COc1cc2c(cc1OCCCF)CCN1C[C@@H](CC(C)C)[C@H](O)C[C@H]21 CHEMBL579217 Ki 0.1 nM
COC(=O)[C@H]1[C@H]2C[C@@H]3c4[nH]c5cc(OC)ccc5c4CCN3C[C@H]2C[C@@H](OC(=O)c2cc(OC)c(OC)c(OC)c2)[C@@H]1OC CHEMBL772 Ki 5.26 nM
CCOC(=O)C1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CCC1c1ccc(F)cc1 CHEMBL4205254 IC50 16.0 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@@H]1c1ccccc1 CHEMBL4207658 IC50 19.7 nM
COc1cc2c(cc1OC)C1CC(=O)C(CC(C)C)CN1CC2 CHEMBL117785 IC50 19.8 nM
COc1cc2c(cc1OC)C1CC(O)C(CC(C)C)CN1CC2 CHEMBL4206824 IC50 28.1 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@@H]1c1ccc(F)cc1 CHEMBL4202787 IC50 39.4 nM
CCC1(O)CC2c3cc(OC)c(OC)cc3CCN2CC1CC(C)C CHEMBL213814 Ki 64.0 nM
O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)[nH]c3ccccc3c2=O)CC1 CHEMBL51 Ki 77.0 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@H]1c1ccc(F)cc1 CHEMBL4214975 IC50 85.5 nM
[3H]CC([3H])OC(=O)[C@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@H]1c1ccc(F)cc1 CHEMBL4207838 Kd 93.0 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@@H]1c1cccs1 CHEMBL4208250 IC50 101.0 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@@H]1c1cccc(C(F)(F)F)c1 CHEMBL4208779 IC50 125.0 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@@H]1c1cccc2c1OCCO2 CHEMBL4213176 IC50 142.0 nM
O=S(=O)(NC1CCC(c2cc(F)ccc2F)(S(=O)(=O)c2ccc(Cl)cc2)CC1)C(F)(F)F CHEMBL1091513 IC50 213.0 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@@H]1c1ccc(C)cc1 CHEMBL4216117 Ki 452.0 nM
CN1[C@@H](CCc2cccc3ccccc23)CCC[C@H]1CCc1cccc2ccccc12 CHEMBL190691 Ki 630.0 nM
CC(=O)Nc1c(C(C)=O)c(=O)n(C)c2nc(-c3ccc(Cl)cc3Cl)c(-c3ccc(Cl)cc3)cc12 CHEMBL204232 Ki 648.0 nM
CCOC(=O)[C@@H]1CN(CCn2c(=O)[nH]c3ccccc3c2=O)CC[C@@H]1c1ccc(C(F)(F)F)cc1 CHEMBL4203894 Ki 720.0 nM
CN1[C@@H](CCc2ccccc2)CCC[C@H]1CCc1ccccc1 CHEMBL333465 Ki 970.0 nM