C[C@@H]1CN(c2nnc(Cc3ccccc3)c3ccc(C#N)cc23)CCN1c1ccc(C#N)cn1 CHEMBL3290335 IC50 24.0 nM
C[C@@H]1CN(c2nnc(Cc3ccccc3)c3ccc(C(F)(F)F)cc23)CCN1c1ccc(C#N)cn1 CHEMBL3290333 IC50 100.0 nM
CCCCOc1cc(C)c(CNCC(NC(=O)c2cc(C)on2)c2ccccc2)cc1C CHEMBL3798814 IC50 117.0 nM
COc1cc(C)c(CNCC(NC(=O)c2cc(C)on2)c2ccc(C#CCO)cc2)cc1C CHEMBL3798147 IC50 150.0 nM
COc1cc(C)c(CNCC(NC(=O)c2cc(C)on2)c2ccc(CCCC(N)=O)cc2)cc1C CHEMBL3799061 IC50 150.0 nM
C[C@@H]1CN(c2nnc(Cc3ccccc3)c3ccc(Cl)cc23)CCN1c1ccc(C#N)cn1 CHEMBL3290331 IC50 210.0 nM
Cc1cc(C(=O)NC(CNCc2cc(C)c(OCC(F)(F)F)cc2C)c2ccccc2)no1 CHEMBL3798874 IC50 240.0 nM
CCOc1cc(C)c(CNCC(NC(=O)c2cc(C)on2)c2ccccc2)cc1C CHEMBL3799085 IC50 260.0 nM
COc1cc(C)c(CNC[C@@H](NC(=O)c2cc(C)on2)c2ccccc2)cc1C CHEMBL3798254 IC50 485.0 nM
COc1cc(C)c(CNCC(NC(=O)c2cc(C)on2)c2ccc(F)cc2)cc1C CHEMBL3797779 IC50 720.0 nM
COc1cc(C)c(CNCC(NC(=O)c2cc(C3CC3)on2)c2ccccc2)cc1C CHEMBL3798062 IC50 730.0 nM
C[C@@H]1CN(c2nnc(Cc3ccccc3)c3ccccc23)CCN1c1ccc([N+](=O)[O-])cn1 CHEMBL3290322 IC50 740.0 nM
COc1cc(C)c(CNCC(NC(=O)c2cc(C)on2)c2ccncc2)cc1C CHEMBL3799254 IC50 850.0 nM
Cc1cc(C(=O)NC(CNCc2cc(C)c(OCc3ccncc3)cc2C)c2ccccc2)no1 CHEMBL3798106 IC50 1000.0 nM
COc1cc(C)c(CNCC(NC(=O)c2cc(C)on2)c2ccccc2)cc1C CHEMBL3799908 IC50 1000.0 nM