Cc1ccccc1[C@@H]1CCc2cc(Oc3ncc(C(=O)NCCOP(=O)(O)O)s3)ccc2O1 CHEMBL3662020 IC50 70.0 nM
O=C(NCc1ccno1)c1csc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)n1 CHEMBL3662028 IC50 92.0 nM
NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3662043 IC50 100.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1cccnc1 CHEMBL3657666 IC50 100.0 nM
O=C(Cc1cccnc1)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657667 IC50 100.0 nM
O=C(Cc1ccccn1)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657670 IC50 100.0 nM
Cc1nccc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657672 IC50 100.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657675 IC50 100.0 nM
CN(C)c1cc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)ccn1 CHEMBL3657680 IC50 100.0 nM
O=C(NCc1ccncc1)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3657687 IC50 100.0 nM
O=C(Cc1cccnc1)NCc1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1 CHEMBL3657696 IC50 100.0 nM
O=S(=O)(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1cccnc1 CHEMBL3657698 IC50 100.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccno1 CHEMBL3657699 IC50 100.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1 CHEMBL3657700 IC50 100.0 nM
Cc1nc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)sc1C(=O)NCc1ccncc1 CHEMBL3657709 IC50 100.0 nM
O=C(NCc1ccncc1)c1cnc(Oc2ccc3c(c2)CCC(c2ccsc2)O3)s1 CHEMBL3657710 IC50 100.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCc5ccno5)s4)ccc3O2)cc1 CHEMBL3657801 IC50 100.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661858 IC50 100.0 nM
O=C(NCCO)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661888 IC50 100.0 nM
c1ccc([C@@H]2CCc3cc(Oc4ncc(CNCc5ccno5)s4)ccc3O2)cc1 CHEMBL3661894 IC50 100.0 nM
COC(=O)CNCc1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661925 IC50 100.0 nM
OCCNCc1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661945 IC50 100.0 nM
OCCNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661987 IC50 100.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)N(CCO)CCO CHEMBL3661988 IC50 100.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)N1CCOCC1 CHEMBL3661990 IC50 100.0 nM
CCCCNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661992 IC50 100.0 nM
CC(C)CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661993 IC50 100.0 nM
Cc1ccccc1[C@@H]1CCc2cc(Oc3ncc(C(=O)NCCO)s3)ccc2O1 CHEMBL3662001 IC50 100.0 nM
CCCNC(=O)c1csc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)n1 CHEMBL3662026 IC50 110.0 nM
O=C(NCCO)c1csc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)n1 CHEMBL3662025 IC50 120.0 nM
CC(O)CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3662029 IC50 160.0 nM
O=C(CN1CCCC1)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3662021 IC50 170.0 nM
COc1c(F)cccc1C1CCc2cc(Oc3ncc(C(=O)NCc4ccno4)s3)ccc2O1 CHEMBL3662041 IC50 180.0 nM
Nc1cc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3cccc(F)c3)O4)s2)ccn1 CHEMBL3657663 IC50 200.0 nM
O=C(NCc1nnc2ccccn12)c1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1 CHEMBL3657668 IC50 200.0 nM
O=C(NCc1ccncc1)c1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1 CHEMBL3657669 IC50 200.0 nM
O=C(NCc1nnc2n1CCC2)c1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1 CHEMBL3657671 IC50 200.0 nM
O=C(NCc1ccnc(N2CCOCC2)c1)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657679 IC50 200.0 nM
Cc1cc(C)nc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657684 IC50 200.0 nM
Cc1noc(C)c1CCNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657685 IC50 200.0 nM
O=C(NCc1ccncc1)c1cnc(Oc2ccc3c(c2)CC[C@H](c2ccccc2)O3)s1 CHEMBL3657688 IC50 200.0 nM
O=C(NCc1ccnc(O)c1)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657693 IC50 200.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1)c1cccnc1 CHEMBL3657695 IC50 200.0 nM
O=C(Cc1ccncc1)NCc1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1 CHEMBL3657697 IC50 200.0 nM
Cn1cnc(S(=O)(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)c1 CHEMBL3657701 IC50 200.0 nM
Cc1c(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3cccc(F)c3)O4)s2)cnn1C CHEMBL3657702 IC50 200.0 nM
C[C@H](NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1nccs1 CHEMBL3657705 IC50 200.0 nM
Cc1nccc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3cccc(F)c3)O4)s2)n1 CHEMBL3657707 IC50 200.0 nM
Cc1noc(C)c1C(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657714 IC50 200.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccncc1 CHEMBL3657727 IC50 200.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccncc1Cl CHEMBL3639565 IC50 200.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccncn1 CHEMBL3657735 IC50 200.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNC5CC5)s4)ccc3O2)cc1 CHEMBL3657748 IC50 200.0 nM
FC(F)(F)CNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657752 IC50 200.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNC5CCC5)s4)ccc3O2)cc1 CHEMBL3657754 IC50 200.0 nM
COCCNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657758 IC50 200.0 nM
CC(CN)Cc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657760 IC50 200.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCc5ccncc5)s4)ccc3O2)cc1 CHEMBL3657777 IC50 200.0 nM
Cc1cc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)no1 CHEMBL3657783 IC50 200.0 nM
Cn1nccc1CNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657789 IC50 200.0 nM
N#Cc1ccc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cn1 CHEMBL3657799 IC50 200.0 nM
Cc1cc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)on1 CHEMBL3657802 IC50 200.0 nM
Cc1nc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)sc1C(=O)NCc1ccno1 CHEMBL3661855 IC50 200.0 nM
CCOC(=O)[C@H](C)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661866 IC50 200.0 nM
COC(=O)CNC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661867 IC50 200.0 nM
C[C@H](O)[C@H](CO)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3639607 IC50 200.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CCC(c2cc(F)ccc2F)O3)s1 CHEMBL3661900 IC50 200.0 nM
OCCN(CCO)Cc1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661938 IC50 200.0 nM
N[C@H]1CC1NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661962 IC50 200.0 nM
COC(=O)CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661971 IC50 200.0 nM
Cc1ccccc1C1CCc2cc(Oc3ncc(C(=O)N4CC[C@@H](O)C4)s3)ccc2O1 CHEMBL3661977 IC50 200.0 nM
CC(C)OC(=O)CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661984 IC50 200.0 nM
CCOC(=O)CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3639608 IC50 200.0 nM
Cc1ccccc1[C@H]1CCc2cc(Oc3ncc(C(=O)NCCO)s3)ccc2O1 CHEMBL3662000 IC50 200.0 nM
Cc1ccc(F)cc1C1CCc2cc(Oc3ncc(C(=O)NCCN4CCNC4=O)s3)ccc2O1 CHEMBL3662024 IC50 200.0 nM
O=C(NCCN1CCNC1=O)c1csc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)n1 CHEMBL3662027 IC50 210.0 nM
O=C(NC1CCCC1O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3662030 IC50 250.0 nM
COc1c(F)cccc1C1CCc2cc(Oc3ncc(C(=O)NCCO)s3)ccc2O1 CHEMBL3662042 IC50 270.0 nM
CCn1cc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cn1 CHEMBL3657652 IC50 300.0 nM
O=C(NCc1nnc2n1CCC2)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657653 IC50 300.0 nM
O=C(NCc1ccncc1)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657655 IC50 300.0 nM
Cc1ncsc1CCNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657658 IC50 300.0 nM
CC(NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2)O3)s1)c1ccncc1 CHEMBL3657664 IC50 300.0 nM
Cc1c(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cnn1C CHEMBL3657665 IC50 300.0 nM
CN(Cc1ccnc(N2CCCC2)c1)C(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657677 IC50 300.0 nM
CC[C@@H](NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccc(OC)nc1 CHEMBL3657678 IC50 300.0 nM
O=C(NCc1ccncc1)c1sc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)nc1C(F)(F)F CHEMBL3657681 IC50 300.0 nM
Cc1noc(C)c1CCCNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657689 IC50 300.0 nM
O=C(NCc1ccnc(Cl)c1)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657690 IC50 300.0 nM
O=C(Cc1ccncc1)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657694 IC50 300.0 nM
Cc1c(CNC(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)cnn1C CHEMBL3657711 IC50 300.0 nM
Cc1nn(C)c(C)c1C(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657716 IC50 300.0 nM
CCn1nccc1C(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657719 IC50 300.0 nM
CCn1cc(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cn1 CHEMBL3657721 IC50 300.0 nM
Cc1nc(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cs1 CHEMBL3657722 IC50 300.0 nM
Cc1ccn(CC(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657723 IC50 300.0 nM
Cc1nc(C)c(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)o1 CHEMBL3657726 IC50 300.0 nM
Cc1cc(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)on1 CHEMBL3662047 IC50 300.0 nM
Cn1nccc1C(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657732 IC50 300.0 nM
Cc1nc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)sc1C(=O)NCc1ccncc1 CHEMBL3657743 IC50 300.0 nM
CCC(C)(C)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657756 IC50 300.0 nM
CC(C)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657757 IC50 300.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CN5CCOCC5)s4)ccc3O2)cc1 CHEMBL3657761 IC50 300.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCC5CC5)s4)ccc3O2)cc1 CHEMBL3657764 IC50 300.0 nM
Cn1nccc1S(=O)(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657771 IC50 300.0 nM
CCn1cc(S(=O)(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cn1 CHEMBL3657775 IC50 300.0 nM
Cc1c(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cnn1C CHEMBL3657781 IC50 300.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCCCn5cccn5)s4)ccc3O2)cc1 CHEMBL3657785 IC50 300.0 nM
Cc1cc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)nn1C CHEMBL3657790 IC50 300.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCCn5cccn5)s4)ccc3O2)cc1 CHEMBL3657792 IC50 300.0 nM
Cc1noc(C)c1CNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657794 IC50 300.0 nM
Oc1cc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)ccn1 CHEMBL3657796 IC50 300.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCc5cn6ccsc6n5)s4)ccc3O2)cc1 CHEMBL3657800 IC50 300.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCc5ccncn5)s4)ccc3O2)cc1 CHEMBL3657803 IC50 300.0 nM
Cc1nc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)sc1C(=O)NCc1ccno1 CHEMBL3661853 IC50 300.0 nM
Cc1nc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)sc1C(=O)NCCc1ccncc1 CHEMBL3661856 IC50 300.0 nM
Cc1nc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)sc1C(=O)NCCc1ccncc1 CHEMBL3661857 IC50 300.0 nM
O=C(NCc1ccncc1)c1sc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)nc1Cl CHEMBL3661864 IC50 300.0 nM
O=C(N[C@H](CO)c1ccccc1)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661887 IC50 300.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)N1CCC[C@H]1CO CHEMBL3661889 IC50 300.0 nM
O=C(NC(CCO)C1CC1)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661890 IC50 300.0 nM
CC[C@@H](C)[C@H](CO)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661893 IC50 300.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CCC(c2ccsc2)O3)s1 CHEMBL3661896 IC50 300.0 nM
Cc1ccccc1C1CCc2cc(Oc3ncc(C(=O)NCc4ccnc(Cl)c4)s3)ccc2O1 CHEMBL3661899 IC50 300.0 nM
COC(=O)C1CN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CC1C(F)(F)F CHEMBL3661904 IC50 300.0 nM
COC(=O)C1CN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CC1C CHEMBL3661907 IC50 300.0 nM
CC(C)CC(CNC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661918 IC50 300.0 nM
O=C(NC1C2CNCC21)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661935 IC50 300.0 nM
N[C@H]1C[C@@H]1NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661936 IC50 300.0 nM
NCCCNC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661967 IC50 300.0 nM
NC1CCN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)C1 CHEMBL3661970 IC50 300.0 nM
C[C@H](N)C(=O)NCc1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661980 IC50 300.0 nM
O=C(NCC(O)CO)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661982 IC50 300.0 nM
CC(C)NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661995 IC50 300.0 nM
CCCNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2C)O3)s1 CHEMBL3662005 IC50 300.0 nM
Cc1ccccc1C1CCc2cc(Oc3nc(C)c(C(=O)NCCO)s3)ccc2O1 CHEMBL3662010 IC50 300.0 nM
Cc1csc(CCNc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3662052 IC50 400.0 nM
CCn1nccc1CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657654 IC50 400.0 nM
Cn1nccc1CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657656 IC50 400.0 nM
CC(NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccncc1 CHEMBL3657657 IC50 400.0 nM
Nc1cc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)ccn1 CHEMBL3657662 IC50 400.0 nM
CC[C@H](NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccc(OC)nc1 CHEMBL3657673 IC50 400.0 nM
O=C(NCc1ccnc(N2CCCC2)c1)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657676 IC50 400.0 nM
O=C(NCc1ccncc1Cl)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657691 IC50 400.0 nM
C[C@H](NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1nc(C2CC2)cs1 CHEMBL3657703 IC50 400.0 nM
Cc1noc(C)c1CC(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657725 IC50 400.0 nM
Cc1cc(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)ccn1 CHEMBL3657729 IC50 400.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ncccn1 CHEMBL3657733 IC50 400.0 nM
CC(C)CNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657746 IC50 400.0 nM
CN1CCN(Cc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)CC1=O CHEMBL3657747 IC50 400.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CN5CCCC5)s4)ccc3O2)cc1 CHEMBL3657749 IC50 400.0 nM
CC(C)(C)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657762 IC50 400.0 nM
CN(C)Cc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657763 IC50 400.0 nM
Cc1c(S(=O)(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cnn1C CHEMBL3657776 IC50 400.0 nM
Cc1nn(C)cc1CNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657780 IC50 400.0 nM
Cc1cc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n(C)n1 CHEMBL3657784 IC50 400.0 nM
Cc1c(C(C)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cnn1C CHEMBL3657791 IC50 400.0 nM
Nc1cc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)ccn1 CHEMBL3657797 IC50 400.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCc5nnc6ccccn56)s4)ccc3O2)cc1 CHEMBL3657798 IC50 400.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCc5ccnc(N6CCOCC6)c5)s4)ccc3O2)cc1 CHEMBL3657804 IC50 400.0 nM
Cc1nc(S(=O)(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cn1C CHEMBL3661850 IC50 400.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CC[C@H](c2ccccc2)O3)s1 CHEMBL3661859 IC50 400.0 nM
O=C(CN1CC[C@@H](O)C1)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661862 IC50 400.0 nM
Cc1ccccc1C1CCc2cc(Oc3ncc(C(=O)NCCc4c(C)noc4C)s3)ccc2O1 CHEMBL3661863 IC50 400.0 nM
Cc1nc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)sc1C(=O)NCc1ccnc(Cl)c1 CHEMBL3661865 IC50 400.0 nM
COC(=O)[C@@H](C)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661870 IC50 400.0 nM
O=C(N[C@H]1CCCC[C@H]1C(=O)O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661885 IC50 400.0 nM
CC(C)[C@@H](CO)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661886 IC50 400.0 nM
CC[C@H](C)[C@@H](CO)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661892 IC50 400.0 nM
O=C(NCc1ccnc(Cl)c1)c1cnc(Oc2ccc3c(c2)CCC(c2ccsc2)O3)s1 CHEMBL3661895 IC50 400.0 nM
CO[C@H]1CNC[C@@H]1NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661934 IC50 400.0 nM
NC1CC(NC(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)C1 CHEMBL3661937 IC50 400.0 nM
Cc1cc(CNC(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)ccn1 CHEMBL3661953 IC50 400.0 nM
CCOC(=O)[C@H](C)NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2cccnc2)O3)s1 CHEMBL3661955 IC50 400.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)N1CCCCC1 CHEMBL3661966 IC50 400.0 nM
NCC1CCCN1C(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661969 IC50 400.0 nM
O=C(NCCO)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661972 IC50 400.0 nM
Cc1noc(C)c1CCC(=O)NCc1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661973 IC50 400.0 nM
Cc1ccccc1C1CCc2cc(Oc3ncc(C(=O)NCCO)s3)ccc2O1 CHEMBL3661976 IC50 400.0 nM
NCC(=O)NCc1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661979 IC50 400.0 nM
CN1CCN(C(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)CC1 CHEMBL3661989 IC50 400.0 nM
CCCNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661996 IC50 400.0 nM
NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3662014 IC50 400.0 nM
Cc1ccc(F)cc1C1CCc2cc(Oc3ncc(C(=O)NCCO)s3)ccc2O1 CHEMBL3662017 IC50 400.0 nM
Cc1ncoc1C(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657718 IC50 500.0 nM
CCn1ccc(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657739 IC50 500.0 nM
CCC(CC)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657751 IC50 500.0 nM
Cc1cnc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cn1 CHEMBL3657778 IC50 500.0 nM
Cc1ccn(CCNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657779 IC50 500.0 nM
CCn1cc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)c(C)n1 CHEMBL3657782 IC50 500.0 nM
Cc1cc(C)nc(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657786 IC50 500.0 nM
Cc1noc(C)c1CCCNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657795 IC50 500.0 nM
O=C(CN1CCCC1=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661852 IC50 500.0 nM
Cc1nc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)sc1C(=O)NCc1ccnc(Cl)c1 CHEMBL3661854 IC50 500.0 nM
Cc1ccccc1C1CCc2cc(Oc3nc(C)c(C(=O)NCc4ccncc4)s3)ccc2O1 CHEMBL3662049 IC50 500.0 nM
COC(=O)[C@@H]1CCCN1C(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661871 IC50 500.0 nM
O=C(O)CNC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661877 IC50 500.0 nM
CCC(C)C(NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661881 IC50 500.0 nM
O=C(NC[C@H]1CCCC[C@H]1O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661891 IC50 500.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)N1CCOCC1 CHEMBL3661898 IC50 500.0 nM
COC(=O)C1(C)CCN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)C1 CHEMBL3661908 IC50 500.0 nM
CC1CN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CC1C(=O)O CHEMBL3661915 IC50 500.0 nM
CN(C)CCNC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661958 IC50 500.0 nM
O=C(NCC1CCCCN1)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661965 IC50 500.0 nM
CC(C)(C)OC(=O)CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661983 IC50 500.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)N1CCCCC1 CHEMBL3661991 IC50 500.0 nM
CCc1ccccc1C1CCc2cc(Oc3ncc(C(=O)NCc4ccno4)s3)ccc2O1 CHEMBL3661999 IC50 500.0 nM
Cc1ccccc1C1CCc2cc(Oc3ncc(CNC(=O)CN4CCCC4=O)s3)ccc2O1 CHEMBL3662002 IC50 500.0 nM
Cc1ccccc1C1CCc2cc(Oc3nc(C)c(C(=O)NCc4ccno4)s3)ccc2O1 CHEMBL3662009 IC50 500.0 nM
CCCNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2cc(F)ccc2C)O3)s1 CHEMBL3662018 IC50 500.0 nM
Cc1ccc(F)cc1C1CCc2cc(Oc3ncc(C(=O)N4CC[C@@H](O)C4)s3)ccc2O1 CHEMBL3662031 IC50 540.0 nM
CCn1nccc1CNC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2cccc(F)c2OC)O3)s1 CHEMBL3662040 IC50 550.0 nM
COc1cc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)ccn1 CHEMBL3657661 IC50 600.0 nM
O=C(NCc1ccncn1)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657683 IC50 600.0 nM
O=C(NCc1nnc2ccccn12)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657686 IC50 600.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CCC(c2cccnc2)O3)s1 CHEMBL3657708 IC50 600.0 nM
Cc1c(CNC(=O)c2cnc(Oc3ccc4c(c3)CC[C@H](c3ccccc3)O4)s2)cnn1C CHEMBL3657712 IC50 600.0 nM
Cc1cc(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n(C)n1 CHEMBL3657715 IC50 600.0 nM
O=C(CCn1cccn1)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657736 IC50 600.0 nM
O=C(CN1C(=O)CNC1=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657741 IC50 600.0 nM
CC(C)CCNCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657759 IC50 600.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CN5C6CCC5CC6)s4)ccc3O2)cc1 CHEMBL3662048 IC50 600.0 nM
Cc1nc(C)c(S(=O)(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)s1 CHEMBL3657769 IC50 600.0 nM
COC(=O)C(C)(C)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661868 IC50 600.0 nM
COC(=O)C1(NC(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CCCC1 CHEMBL3661873 IC50 600.0 nM
CCOC(=O)C1(NC(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CC1 CHEMBL3662050 IC50 600.0 nM
CCOC(=O)[C@@H]1CCCC[C@@H]1NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661874 IC50 600.0 nM
C[C@H](NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661876 IC50 600.0 nM
CC(C)(NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661878 IC50 600.0 nM
CC(C)[C@H](NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661882 IC50 600.0 nM
COC(=O)[C@@H](NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(C)(C)C CHEMBL3661903 IC50 600.0 nM
CC(C)C[C@H](NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661921 IC50 600.0 nM
O=C(N[C@@H](Cc1ccccc1)C(=O)O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661924 IC50 600.0 nM
O=C(O)CNCc1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661926 IC50 600.0 nM
O=C(NCCO)c1cnc(Oc2ccc3c(c2)CCC(c2cncc(F)c2)O3)s1 CHEMBL3661933 IC50 600.0 nM
N[C@H]1C[C@@H]1NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2cccnc2)O3)s1 CHEMBL3661946 IC50 600.0 nM
CCCNC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661959 IC50 600.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)N1CC[C@H]2CNC[C@H]21 CHEMBL3661961 IC50 600.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)N1CCC2(CCCNC2)C1 CHEMBL3661968 IC50 600.0 nM
O=C(c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)N1CC[C@@H](O)C1 CHEMBL3661975 IC50 600.0 nM
Cc1ccccc1C1CCc2cc(Oc3ncc(CNC(=O)c4ccno4)s3)ccc2O1 CHEMBL3662004 IC50 600.0 nM
Cc1ccccc1C1CCc2cc(Oc3nc(C)c(C(=O)NCCN4CCNC4=O)s3)ccc2O1 CHEMBL3662008 IC50 600.0 nM
Cc1ccccc1C1CCc2cc(Oc3nc(C)c(C(=O)N4CC[C@@H](O)C4)s3)ccc2O1 CHEMBL3662011 IC50 600.0 nM
Cc1cc2c(cc1Oc1ncc(C(=O)NCCO)s1)CCC(c1ccccc1C)O2 CHEMBL3662032 IC50 600.0 nM
Cc1ccc(F)cc1C1CCc2cc(Oc3ncc(C(=O)N(C)C)s3)ccc2O1 CHEMBL3662023 IC50 640.0 nM
CC(C)c1csc([C@H](C)NC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657704 IC50 700.0 nM
Cc1c(C(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cnn1C CHEMBL3657720 IC50 700.0 nM
CCCCN(C)Cc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657744 IC50 700.0 nM
FC1(F)CCN(Cc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)CC1 CHEMBL3657753 IC50 700.0 nM
Cc1c(S(=O)(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cnn1C(C)C CHEMBL3657773 IC50 700.0 nM
CN1CC(=O)N(CC(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)C1=O CHEMBL3661851 IC50 700.0 nM
CCOC(=O)[C@@H](NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(C)C CHEMBL3661872 IC50 700.0 nM
C[C@@H](NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661879 IC50 700.0 nM
O=C(NC1(C(=O)O)CCCC1)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661880 IC50 700.0 nM
COC(=O)[C@H](O)[C@H](CC(C)C)NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661909 IC50 700.0 nM
CC(C)CC(C)(NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661922 IC50 700.0 nM
O=C(O)C1CN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CC1C(F)(F)F CHEMBL3661923 IC50 700.0 nM
O=C(NCc1ccnc(Cl)c1)c1cnc(Oc2ccc3c(c2)CCC(c2cncc(F)c2)O3)s1 CHEMBL3661927 IC50 700.0 nM
Cc1c(C(C)NC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cnn1C CHEMBL3657659 IC50 800.0 nM
Cc1cc(CNC(=O)c2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)ccn1 CHEMBL3657660 IC50 800.0 nM
Cc1nn(C)cc1C(C)NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657674 IC50 800.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)c1ccnc(Cl)c1 CHEMBL3657717 IC50 800.0 nM
CC(C)Oc1cccc(C2CCc3cc(Oc4ncc(C(=O)NCc5ccncc5)s4)ccc3O2)c1 CHEMBL3657742 IC50 800.0 nM
CC(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)C(C)(C)C CHEMBL3657750 IC50 800.0 nM
Cc1cc(NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)on1 CHEMBL3657755 IC50 800.0 nM
CN1CCN(Cc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)CC1 CHEMBL3657765 IC50 800.0 nM
C1=C(CNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)N2CCCN=C2S1 CHEMBL3657787 IC50 800.0 nM
Cc1cc(C)n(CCNCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)n1 CHEMBL3657793 IC50 800.0 nM
O=C(NCc1ccncc1)c1cnc(Oc2ccc3c(c2)CCC(c2cccc(O)c2)O3)s1 CHEMBL3661861 IC50 800.0 nM
CN1CCN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CC1 CHEMBL3661897 IC50 800.0 nM
CC(Cc1ccccc1)(NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661913 IC50 800.0 nM
CC(C)C[C@@H](NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1)C(=O)O CHEMBL3661917 IC50 800.0 nM
O=C(NCc1ccno1)c1cnc(Oc2ccc3c(c2)CCC(c2cncc(F)c2)O3)s1 CHEMBL3661928 IC50 800.0 nM
CCOC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2cccnc2)O3)s1 CHEMBL3661941 IC50 800.0 nM
OCCN(CCO)Cc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3661994 IC50 800.0 nM
Cc1ccc(F)cc1C1CCc2cc(Oc3ncc(C(=O)NCc4ccno4)s3)ccc2O1 CHEMBL3662019 IC50 800.0 nM
Cc1cc2c(cc1Oc1ncc(C(=O)NCc3ccno3)s1)CCC(c1ccccc1C)O2 CHEMBL3662033 IC50 830.0 nM
Cc1noc(C)c1CCC(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657740 IC50 900.0 nM
Cc1nc2ccc(S(=O)(=O)NCc3cnc(Oc4ccc5c(c4)CCC(c4ccccc4)O5)s3)cc2s1 CHEMBL3657767 IC50 900.0 nM
Cn1cc(S(=O)(=O)NCc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)cn1 CHEMBL3657772 IC50 900.0 nM
c1ccc(C2CCc3cc(Oc4ncc(CNCc5cccnc5N5CCOCC5)s4)ccc3O2)cc1 CHEMBL3657788 IC50 900.0 nM
CN(CC(=O)O)C(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661875 IC50 900.0 nM
COC(=O)[C@@H]1[C@@H]2C[C@@H]2CN1C(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661905 IC50 900.0 nM
CN[C@H]1CN(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)CC[C@H]1C CHEMBL3661963 IC50 900.0 nM
CCc1ccccc1C1CCc2cc(Oc3ncc(C(=O)NCCc4c(C)noc4C)s3)ccc2O1 CHEMBL3661998 IC50 900.0 nM
Cc1ccccc1C1CCc2cc(Oc3ncc(CNC(=O)CN4C(=O)CNC4=O)s3)ccc2O1 CHEMBL3662003 IC50 900.0 nM
N[C@@H](CO)C(=O)NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3662015 IC50 900.0 nM
O=C(NCc1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1)[C@@H]1CCCN1 CHEMBL3662016 IC50 900.0 nM
CC1Cc2cc(Oc3ncc(C(=O)NCCO)s3)ccc2OC1c1ccccc1 CHEMBL3662039 IC50 960.0 nM
Cc1n[nH]c(C)c1C(C)NC(=O)c1cnc(Oc2ccc3c(c2)CCC(c2ccccc2)O3)s1 CHEMBL3657682 IC50 1000.0 nM
C[C@@H]1CN(Cc2cnc(Oc3ccc4c(c3)CCC(c3ccccc3)O4)s2)C[C@H](C)O1 CHEMBL3657745 IC50 1000.0 nM
O=C(NC1(C(=O)O)CC1)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3661884 IC50 1000.0 nM
CC1(C)C[C@@H](C(=O)O)N(C(=O)c2cnc(Oc3ccc4c(c3)CC[C@@H](c3ccccc3)O4)s2)C1 CHEMBL3661914 IC50 1000.0 nM
CNC1C2CCC(C2)C1NC(=O)c1cnc(Oc2ccc3c(c2)CC[C@@H](c2ccccc2)O3)s1 CHEMBL3662046 IC50 1000.0 nM