(=O)N[C@@H]3CCC[C@H](N4CC[C@H](N(C)S(C)(=O)=O)C4)C3)[nH]c12 CHEMBL5091591 IC50 8.0 nM
Cc1ccc(F)c2cc(C(=O)Nc3cc(Cl)cc(N4CCC(N(C)C)CC4)c3)[nH]c12 CHEMBL5093241 IC50 8.0 nM
CC(=O)N1CC[C@H]2CN([C@H]3CCC[C@@H](NC(=O)c4cc5c(F)ccc(C)c5[nH]4)C3)C[C@H]21 CHEMBL5206271 IC50 11.0 nM
Cc1ccc(F)c2cc(C(=O)N[C@@H]3CCC[C@H](N4CCN5C(=O)CC[C@H]5C4)C3)[nH]c12 CHEMBL5195440 IC50 11.0 nM
Cc1ccc(F)c2cc(C(=O)N[C@@H]3CCC[C@H](N4CC[C@@H](N(C)S(C)(=O)=O)C4)C3)[nH]c12 CHEMBL5082544 IC50 12.0 nM
Cc1ccc(F)c2cc(C(=O)N[C@@H]3CCC[C@H](c4ccncc4)C3)[nH]c12 CHEMBL5082960 IC50 12.0 nM
CC(=O)N(C)C1CCN(c2cccc(NC(=O)c3cc4c(F)ccc(C)c4[nH]3)c2)C1 CHEMBL5094380 IC50 12.0 nM
CC(=O)N1CCN(c2cc(F)cc(NC(=O)c3cc4c(F)ccc(C)c4[nH]3)c2)CC1 CHEMBL5189290 IC50 12.0 nM
CC(=O)N(C)[C@@H]1CCN([C@H]2CCC[C@@H](NC(=O)c3cc4c(F)ccc(C)c4[nH]3)C2)C1 CHEMBL5071957 IC50 15.0 nM
Cc1cc(NC(=O)c2cc3c(F)ccc(C)c3[nH]2)cc(N2CCC(N(C)C)CC2)c1 CHEMBL5072597 IC50 17.0 nM
Cc1ccc(F)c2cc(C(=O)Nc3cccc(N4CCC(N(C)C)CC4)c3)[nH]c12 CHEMBL5076615 IC50 18.0 nM
CC(=O)N1CCN([C@H]2CCC[C@@H](NC(=O)c3cc4c(F)ccc(C)c4[nH]3)C2)CC1 CHEMBL5095235 IC50 18.0 nM
CC(=O)N(C)[C@H]1CCN([C@H]2CCC[C@@H](NC(=O)c3cc4c(F)ccc(C)c4[nH]3)C2)C1 CHEMBL5088515 IC50 23.0 nM
CC(=O)N1CCN(c2cccc(NC(=O)c3cc4c(F)ccc(C)c4[nH]3)c2)CC1 CHEMBL5184871 IC50 27.0 nM
Cc1ccc(F)c2cc(C(=O)N[C@@H]3CCC[C@H](N4CCN(S(C)(=O)=O)CC4)C3)[nH]c12 CHEMBL5077994 IC50 56.0 nM
Cc1ccc(F)c2cc(C(=O)Nc3cccc(N4CCN(C)CC4)c3)[nH]c12 CHEMBL5091735 IC50 66.0 nM
Cc1ccc(F)c2cc(C(=O)Nc3cccc(N4CCOCC4)c3)[nH]c12 CHEMBL5071333 IC50 101.0 nM
Cc1ccc(F)c2cc(C(=O)N[C@@H]3CCC[C@H](N4CCN(C)C(=O)C4)C3)[nH]c12 CHEMBL5080149 IC50 118.0 nM
Cc1ccc(F)c2cc(C(=O)N[C@@H]3CCC[C@H](N4CCOCC4)C3)[nH]c12 CHEMBL5072302 IC50 147.0 nM
Cc1cccnc1C(NC(=O)c1cc2c(F)ccc(C)c2[nH]1)C1CC1 CHEMBL5085128 IC50 674.0 nM
CCCN[C@@H](CC[C@H](N)C(=O)O)C[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O CHEMBL3414624 IC50(app) 800.0 nM
CCCN(CC[C@H](N)C(=O)O)C[C@@H]1O[C@H](n2cnc3c(N)ncnc32)[C@@H](O)[C@H]1O CHEMBL5187924 IC50 800.0 nM
Cc1cccc2cc(C(=O)Nc3cccc(N4CCOCC4)c3)[nH]c12 CHEMBL5076782 IC50 818.0 nM