N#Cc1cc(Oc2cc(F)c(S(=O)(=O)Nc3ncccn3)cc2Cl)ccc1F CHEMBL3688167 IC50 0.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(CO)c(Cl)c1 CHEMBL3688197 IC50 1.0 nM
O=S(=O)(Nc1ccc(F)cn1)c1ccc(Oc2cnc(CO)c(Cl)c2)cc1F CHEMBL3688190 IC50 2.0 nM
N#Cc1ccc(-c2cnccc2NS(=O)(=O)C(F)(F)F)cc1 CHEMBL4087516 IC50 2.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(Cl)c(C#N)c(Cl)c1 CHEMBL3688192 IC50 3.0 nM
N#Cc1c(Cl)cc(NS(=O)(=O)c2ccccc2OC(F)(F)F)cc1Cl CHEMBL5414132 IC50 4.0 nM
N#Cc1ccc(NS(=O)(=O)c2ccccc2OC(F)(F)F)cc1Cl CHEMBL5399348 IC50 6.0 nM
O=S(=O)(Nc1cnc2ccccc2c1)c1ccccc1C(F)(F)F CHEMBL3971610 IC50 7.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc(C)c1C#N CHEMBL3683365 IC50 7.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)c(C#N)c(Cl)c1 CHEMBL3688188 IC50 8.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(CCC(=O)O)ccc12 CHEMBL3692018 IC50 10.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(Cc3n[nH]c(=S)o3)ccc12 CHEMBL3692028 IC50 10.0 nM
N#Cc1ccc(-c2cnccc2NS(=O)(=O)C(F)(F)F)c2ccccc12 CHEMBL4088988 IC50 10.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3683287 IC50 12.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(Cl)cn3)cc2C#N)cc1Cl CHEMBL3688185 IC50 12.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(Cc3nnn[nH]3)ccc12 CHEMBL3692025 IC50 13.0 nM
Cc1cn(Cc2c(Cl)cccc2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3691994 IC50 15.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(F)(F)C(=O)O)ccc12 CHEMBL3692056 IC50 15.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3cc(F)ccn3)cc2C#N)cc1Cl CHEMBL3683388 IC50 15.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(CCCC(=O)O)ccc12 CHEMBL3692024 IC50 16.0 nM
Cc1nn(Cc2c(Cl)cccc2C2CC2)c2cc(CCC(=O)O)ccc12 CHEMBL3692057 IC50 17.0 nM
N#Cc1ccc(NS(=O)(=O)c2ccccc2C(F)(F)F)cc1Cl CHEMBL3902309 IC50 18.0 nM
N#Cc1cc(NS(=O)(=O)c2ccccc2C(F)(F)F)ccc1Cl CHEMBL3899557 IC50 18.0 nM
Cc1cccc(C)c1CN1CC(C)(C)c2ccc(CC(=O)O)cc21 CHEMBL3691993 IC50 18.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3692003 IC50 18.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)c(Cl)c1 CHEMBL3683364 IC50 19.0 nM
COC(=O)C(Sc1nnc(Br)n1-c1ccc(Br)c2ccccc12)C(=O)OC CHEMBL5396351 IC50 19.7 nM
N#Cc1cc(NS(=O)(=O)c2ccccc2OC(F)(F)F)ccc1Cl CHEMBL3947681 IC50 20.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)c(F)c2)cc(C)c1C#N CHEMBL3948311 IC50 21.0 nM
CCc1oc2ccccc2c1C(=O)c1cc(Br)c(O)c(Br)c1 CHEMBL388590 IC50 22.0 nM
Cc1cccc(C)c1Cn1cc(C)c2ccc(CC(=O)O)cc21 CHEMBL3691988 IC50 22.0 nM
CC(C)(Sc1ccncc1-c1ccc(C#N)c2ccccc12)C(=O)O CHEMBL3707347 IC50 23.0 nM
N#Cc1c(Cl)cccc1NS(=O)(=O)c1ccccc1C(F)(F)F CHEMBL3978281 IC50 23.0 nM
Cc1cn(Cc2c(Cl)cccc2Cl)c2cc(CCC(=O)O)ccc12 CHEMBL3692000 IC50 23.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(CCc3nnn[nH]3)ccc12 CHEMBL3692026 IC50 23.0 nM
Cc1cccc(C)c1CN1CC(C)c2ccc(CC(=O)O)cc21 CHEMBL3691992 IC50 24.0 nM
CCc1nn(Cc2c(Cl)cccc2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3692031 IC50 24.0 nM
COc1cccc(C)c1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683399 IC50 24.0 nM
COc1ncc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3683356 IC50 25.0 nM
CCc1nn(Cc2c(Cl)cccc2Cl)c2cc(CCC(=O)O)ccc12 CHEMBL3692035 IC50 26.0 nM
N#Cc1cc(Cl)cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683348 IC50 27.0 nM
COc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc1Cl CHEMBL3683357 IC50 27.0 nM
Cc1cn(Cc2c(F)cccc2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3691997 IC50 28.0 nM
N#Cc1ccc(NS(=O)(=O)c2ccccc2C(F)(F)F)cc1C(F)(F)F CHEMBL3900479 IC50 29.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)c(F)c2)cc1F CHEMBL3683383 IC50 29.0 nM
Cc1cccc(C)c1Cn1cc(Cl)c2ccc(CC(=O)O)cc21 CHEMBL3691990 IC50 30.0 nM
Cc1nn(Cc2csc3ccc(Cl)cc23)c2cc(CCC(=O)O)ccc12 CHEMBL3692019 IC50 31.0 nM
N#Cc1cc(NS(=O)(=O)c2ccccc2C(F)(F)F)ccc1C(F)(F)F CHEMBL3973326 IC50 32.0 nM
O=S(=O)(CSc1nnc(Br)n1Cc1ccc(Br)c2ccccc12)Nc1cccnc1 CHEMBL4546569 IC50 32.0 nM
O=C(O)C1(Sc2ccnc3ccc(Br)cc23)CCC1 CHEMBL3746329 IC50 33.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(Cc3n[nH]c(=O)o3)ccc12 CHEMBL3692027 IC50 34.0 nM
O=S(=O)(Nc1cncc(Br)c1)c1ccccc1C(F)(F)F CHEMBL3984949 IC50 35.0 nM
CCc1nn(Cc2c(C)cccc2C)c2cc(C(=O)O)ccc12 CHEMBL3692033 IC50 35.0 nM
O=C([O-])CSc1nnc(Br)n1Cc1cccs1 CHEMBL5422088 IC50 35.0 nM
O=S(=O)(Nc1cncc(C(F)(F)F)c1)c1ccccc1C(F)(F)F CHEMBL3929544 IC50 36.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cncc(Cl)c1 CHEMBL3683481 IC50 37.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(C#N)c(C2CC2)c1 CHEMBL3683482 IC50 37.0 nM
O=C(c1cc(Cl)c(O)c(Cl)c1)N1CS(=O)(=O)c2ccccc21 CHEMBL4594446 IC50 37.2 nM
COc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1F CHEMBL3683416 IC50 38.0 nM
N#Cc1ccc(NS(=O)(=O)c2ccccc2C(F)(F)F)c(Cl)c1 CHEMBL3979882 IC50 39.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc1C#N CHEMBL3683347 IC50 39.0 nM
COc1cc(F)c(F)cc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683428 IC50 40.0 nM
Cc1nn(Cc2cccc(Cl)c2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3692004 IC50 41.0 nM
Cc1cccc(C)c1Cn1nc(C)c2ccc(CCC(=O)O)cc21 CHEMBL3692017 IC50 41.0 nM
CCc1oc2ccc(OC)cc2c1C(=O)c1cc(Br)c(O)c(Br)c1 CHEMBL1767106 IC50 42.0 nM
O=S(=O)(Nc1ccc(C(F)(F)F)nc1)c1ccccc1C(F)(F)F CHEMBL3924161 IC50 42.0 nM
CCc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(=O)O)ccc12 CHEMBL3692034 IC50 42.0 nM
CCc1cn(Cc2c(C)cccc2C)c2cc(C(=O)O)ccc12 CHEMBL3692001 IC50 43.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)c(F)c1 CHEMBL3683363 IC50 43.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc1F CHEMBL3683425 IC50 43.0 nM
Cc1cccc(C)c1Cn1cc(C)c2ccc(C(=O)O)cc21 CHEMBL3691987 IC50 46.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(F)c1 CHEMBL3683297 IC50 47.0 nM
O=C(O)Cc1ccc2c(C3CC3)nn(Cc3c(Cl)cccc3Cl)c2c1 CHEMBL3692038 IC50 49.0 nM
CCc1nn(Cc2c(C)cccc2C)c2cc(CC(=O)O)ccc12 CHEMBL3692032 IC50 50.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(Cl)cc1F CHEMBL3683333 IC50 50.0 nM
Cc1cccc(C)c1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683436 IC50 50.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)c(F)c1Cl CHEMBL3683451 IC50 50.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)c(F)c1F CHEMBL3683441 IC50 51.0 nM
Cc1cccc(Cl)c1Cn1nc(C)c2ccc(CC(=O)O)cc21 CHEMBL3692005 IC50 52.0 nM
CCc1nn(Cc2c(Cl)cccc2Cl)c2cc(-c3nnn[nH]3)cnc12 CHEMBL3692050 IC50 52.0 nM
CCc1nn(Cc2c(Cl)cccc2Cl)c2cc(-c3nnn[nH]3)ccc12 CHEMBL3692055 IC50 52.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1F CHEMBL3683329 IC50 53.0 nM
Cc1cn(Cc2cccc(Cl)c2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3691995 IC50 53.0 nM
CCc1nn(Cc2c(Cl)cccc2Cl)c2cc(/C=C/C(=O)O)ccc12 CHEMBL3692036 IC50 53.0 nM
Cc1cccc(C)c1Cn1nc(Cl)c2ccc(C(=O)O)cc21 CHEMBL3692039 IC50 53.0 nM
COc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3683432 IC50 53.0 nM
COc1ccc(C)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683479 IC50 53.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cnc(OC(F)F)c(Cl)c1 CHEMBL3688184 IC50 53.0 nM
Cc1nn(Cc2csc3ccc(Cl)cc23)c2cc(CC(=O)O)ccc12 CHEMBL3692007 IC50 55.0 nM
Cc1nn(Cc2c(Cl)cccc2C2CC2)c2cc(-c3nnn[nH]3)cnc12 CHEMBL3692047 IC50 55.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)c(Cl)c1Cl CHEMBL3683324 IC50 55.0 nM
N#Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc1F CHEMBL3683305 IC50 57.0 nM
Cc1cc(Cl)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1C#N CHEMBL3683312 IC50 57.0 nM
COc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc1C#N CHEMBL3683362 IC50 57.0 nM
O=C(c1cc(Br)c(O)c(Br)c1)N1CCOc2ccncc21 CHEMBL4640580 Ki 57.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3nccs3)cc2C#N)cc1Cl CHEMBL3966948 IC50 58.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(Cl)c(F)cc1Cl CHEMBL3683391 IC50 58.0 nM
O=C(O)C1(Sc2ccnc3ccc(C(F)(F)F)cc23)CCC1 CHEMBL3746480 IC50 61.2 nM
N#Cc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(F)c(Cl)c3)c(C#N)c2)nc1 CHEMBL3688183 IC50 62.0 nM
Cc1ccc(C)c(Cn2cc(C)c3ccc(CC(=O)O)cc32)c1 CHEMBL3691996 IC50 63.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)cc1F CHEMBL3683293 IC50 64.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(=O)O)ccc12 CHEMBL3692015 IC50 65.0 nM
Cc1cccc(C)c1Cn1nc(C)c2ccc(CC(=O)O)cc21 CHEMBL3691989 IC50 67.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(=O)CCC(=O)O)ccc12 CHEMBL3692022 IC50 68.0 nM
COc1cccc(Cl)c1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683398 IC50 69.0 nM
N#Cc1ccc(Cl)c(NS(=O)(=O)c2ccccc2C(F)(F)F)c1 CHEMBL3950939 IC50 71.0 nM
Cc1cccc(C)c1Cn1cc(C(C)C)c2ccc(C(=O)O)cc21 CHEMBL3692002 IC50 71.0 nM
Cc1nn(Cc2c(Cl)cccc2C#N)c2cc(CCC(=O)O)ccc12 CHEMBL3692020 IC50 72.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1 CHEMBL3683299 IC50 74.0 nM
COc1cccc(F)c1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683395 IC50 74.0 nM
COc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(C)c1 CHEMBL3683480 IC50 74.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(C)C(=O)O)ccc12 CHEMBL3692011 IC50 75.0 nM
COc1ccccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683426 IC50 75.0 nM
Cc1cccc(C)c1Cn1nc(C(C)C)c2ccc(CC(=O)O)cc21 CHEMBL3692037 IC50 76.0 nM
Cc1cccc(C)c1CN1CCc2ccc(CC(=O)O)cc21 CHEMBL3691991 IC50 77.0 nM
Cc1nn(Cc2cccc3ccccc23)c2cc(CC(=O)O)ccc12 CHEMBL3692008 IC50 77.0 nM
N#Cc1cc(F)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1F CHEMBL3683358 IC50 77.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)cc1Cl CHEMBL3683317 IC50 78.0 nM
COc1cc(Cl)ccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683427 IC50 79.0 nM
CCc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(=O)O)cnc12 CHEMBL3692048 IC50 80.0 nM
CCc1nn(Cc2c(C)cccc2Cl)c2cc(C(=O)O)cnc12 CHEMBL3692049 IC50 80.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc1Cl CHEMBL3683320 IC50 80.0 nM
Cc1ccc(Cl)cc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683325 IC50 80.0 nM
Cc1ccc(CC(=O)O)cc1OCc1c(C)cccc1C CHEMBL4096685 IC50 80.0 nM
N#Cc1ccc(NS(=O)(=O)c2ccccc2Cl)cc1Cl CHEMBL3960689 IC50 81.0 nM
N#Cc1cc(NS(=O)(=O)c2ccccc2Cl)ccc1Cl CHEMBL3933221 IC50 81.0 nM
CCc1cc2c(C(=O)c3cc(Br)c(O)c(Br)c3)c(O)ccc2o1 CHEMBL1767109 IC50 83.0 nM
O=S(=O)(Nc1ccnc2ccc(Br)cc12)C(F)(F)F CHEMBL4100597 IC50 83.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(Cl)cc1Cl CHEMBL3683298 IC50 84.0 nM
Cc1ccc(F)cc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683307 IC50 84.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cccc(Cl)c1 CHEMBL3683311 IC50 86.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cnc(N)c(Cl)c1 CHEMBL3688196 IC50 87.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2)cc1F CHEMBL3893511 IC50 88.0 nM
Cc1cn(Cc2ccccc2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3691998 IC50 88.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(Cl)cc1 CHEMBL3683306 IC50 88.0 nM
Cc1ncc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3688189 IC50 88.0 nM
Cc1ccccc1S(=O)(=O)Nc1ccc(C#N)c(Cl)c1 CHEMBL3971816 IC50 89.0 nM
COc1cncc(NS(=O)(=O)c2ccccc2C(F)(F)F)c1 CHEMBL3892944 IC50 89.0 nM
Cc1ccc(F)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1F CHEMBL3683403 IC50 90.0 nM
Cc1cccc(C)c1Cn1nc(C)c2ccc(C(=O)O)cc21 CHEMBL3692014 IC50 91.0 nM
Cc1nn(Cc2cccc(Cl)c2Cl)c2cc(C(=O)O)ccc12 CHEMBL3692016 IC50 91.0 nM
Cc1cccc(Cl)c1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683407 IC50 91.0 nM
N#Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc1Cl CHEMBL3683346 IC50 92.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)cc(Cl)c1 CHEMBL3683314 IC50 92.0 nM
Cc1cc(C)c(Cn2nc(C)c3ccc(CC(=O)O)cc32)c(C)c1 CHEMBL3692009 IC50 94.0 nM
O=C([O-])CSc1nnc(Br)n1Cc1ccc(Br)c2ccccc12 CHEMBL4453888 IC50 94.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc(C)c1Cl CHEMBL3683433 IC50 95.0 nM
Cc1cc(F)ccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683429 IC50 96.0 nM
Cc1cn(Cc2cc3c(cc2Cl)OCO3)c2cc(CC(=O)O)ccc12 CHEMBL3691999 IC50 98.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(C)(C)C(=O)O)ccc12 CHEMBL3692012 IC50 98.0 nM
Cc1ccc(F)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1Cl CHEMBL3683392 IC50 98.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(Cl)c(Cl)c1 CHEMBL3683406 IC50 99.0 nM
Cc1nn(Cc2c(F)cccc2Cl)c2cc(CC(=O)O)ccc12 CHEMBL3692006 IC50 101.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccccc1Br CHEMBL3683471 IC50 103.0 nM
Cc1cccc(Cl)c1Cn1nc(Cl)c2ncc(-c3nnn[nH]3)cc21 CHEMBL3692054 IC50 104.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccccn3)cc2C#N)cc1Cl CHEMBL3683373 IC50 105.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(Cl)c(CO)c1 CHEMBL3688191 IC50 106.0 nM
CCc1ccccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683332 IC50 107.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3cscn3)cc2C#N)cc1Cl CHEMBL3937205 IC50 110.0 nM
CCc1oc2cc(OC)ccc2c1C(=O)c1cc(Br)c(O)c(Br)c1 CHEMBL1767112 IC50 111.0 nM
N#Cc1cc(Cl)ccc1NS(=O)(=O)c1ccccc1C(F)(F)F CHEMBL3890592 IC50 111.0 nM
Cc1ccc(C)c(Cn2nc(C)c3ncc(-c4nnn[nH]4)cc32)c1 CHEMBL3692046 IC50 113.0 nM
O=C(O)C1(Sc2ccnc3ccc(-c4ccccc4C(F)(F)F)cc23)CCC1 CHEMBL3747573 IC50 115.3 nM
COc1ccc(F)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683450 IC50 116.0 nM
Cc1ccc(F)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683319 IC50 117.0 nM
N#Cc1ccc(NS(=O)(=O)c2ccccc2C(F)(F)F)cc1 CHEMBL3944865 IC50 119.0 nM
COc1cc(F)cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683294 IC50 119.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)c(F)cc1F CHEMBL3683414 IC50 119.0 nM
Cc1ccc(C)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683442 IC50 122.0 nM
CCOc1cc(Cl)ccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683394 IC50 123.0 nM
Cc1cccc(Cl)c1Cn1nc(C)c2ncc(-c3nnn[nH]3)cc21 CHEMBL3692045 IC50 124.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)cc(F)c1 CHEMBL3683296 IC50 125.0 nM
COc1cc(Cl)cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683446 IC50 125.0 nM
N#Cc1ccnc(NS(=O)(=O)c2ccc(Oc3ccc(F)c(Cl)c3)c(C#N)c2)c1 CHEMBL3688182 IC50 126.0 nM
N#Cc1cc(NS(=O)(=O)c2ccccc2C#N)ccc1Cl CHEMBL3938886 IC50 127.0 nM
N#Cc1ccc(-c2cnccc2NS(=O)(=O)c2ccccc2)c2ccccc12 CHEMBL4104410 IC50 127.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(Cl)c(F)c1 CHEMBL3683341 IC50 129.0 nM
COc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cn1 CHEMBL3683478 IC50 129.0 nM
O=C(O)C1(Sc2ccnc3cc(Br)ccc23)CCC1 CHEMBL3745847 IC50 129.8 nM
Cc1ccc(Cc2nnn[nH]2)cc1OCc1c(C)cccc1C CHEMBL3702600 IC50 130.0 nM
COc1c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)ccc(F)c1C CHEMBL3683457 IC50 131.0 nM
Cc1ccc(Cl)c(C)c1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683453 IC50 134.0 nM
Cc1cc(Cl)cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683301 IC50 135.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cccc(Cl)c1F CHEMBL3683310 IC50 135.0 nM
COc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1C#N CHEMBL3683352 IC50 135.0 nM
CCc1oc2cc(O)ccc2c1C(=O)c1cc(Br)c(O)c(Br)c1 CHEMBL1767079 IC50 138.0 nM
COc1c(F)ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1C CHEMBL3683449 IC50 139.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cccc(Cl)c1Cl CHEMBL3683289 IC50 141.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ncccc3F)cc2C#N)cc1Cl CHEMBL3683387 IC50 145.0 nM
Cc1cccc(Cl)c1Cn1nc(Cl)c2ncc(C(=O)O)cc21 CHEMBL3692052 IC50 148.0 nM
Cc1cc(Cl)ccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683291 IC50 148.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cnc(C#N)c(Cl)c1 CHEMBL3683354 IC50 155.0 nM
N#Cc1ccc(NS(=O)(=O)c2ccccc2C#N)cc1Cl CHEMBL3920396 IC50 156.0 nM
O=C(O)C1(Sc2ccnc3ccc(-c4ccc(F)cc4)cc23)CCC1 CHEMBL3745776 IC50 158.8 nM
O=C(O)c1cnc2c(Cl)nn(Cc3c(Cl)cccc3Cl)c2c1 CHEMBL3692051 IC50 162.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccccc1F CHEMBL3683327 IC50 162.0 nM
Clc1cccc(Cl)c1Cn1nc(Cl)c2ncc(-c3nnn[nH]3)cc21 CHEMBL3692053 IC50 163.0 nM
Cc1cccc(C)c1Cn1c(=O)n(C(C)C)c2ccc(C(=O)O)cc21 CHEMBL3692058 IC50 165.0 nM
N#Cc1cccc(NS(=O)(=O)c2ccccc2C(F)(F)F)c1 CHEMBL3965811 IC50 166.0 nM
COc1ccc(Cl)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683330 IC50 167.0 nM
CC(C)(Sc1ccncc1-c1ccc(C#N)c2ccccc12)C(=O)[O-] CHEMBL5170470 IC50 170.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccccc1C(F)(F)F CHEMBL3683337 IC50 171.0 nM
N#Cc1cc(Cl)ccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683331 IC50 174.0 nM
COc1cc(C)cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683466 IC50 175.0 nM
CCc1cc2c(C(=O)c3cc(Br)c(O)c(Br)c3)cc(Br)c(O)c2o1 CHEMBL1767114 IC50 177.0 nM
COc1c(F)ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1Cl CHEMBL3683396 IC50 177.0 nM
CCc1cc(F)ccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683342 IC50 182.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(Cl)ccc1C#N CHEMBL3683351 IC50 182.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(Cl)c1 CHEMBL3683316 IC50 183.0 nM
Cc1ccccc1S(=O)(=O)Nc1ccc(Cl)c(C#N)c1 CHEMBL3942205 IC50 183.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)cc1 CHEMBL3683467 IC50 183.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2nc(Cc3nnn[nH]3)ccc12 CHEMBL3692041 IC50 184.0 nM
Cc1cncc(NS(=O)(=O)c2ccccc2C(F)(F)F)c1 CHEMBL3983987 IC50 185.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(CCC(N)=O)ccc12 CHEMBL3692023 IC50 186.0 nM
N#Cc1ccc(Cl)cc1NS(=O)(=O)c1ccccc1C(F)(F)F CHEMBL3923480 IC50 187.0 nM
Cc1c(F)ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1Cl CHEMBL3683431 IC50 187.0 nM
CCc1oc2ccc(O)cc2c1C(=O)c1cc(Br)c(O)c(Br)c1 CHEMBL1767107 IC50 189.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)ccc1F CHEMBL3683339 IC50 191.0 nM
COc1ccc(C)cc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683439 IC50 191.0 nM
Cc1ccc(Cl)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683323 IC50 196.0 nM
COCc1ccc2nccc(SC3(C(=O)O)CCC3)c2c1 CHEMBL3746658 IC50 197.8 nM
COc1ccccc1S(=O)(=O)Nc1ccc(C#N)c(Cl)c1 CHEMBL3919891 IC50 199.0 nM
CS(=O)(=O)Nc1ccncc1-c1ccc(C#N)cc1 CHEMBL4103898 IC50 203.0 nM
N#Cc1cccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683300 IC50 206.0 nM
COCCOc1ccc2nccc(SC3(C(=O)O)CCC3)c2c1 CHEMBL3746426 IC50 206.9 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccccc1Cl CHEMBL3683295 IC50 208.0 nM
Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3683308 IC50 209.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)cc(F)c1Cl CHEMBL3683318 IC50 212.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc(Cl)c1C CHEMBL3683455 IC50 215.0 nM
COc1ccc(-c2cnccc2NS(=O)(=O)C(F)(F)F)cc1 CHEMBL4066146 IC50 215.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cccc(F)c1F CHEMBL3683302 IC50 218.0 nM
O=C([O-])CCCc1nnc(Br)n1Cc1ccc(Br)c2ccccc12 CHEMBL5433470 IC50 230.0 nM
Cc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(C#N)c(Cl)c3)c(C#N)c2)nc1 CHEMBL3688186 IC50 233.0 nM
CCOc1ncc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3683409 IC50 237.0 nM
Cc1cccc(C)c1COc1cccc(Cc2nnn[nH]2)c1 CHEMBL3702597 IC50 240.0 nM
N#Cc1ccc(Nc2cnccc2SCc2ccccc2C(=O)[O-])c2ccccc12 CHEMBL5202967 IC50 240.0 nM
N#Cc1cc(F)ccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683322 IC50 241.0 nM
COc1ccccc1-c1cnccc1NS(=O)(=O)C(F)(F)F CHEMBL4079640 IC50 241.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2Cl)cc1F CHEMBL3688181 IC50 244.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)c(F)cc1Cl CHEMBL3683461 IC50 246.0 nM
COc1ccc(Cc2nnn[nH]2)cc1OCc1c(C)cccc1C CHEMBL3702598 IC50 250.0 nM
CNc1ncc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3688194 IC50 258.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cccc(F)c1 CHEMBL3683338 IC50 259.0 nM
CS(=O)(=O)Nc1ccncc1-c1ccc(C#N)c2ccccc12 CHEMBL4078667 IC50 261.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(C#N)c(C(F)(F)F)c1 CHEMBL3683292 IC50 267.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccccc1OC(F)(F)F CHEMBL3683313 IC50 274.0 nM
O=S(=O)(CSc1nnc(Br)n1Cc1ccc(Br)c2ccccc12)Nc1cccnc1Br CHEMBL4458898 IC50 280.0 nM
CCc1cc2cc(O)cc(C(=O)c3cc(Br)c(O)c(Br)c3)c2o1 CHEMBL1767111 IC50 287.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(Cl)cc1I CHEMBL3683344 IC50 287.0 nM
Cc1nn(Cc2cccc(Cl)c2Cl)c2cc(-c3nnn[nH]3)cnc12 CHEMBL3692044 IC50 292.0 nM
[C-]#[N+]c1nn(Cc2c(Cl)cccc2Cl)c2cc(C(=O)O)ccc12 CHEMBL3692040 IC50 295.0 nM
N#Cc1ccc(Cl)c(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683349 IC50 321.0 nM
Cc1ccccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683468 IC50 324.0 nM
N#Cc1ccc(Oc2c(F)cc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3688198 IC50 324.0 nM
O=C(O)C1(Sc2ccnc3ccc(Br)cc23)CCCC1 CHEMBL3747526 IC50 324.3 nM
Cc1cc(C)cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1 CHEMBL3683434 IC50 329.0 nM
O=C(O)C1(Sc2ccnc3ccc(-c4ccccc4F)cc23)CCC1 CHEMBL3747053 IC50 333.4 nM
Cc1nn(Cc2c(Cl)cccc2C#N)c2cc(CC(=O)O)ccc12 CHEMBL3692010 IC50 335.0 nM
COc1ccc2nccc(SC3(C(=O)O)CCC3)c2c1 CHEMBL3746049 IC50 342.8 nM
Cc1ccc2nccc(SC3(C(=O)O)CCC3)c2c1 CHEMBL3746315 IC50 343.2 nM
O=C(O)C1(Sc2ccnc3ccc(Br)cc23)CC1 CHEMBL3747024 IC50 352.3 nM
CCc1cc2c(C(=O)c3cc(Br)c(O)c(Br)c3)c(OC)ccc2o1 CHEMBL1767108 IC50 358.0 nM
O=C(O)C1(Sc2ccnc3ccc(-c4cccc(C(F)(F)F)c4)cc23)CCC1 CHEMBL3747747 IC50 358.7 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(=O)O)cnc12 CHEMBL3692042 IC50 361.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2F)cc1F CHEMBL3683381 IC50 382.0 nM
Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(Cl)c1 CHEMBL3683328 IC50 383.0 nM
Cc1ncccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3639823 IC50 385.0 nM
N#Cc1ccc(-c2cnccc2NS(=O)(=O)c2ccccc2)cc1 CHEMBL4074756 IC50 390.0 nM
O=C(Nc1ccc(-c2nnn[nH]2)cc1)c1c(O)[nH]c(=S)[nH]c1=O CHEMBL5400912 IC50 390.0 nM
Cc1nn(Cc2cccc3cccnc23)c2cc(CC(=O)O)ccc12 CHEMBL3692013 IC50 394.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3cccnc3)cc2C#N)cc1Cl CHEMBL3683376 IC50 395.0 nM
N#Cc1ccc2nccc(SC3(C(=O)O)CCC3)c2c1 CHEMBL3747493 IC50 398.8 nM
COc1cc(Cl)ccc1Oc1ccc(S(=O)(=O)Nc2cccnc2)cc1C#N CHEMBL3977539 IC50 409.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1c(Cl)cccc1C#N CHEMBL3683359 IC50 418.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3nncs3)cc2C#N)cc1Cl CHEMBL3975435 IC50 426.0 nM
N#Cc1ccc(Oc2ccc(S(=O)(=O)Nc3cccnn3)cc2C#N)cc1F CHEMBL3683372 IC50 429.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(-c3nnn[nH]3)cnc12 CHEMBL3692043 IC50 438.0 nM
O=C(O)C1(Sc2ccnc3ccccc23)CCC1 CHEMBL3747343 IC50 448.0 nM
Cc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(C)c1Cl CHEMBL3683459 IC50 455.0 nM
COc1cc(C(=O)[O-])ccc1CSc1ccncc1N(C)c1ccc(C#N)c2ccccc12 CHEMBL5190525 IC50 460.0 nM
CN(C)c1ncc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)cc1Cl CHEMBL3688195 IC50 472.0 nM
O=S(=O)(Nc1ccc(F)c(C(F)(F)F)c1)c1ccccc1C(F)(F)F CHEMBL3893319 IC50 484.0 nM
N#Cc1ccccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683303 IC50 495.0 nM
Cc1c(F)ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1C CHEMBL3683456 IC50 502.0 nM
CSc1ccccc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683430 IC50 506.0 nM
Cc1cc(Cl)cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c1C CHEMBL3683443 IC50 514.0 nM
O=C(O)C1(Sc2ccnc3ccc(F)cc23)CCC1 CHEMBL3746433 IC50 557.6 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(Cl)ccc1Cl CHEMBL3683454 IC50 570.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(C(O)C(=O)O)ccc12 CHEMBL3692021 IC50 576.0 nM
Cc1cccnc1NS(=O)(=O)c1ccc(Oc2ccc(C#N)c(Cl)c2)c(C#N)c1 CHEMBL3683385 IC50 594.0 nM
CC(C)CS(=O)(=O)Nc1ccncc1-c1ccc(C#N)c2ccccc12 CHEMBL4094280 IC50 597.0 nM
COc1ccc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(Cl)c1 CHEMBL3683452 IC50 612.0 nM
N#Cc1ccccc1NS(=O)(=O)c1ccccc1C(F)(F)F CHEMBL3935920 IC50 616.0 nM
O=C(CSc1nnc(Br)n1Cc1ccc(Br)c2ccccc12)NO CHEMBL4468962 IC50 640.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(CS(=O)(=O)O)ccc12 CHEMBL3692030 IC50 653.0 nM
O=C(O)C1(Sc2ccnc3ccc(C4CC4)cc23)CCC1 CHEMBL3747353 IC50 659.2 nM
CCc1oc2c(Br)c(O)c(Br)cc2c1C(=O)c1ccc(OC)cc1 CHEMBL1767116 IC50 667.0 nM
N#CCOc1ccc2nccc(SC3(C(=O)O)CCC3)c2c1 CHEMBL3746317 IC50 680.2 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1ccc(F)c(C(F)(F)F)c1 CHEMBL3683334 IC50 683.0 nM
O=C(Nc1ccc(-c2cnn[nH]2)cc1)c1c(O)nc(O)[nH]c1=O CHEMBL5428787 IC50 690.0 nM
CCS(=O)(=O)Nc1ccncc1-c1ccc(C#N)c2ccccc12 CHEMBL4067774 IC50 713.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccccn2)ccc1Oc1ccc(Cl)cc1I CHEMBL3683366 IC50 728.0 nM
Cc1cccc(C)c1COc1cccc(CCc2nnn[nH]2)c1 CHEMBL3702599 IC50 740.0 nM
CCc1cc2c(C(=O)c3ccc(OC)cc3)cc(Br)c(O)c2o1 CHEMBL1767117 IC50 772.0 nM
Cc1ccncc1Oc1ccc(S(=O)(=O)Nc2ccc(F)cn2)cc1C#N CHEMBL3683477 IC50 792.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(C(C)C)cc1Cl CHEMBL3683417 IC50 793.0 nM
O=C(c1cc(Cl)c(O)c(Cl)c1)n1ccc2cccnc21 CHEMBL5439993 IC50 800.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cnc(C2CC2)c(Cl)c1 CHEMBL3683464 IC50 877.0 nM
Cc1cc(Oc2ccc(S(=O)(=O)Nc3ccc(F)cn3)cc2C#N)c(Cl)cc1Cl CHEMBL3683393 IC50 892.0 nM
Cc1nn(Cc2c(Cl)cccc2Cl)c2cc(OCC(=O)O)ccc12 CHEMBL3692029 IC50 916.0 nM
N#Cc1ccc(SC2(C(=O)O)CCC2)c2ccccc12 CHEMBL3747094 IC50 926.4 nM
Cc1cccc(C)c1COc1cccc(-c2nnn[nH]2)c1 CHEMBL3702596 IC50 930.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cc(F)cc(C(F)(F)F)c1 CHEMBL3683326 IC50 988.0 nM
N#Cc1cc(S(=O)(=O)Nc2ccc(F)cn2)ccc1Oc1cnc(N2CCC2)c(Cl)c1 CHEMBL3688193 IC50 1000.0 nM