Cc1cn(-c2nccc(N3C[C@@H](C)N(c4ccnc([C@@H](C)O)n4)[C@@H](C)C3)n2)c(C)n1 CHEMBL136420 IC50 4.0 nM
C[C@@H]1CN(c2ccnc(N3CCN(C)CC3)n2)C[C@H](C)N1c1ccnc([C@@H](C)O)n1 CHEMBL136900 IC50 4.0 nM
Cc1nc(C)nc(N2C[C@@H](C)N(c3ccnc([C@@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL136680 IC50 5.0 nM
CC(=O)c1nccc(N2[C@H](C)CN(c3ccnc([C@@H](C)O)n3)C[C@@H]2C)n1 CHEMBL34667 IC50 6.0 nM
C[C@@H]1CN(c2ncnc(-c3ccccc3)n2)C[C@H](C)N1c1ccnc([C@@H](C)O)n1 CHEMBL136103 IC50 7.0 nM
Cc1ncnc(N2C[C@@H](C)N(c3ccnc([C@@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL342697 IC50 7.0 nM
Cc1nc2ccccc2nc1N1CCN(c2ccnc([C@@H](C)O)n2)CC1 CHEMBL151486 IC50 8.0 nM
C[C@@H]1CN(c2ccnc(CCO)n2)C[C@H](C)N1c1ccnc([C@@H](C)O)n1 CHEMBL151017 IC50 10.0 nM
C[C@H](O)c1nccc(N2C[C@@H](C)N(c3ccnc([C@@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL287890 IC50 10.0 nM
C[C@@H]1CN(c2ccnc([C@@H](C)O)n2)C[C@H](C)N1c1ccnc([C@@H](C)O)n1 CHEMBL36514 IC50 10.0 nM
C[C@@H]1CN(c2ccnc(CCO)n2)CCN1c1ccnc([C@@H](C)O)n1 CHEMBL347716 IC50 12.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nsc4ccccc34)CC2)n1 CHEMBL147064 IC50 12.0 nM
Cc1cn(-c2nccc(N3C[C@@H](C)N(c4ccnc([C@@H](C)O)n4)[C@@H](C)C3)n2)cn1 CHEMBL435428 IC50 13.0 nM
C[C@H](O)c1nccc(N2[C@H](C)CN(c3ccnc([C@@H](C)O)n3)C[C@@H]2C)n1 CHEMBL34965 IC50 19.0 nM
CC(=O)c1nccc(N2C[C@@H](C)N(c3ccnc([C@@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL286539 IC50 19.0 nM
Cc1cc(CO)nc(N2CCN(c3ccnc([C@@H](C)O)n3)CC2)n1 CHEMBL151615 IC50 20.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nc4ccncc4o3)[C@@H](C)C2)n1 CHEMBL149048 IC50 23.0 nM
Cc1cc(C)nc(N2CCN(c3ccnc([C@@H](C)O)n3)CC2)n1 CHEMBL151439 IC50 23.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nc4ccncc4o3)CC2)n1 CHEMBL348496 IC50 24.0 nM
C[C@@H](O)c1nccc(N2CCN(S(=O)(=O)N(C)C)CC2)n1 CHEMBL90344 IC50 27.0 nM
CC(O)c1nccc(N2C[C@@H](C)N(c3ccnc(C(C)O)n3)[C@@H](C)C2)n1 CHEMBL36368 IC50 28.0 nM
Cc1cc(N2CCN(c3ccnc([C@@H](C)O)n3)CC2)nc(C)n1 CHEMBL359089 IC50 31.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nc4cccnc4o3)CC2)n1 CHEMBL151311 IC50 32.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nccc4ccccc34)CC2)n1 CHEMBL346418 IC50 34.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nc4ccccc4o3)CC2)n1 CHEMBL150642 IC50 35.0 nM
C[C@@H](O)c1nccc(N2CCN(c3cnc4ccccc4n3)CC2)n1 CHEMBL359168 IC50 36.0 nM
C[C@@H](O)c1nccc(N2CCN(c3noc4ccccc34)CC2)n1 CHEMBL151764 IC50 37.0 nM
C[C@@H](O)c1nccc(N2CCN(c3ccnc(CCO)n3)CC2)n1 CHEMBL149981 IC50 40.0 nM
Cc1nc(-c2ccccc2)nc(N2C[C@@H](C)N(c3ccnc([C@@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL139187 IC50 43.0 nM
C[C@@H](O)c1nccc(N2CCN(c3ccc4ccccc4n3)CC2)n1 CHEMBL556517 IC50 44.0 nM
C[C@@H](O)c1nccc(N2CCN(c3ccnc(CCO)n3)C[C@@H]2C)n1 CHEMBL150296 IC50 59.0 nM
OCc1nccc(N2CCN(c3nsc4ccccc34)CC2)n1 CHEMBL146805 IC50 64.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nccc(-c4ccccc4)n3)CC2)n1 CHEMBL151394 IC50 67.0 nM
CC(C)c1cc(C(C)C)nc(N2CCN(c3ccnc([C@@H](C)O)n3)CC2)n1 CHEMBL150734 IC50 72.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nc4cnccc4o3)CC2)n1 CHEMBL356692 IC50 80.0 nM
CCc1cc(CC)nc(N2CCN(c3ccnc([C@@H](C)O)n3)CC2)n1 CHEMBL348427 IC50 80.0 nM
Cc1cc(CO)nc(N2CCN(c3ccnc([C@@H](C)O)n3)C[C@@H]2C)n1 CHEMBL150803 IC50 80.0 nM
OCc1nccc(N2CCN(c3ccc4ccccc4n3)CC2)n1 CHEMBL151605 IC50 87.0 nM
Cc1cc(C)nc(N2CCN(c3ccnc(CO)n3)CC2)n1 CHEMBL151268 IC50 93.0 nM
C[C@@H](O)c1nccc(N2CCN(c3cnc4ccccc4n3)[C@@H](C)C2)n1 CHEMBL149409 IC50 99.0 nM
Cc1cc(CO)nc(N2C[C@@H](C)N(c3ccnc([C@@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL151560 IC50 100.0 nM
Cc1ccnc(N2CCN(c3ccnc([C@@H](C)O)n3)CC2)n1 CHEMBL347575 IC50 110.0 nM
C[C@@H](O)c1nccc(N2CCN(c3cnc4cc(Cl)c(Cl)cc4n3)CC2)n1 CHEMBL151690 IC50 120.0 nM
OCc1nccc(N2CCN(c3noc4ccccc34)CC2)n1 CHEMBL357712 IC50 120.0 nM
Cc1cc(CO)nc(N2[C@H](C)CN(c3ccnc([C@@H](C)O)n3)C[C@@H]2C)n1 CHEMBL346682 IC50 130.0 nM
Cc1cc(N2CCN(c3ccnc(CO)n3)CC2)nc(C)n1 CHEMBL423753 IC50 140.0 nM
Cc1cc(CO)nc(N2CCN(c3ccnc([C@@H](C)O)n3)C[C@H]2C)n1 CHEMBL148936 IC50 140.0 nM
OCc1nccc(N2CCN(c3nccc4ccccc34)CC2)n1 CHEMBL358327 IC50 150.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nc4ncccc4o3)CC2)n1 CHEMBL147197 IC50 170.0 nM
Cc1cc(CO)nc(N2CCN(c3ccnc([C@@H](C)O)n3)[C@H](C)C2)n1 CHEMBL151567 IC50 170.0 nM
CC(O)c1nccc(N2CCN(S(=O)(=O)N(C)C)CC2)n1 CHEMBL91846 IC50 173.0 nM
C[C@@H]1CN(c2cnc3ccccc3n2)C[C@H](C)N1c1ccnc([C@@H](C)O)n1 CHEMBL345259 IC50 180.0 nM
OCc1nccc(N2CCN(c3nc4ccccc4o3)CC2)n1 CHEMBL148647 IC50 190.0 nM
C[C@@H](O)c1nccc(N2CCN(c3nc(C(F)(F)F)cc(C(F)(F)F)n3)CC2)n1 CHEMBL148436 IC50 190.0 nM
Cc1cc(CO)nc(N2CCN(c3ccnc([C@@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL151602 IC50 200.0 nM
CC(=O)c1nccc(N2C[C@@H](C)N(c3ccnc(C(C)=O)n3)[C@@H](C)C2)n1 CHEMBL277816 IC50 212.0 nM
Cc1cc(-c2ccccc2)nc(N2CCN(c3ccnc([C@@H](C)O)n3)CC2)n1 CHEMBL151704 IC50 220.0 nM
CN(C)S(=O)(=O)N1CCN(c2ccnc(CO)n2)CC1 CHEMBL90488 IC50 240.0 nM
OCc1nccc(N2CCN(c3ccnc(CO)n3)CC2)n1 CHEMBL348663 IC50 260.0 nM
C[C@@H]1CN(c2nc3ccncc3o2)C[C@H](C)N1c1ccnc([C@@H](C)O)n1 CHEMBL345725 IC50 270.0 nM
CO[C@@H](C)c1nccc(N2CCN(S(=O)(=O)N(C)C)CC2)n1 CHEMBL330334 IC50 486.0 nM
OCc1nccc(N2CCN(c3nc(Cl)nc(Cl)n3)CC2)n1 CHEMBL148935 IC50 490.0 nM
C[C@H](O)c1nccc(N2C[C@@H](C)N(c3ccnc([C@H](C)O)n3)[C@@H](C)C2)n1 CHEMBL284537 IC50 831.0 nM
OCc1nccc(N2CCN(c3ncnc4ccccc34)CC2)n1 CHEMBL148822 IC50 890.0 nM