O=C(c1ccc(-c2cccc(Cl)c2)cc1)N1C2CCC1CN(c1ncccn1)C2 CHEMBL3318586 IC50 18.0 nM
C[C@H]1CN(c2ncccn2)CCN1C(=O)c1ccc(-c2ccc(Cl)cc2)cc1 CHEMBL3318579 IC50 21.0 nM
CC1CN(c2ncccn2)CC(C)N1C(=O)c1ccc(-c2cccc(Cl)c2)cc1 CHEMBL3318574 IC50 24.0 nM
O=C(c1ccc(-c2cccc(Cl)c2)cc1)N1CC2CCC(C1)N2c1ncccn1 CHEMBL3318585 IC50 27.0 nM
Cc1csc(-c2ccc(C(=O)N3CCN(c4ncccn4)CC3)cc2)c1 CHEMBL3318563 IC50 34.0 nM
Cc1ccc(-c2ccc(C(=O)N3CCN(c4ncccn4)CC3)cc2)cc1 CHEMBL3318552 IC50 34.0 nM
O=C(c1ccc(-c2cccc(Cl)c2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318548 IC50 36.0 nM
O=C(c1ccc(-c2cccc(Cl)c2)cc1)N1CC2CN(c3ncccn3)CC2C1 CHEMBL3318584 IC50 36.0 nM
O=C(c1ccc(-c2ccc(Cl)cc2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3317462 IC50 52.0 nM
CC1(C)CN(c2ncccn2)CCN1C(=O)c1ccc(-c2cccc(Cl)c2)cc1 CHEMBL3318573 IC50 53.0 nM
C[C@@H]1CN(c2ncccn2)CCN1C(=O)c1ccc(-c2ccc(Cl)cc2)cc1 CHEMBL3318580 IC50 57.0 nM
Cc1ccc(-c2ccc(C(=O)N3CCN(c4ncccn4)CC3)cc2)s1 CHEMBL3318564 IC50 61.0 nM
O=C(c1ccc(-c2cccc(C(F)(F)F)c2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318549 IC50 71.0 nM
O=C(c1ccc(-c2cccc(OC(F)(F)F)c2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318550 IC50 73.0 nM
O=C(c1ccc(-c2ccc(C(F)(F)F)cc2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318554 IC50 76.0 nM
O=C(c1ccc(-c2cccc(Cl)c2)cc1)N1CCN(c2ncccn2)CC1CO CHEMBL3318576 IC50 76.0 nM
CCc1ccc(-c2ccc(C(=O)N3CCN(c4ncccn4)CC3)cc2)cc1 CHEMBL3318553 IC50 77.0 nM
O=C(c1ccc(-c2cccc(Cl)c2)cc1)N1CCCN(c2ncccn2)CC1 CHEMBL3318581 IC50 89.0 nM
O=C(O)C1CN(c2ncccn2)CCN1C(=O)c1ccc(-c2cccc(Cl)c2)cc1 CHEMBL3318577 IC50 128.0 nM
O=C(c1ccc(-c2ccccc2)cc1)N1CCN(c2nccs2)CC1 CHEMBL3318540 IC50 146.0 nM
O=C(c1ccc(-c2ccc(Cl)s2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318562 IC50 150.0 nM
O=C(c1ccc(-c2ccccc2)cc1)N1CCN(c2ccccn2)CC1 CHEMBL1543754 IC50 160.0 nM
N#Cc1ccc(-c2ccc(C(=O)N3CCN(c4ncccn4)CC3)cc2)cc1 CHEMBL3318555 IC50 190.0 nM
N#Cc1cccc(-c2ccc(C(=O)N3CCN(c4ncccn4)CC3)cc2)c1 CHEMBL3318551 IC50 190.0 nM
COc1ccc(-c2ccc(C(=O)N3CCN(c4ncccn4)CC3)cc2)cc1 CHEMBL3318556 IC50 230.0 nM
O=C(c1ccc(-c2ccc(F)cc2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318557 IC50 260.0 nM
O=C(c1ccc(OCc2ccccc2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318567 IC50 270.0 nM
Cc1ccnc(N2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)n1 CHEMBL3318543 IC50 270.0 nM
O=C(c1ccc(-c2ccccc2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL1594803 IC50 280.0 nM
CN(C)C(=O)C1CN(c2ncccn2)CCN1C(=O)c1ccc(-c2cccc(Cl)c2)cc1 CHEMBL3318578 IC50 392.0 nM
CC1CN(C(=O)c2ccc(-c3ccccc3)cc2)CCN1c1ncccn1 CHEMBL3318575 IC50 477.0 nM
CN(CCN(C)c1ncccn1)C(=O)c1ccc(-c2cccc(Cl)c2)cc1 CHEMBL3318582 IC50 586.0 nM
Cc1ccccc1-c1ccc(C(=O)N2CCN(c3ncccn3)CC2)cc1 CHEMBL3318587 IC50 653.0 nM
CC(C)(C)C1CN(c2ncccn2)CCN1C(=O)c1ccc(-c2cccc(Cl)c2)cc1 CHEMBL3318572 IC50 700.0 nM
O=C(c1ccc(NCc2ccccc2)cc1)N1CCN(c2ncccn2)CC1 CHEMBL3318569 IC50 870.0 nM