CC(C)C[C@H]1C[C@@H](C)[C@]2(C(=O)Nc3ccc(F)cc32)N1C(=O)c1cn(Cc2ccccc2)cn1 CHEMBL4091579 IC50 11.0 nM
CC(C)C[C@H]1C[C@@H](C)[C@]2(C(=O)Nc3ccc(F)cc32)N1C(=O)c1cn(C)cn1 CHEMBL4070683 IC50 21.0 nM
COC(=O)[C@@H]1C[C@H](CC(C)C)N(C(=O)c2cn(Cc3ccccc3)cn2)[C@@]12C(=O)Nc1ccc(F)cc12 CHEMBL4104317 IC50 44.0 nM
O=C1Nc2cc(=O)n(Cc3ccccc3)cc2CN1c1cccc(OCc2cncs2)c1 CHEMBL4084949 IC50 79.0 nM
COC(=O)[C@@H]1C[C@H](CC(C)C)N(C(=O)c2cn(C)cn2)[C@@]12C(=O)Nc1ccc(F)cc12 CHEMBL4100976 IC50 110.0 nM
O=C1Nc2cc(=O)n(Cc3ccccc3)cc2CN1c1cccc(OCc2cccnc2)c1 CHEMBL4097764 IC50 180.0 nM
CC(C)C[C@H]1C[C@@H](C)[C@]2(C(=O)Nc3ccccc32)N1C(=O)c1ccccn1 CHEMBL4088975 IC50 360.0 nM
COC(=O)[C@@H]1C[C@H](CC(C)C)N(C(=O)c2c[nH]cn2)[C@@]12C(=O)Nc1ccc(F)cc12 CHEMBL4080080 IC50 390.0 nM
O=C1Nc2cc(=O)n(Cc3ccccc3)cc2CN1c1cccc(OCc2ccccc2)c1 CHEMBL4065018 IC50 790.0 nM
COC(=O)[C@@H]1C[C@H](CC(C)C)N(C(=O)c2ccccn2)[C@@]12C(=O)Nc1ccc(F)cc12 CHEMBL4076145 IC50 910.0 nM
