CC1(C)C(N)=Nc2cc(OCCCN3Cc4ccc(OCc5cn(CCC(=O)N6CCC(CCN7CCCC7)CC6)nn5)cc4C3)c(OCC3CC3)cc21 CHEMBL4573889 Kd 6.6 nM
CC1(C)C(N)=Nc2cc(OCCCN3Cc4ccc(OCCc5cn(CC(=O)N6CCC(CCN7CCCC7)CC6)nn5)cc4C3)c(OCC3CC3)cc21 CHEMBL4451634 Kd 9.9 nM
CC1(C)C(N)=Nc2cc(OCCCN3Cc4ccc(OCCc5cn(CCC(=O)N6CCC(CCN7CCCC7)CC6)nn5)cc4C3)c(OCC3CC3)cc21 CHEMBL4570122 Kd 10.1 nM
CC1(C)C(N)=Nc2cc(OCCCN3Cc4ccccc4C3)c(OCC3CC3)cc21 CHEMBL4528213 Kd 15.4 nM
CC1(C)C(N)=Nc2cc(OCCCN3Cc4ccc(OCc5cn(CC(=O)N6CCC(CCN7CCCC7)CC6)nn5)cc4C3)c(OCC3CC3)cc21 CHEMBL4577068 Kd 60.0 nM
COc1cc2c(cc1OCCCN1CCCC1)N=C(N)C21CCC1 CHEMBL3109630 IC50 72.0 nM
COc1c(CN)cc(CN)cc1OCCCN1Cc2ccccc2C1 CHEMBL4552020 IC50 77.0 nM
COc1c(CN)cc(CN)cc1OCCCN1CCCC1 CHEMBL4588285 IC50 338.0 nM
COc1ccc2c(c1)CN(CCCOc1cc3c(cc1OCC1CC1)C1(CCCC1)C(N)=N3)C2 CHEMBL4591023 IC50 340.0 nM
NC1=Nc2cc(OCCCN3Cc4ccccc4C3)c(OCC3CC3)cc2C12CCCC2 CHEMBL4476309 IC50 390.0 nM
COc1ccc2c(c1)CN(CCCOc1cc3c(cc1OC)C1(CCCC1)C(N)=N3)C2 CHEMBL4518756 IC50 600.0 nM
COc1cc2c(cc1OCCCN1Cc3ccccc3C1)N=C(N)C21CCCC1 CHEMBL4569420 IC50 660.0 nM
COc1cc2c(cc1OCCCN1CCCC1)N=C(N)C21CCCC1 CHEMBL4458252 IC50 760.0 nM