C[C@H](C(=O)NCc1ccccc1F)N1C(=O)CCC1=O CHEMBL5187206 EC50 0.1 nM
COc1ccc2[nH]c(=O)c(C(c3nnnn3CCc3ccccc3)N3CCN(C4CCCCC4)CC3)cc2c1 CHEMBL5178416 EC50 0.26 nM
COc1ccc2[nH]c(=O)c(C(c3nnnn3CCc3ccccc3)N3CCN(c4cccc(C(F)(F)F)c4)CC3)cc2c1 CHEMBL5202745 EC50 0.3 nM
COc1ccc(NC(=O)C(=O)N2CCN(c3ccccc3)CC2)cc1 CHEMBL5181457 EC50 3.8 nM
N[C@H](C(=O)O)[C@H](OCc1cccc(NC(=O)c2ccc(C(F)(F)F)cc2)c1)C(=O)O CHEMBL1257519 IC50 10.0 nM
C[C@H](C(=O)NCc1ccccc1)N1C(=O)CCC1=O CHEMBL5206486 EC50 11.0 nM
N[C@H](C(=O)O)[C@H](OCc1cccc(NC(=O)c2cccc(C(F)(F)F)c2)c1)C(=O)O CHEMBL4173045 pIC50 16.6 nM
N[C@H](C(=O)O)[C@H](OCc1cccc(NC(=O)CCc2ccc(C(F)(F)F)cc2)c1)C(=O)O CHEMBL4176427 IC50 18.0 nM
N[C@H](C(=O)O)[C@H](OCc1cccc(NC(=O)c2ccc(-c3ccccc3)cc2)c1)C(=O)O CHEMBL5409124 IC50 21.0 nM
COc1ccc(NC(=O)C(=O)NCC(c2ccccc2)N2CCN(C)CC2)cc1 CHEMBL5208038 EC50 35.1 nM
N[C@H](C(=O)O)[C@H](OCc1ccccc1)C(=O)Nc1ccc(Oc2cc(F)c(F)cc2Br)cc1 CHEMBL4176482 IC50 36.0 nM
N[C@H](C(=O)O)[C@H](OCc1ccccc1)C(=O)Nc1ccc2c(c1)Cc1ccccc1-2 CHEMBL4177507 pIC50 46.77 nM
COc1ccc(C(=O)Nc2cccc(CO[C@H](C(=O)O)[C@H](N)C(=O)O)c2)cc1 CHEMBL5423219 IC50 59.0 nM
N[C@@H](CC(=O)Nc1ccc(-c2cccc(C(F)(F)F)c2)cc1)C(=O)O CHEMBL2113122 IC50 60.0 nM
N[C@@H](CC(=O)Nc1ccc(Oc2cc(F)c(F)cc2Br)cc1)C(=O)O CHEMBL1628669 pIC50 70.79 nM
COc1cc2cc(C(c3nnnn3Cc3ccncc3)N3CCN(C4CCCCC4)CC3)c(=O)[nH]c2cc1OC CHEMBL5207363 EC50 78.5 nM
N[C@@H](CC(=O)Nc1ccc2c(c1)Cc1cc(F)ccc1-2)C(=O)O CHEMBL2113115 IC50 80.0 nM
N[C@H](C(=O)O)[C@H](OCc1cccc(NC(=O)c2ccccc2C(F)(F)F)c1)C(=O)O CHEMBL4162363 IC50 84.0 nM
Cc1ccccc1-c1ccc(NC(=O)C[C@H](N)C(=O)O)cc1 CHEMBL2113110 IC50 100.0 nM
Cc1cc(NC(=O)C[C@H](N)C(=O)O)ccc1-c1cccc(C(F)(F)F)c1 CHEMBL2113112 IC50 100.0 nM
N[C@@H](CC(=O)Nc1ccc2c(c1)Cc1cc(Cl)ccc1-2)C(=O)O CHEMBL2113116 IC50 100.0 nM
N[C@@H](CC(=O)Nc1ccc2c(c1)Cc1cc(C(F)(F)F)ccc1-2)C(=O)O CHEMBL2113119 IC50 100.0 nM
Cc1cc(NC(=O)C[C@H](N)C(=O)O)ccc1-c1ccc(Cl)c(Cl)c1 CHEMBL2113126 IC50 100.0 nM
N[C@H](C(=O)O)[C@H](OCc1cccc(NC(=O)Cc2ccc(C(F)(F)F)cc2)c1)C(=O)O CHEMBL4165811 pIC50 107.15 nM
N[C@@H](CC(=O)Nc1ccc(Oc2ccc(F)c(F)c2)cc1)C(=O)O CHEMBL2113121 IC50 130.0 nM
Cc1cc(-c2ccccc2)ccc1NC(=O)CC(N)C(=O)O CHEMBL424838 IC50 200.0 nM
N[C@@H](CC(=O)Nc1ccc(-c2ccc(F)c(Cl)c2)c(C(F)(F)F)c1)C(=O)O CHEMBL2113113 IC50 200.0 nM
N[C@@H](CC(=O)Nc1ccc2c(c1)Cc1cc(Br)ccc1-2)C(=O)O CHEMBL2113117 IC50 200.0 nM
Cc1cc(NC(=O)C[C@H](N)C(=O)O)ccc1-c1ccc(Cl)cc1 CHEMBL2113125 IC50 200.0 nM
Cc1ccc(S(=O)(=O)n2cc(-c3ccsc3)c3ccc(CO[C@H](C(=O)O)[C@H](N)C(=O)O)cc32)cc1 CHEMBL4759043 pIC50 208.93 nM
N[C@@H](CC(=O)Nc1ccc2c(c1)Cc1c(Cl)cc(Cl)cc1-2)C(=O)O CHEMBL2113118 IC50 300.0 nM
CCN1c2ccccc2Oc2ccc(NC(=O)CC(N)C(=O)O)cc21 CHEMBL425569 IC50 300.0 nM
Cc1cc(NC(=O)C[C@H](N)C(=O)O)ccc1-c1ccc(C(F)(F)F)cc1 CHEMBL2113124 IC50 300.0 nM
N[C@@H](CC(=O)Nc1ccc(-c2ccc3ccccc3c2)cc1)C(=O)O CHEMBL2113128 IC50 300.0 nM
Cc1ccc(S(=O)(=O)n2cc(-c3ccc(C(F)(F)F)cc3)c3ccc(CO[C@H](C(=O)O)[C@H](N)C(=O)O)cc32)cc1 CHEMBL4790691 pIC50 309.03 nM
Cc1cc(-c2cccc(C(F)(F)F)c2)ccc1NC(=O)C[C@H](N)C(=O)O CHEMBL2113123 IC50 400.0 nM
N[C@H](C(=O)O)[C@H](OCC1CCCCC1)C(=O)O CHEMBL4164207 pIC50 489.78 nM
Cc1ccc(NC(=O)CC(N)C(=O)O)cc1-c1ccc(F)c(Cl)c1 CHEMBL373283 IC50 500.0 nM
N[C@@H](CC(=O)Nc1ccc2oc3cc(F)c(F)cc3c2c1)C(=O)O CHEMBL2113120 IC50 500.0 nM
N[C@H](C(=O)O)C(NS(=O)(=O)c1ccc(-c2ccccc2)cc1)C(=O)O CHEMBL3939524 IC50 500.0 nM
CCc1cc(-c2ccc(F)c(Cl)c2)ccc1NC(=O)C[C@H](N)C(=O)O CHEMBL2113111 IC50 600.0 nM
N[C@H](C(=O)O)[C@H](OCC1CCC1)C(=O)O CHEMBL4173825 IC50 690.0 nM
Cc1ccc(NC(=O)C[C@H](N)C(=O)O)cc1-c1cccc(C(F)(F)F)c1 CHEMBL2113114 IC50 700.0 nM
NC(CC(=O)Nc1ccc(-c2ccccc2)cc1)C(=O)O CHEMBL198315 IC50 700.0 nM
N[C@@H](CC(=O)Nc1ccc2c(c1)Cc1ccccc1-2)C(=O)O CHEMBL1628570 IC50 700.0 nM
N[C@H](C(=O)O)[C@H](OCc1ccoc1)C(=O)O CHEMBL4177165 pIC50 758.58 nM
N[C@H](C(=O)O)[C@H](OCc1cccs1)C(=O)O CHEMBL4163105 IC50 770.0 nM
N[C@H](C(=O)O)[C@H](OCc1ccco1)C(=O)O CHEMBL4166545 IC50 830.0 nM
N[C@H](C(=O)O)[C@H](OCc1ccsc1)C(=O)O CHEMBL4169695 IC50 920.0 nM
N[C@H](C(=O)O)[C@H](OCC1CCCC1)C(=O)O CHEMBL4165574 pIC50 933.25 nM
N[C@H](C(=O)O)[C@H](OCc1ccccc1)C(=O)O CHEMBL79140 pIC50 954.99 nM
N[C@@H](CC(=O)Nc1c(F)c(F)c(-c2cccc(C(F)(F)F)c2)c(F)c1F)C(=O)O CHEMBL2113127 IC50 1000.0 nM
N[C@@H](CC(=O)Nc1ccc(Cc2ccccc2)cc1)C(=O)O CHEMBL2113129 IC50 1000.0 nM