CCCCCCC(=O)CCCCCC/C=C/C[C@@H](O)[C@H](O)[C@@](N)(CO)C(=O)O CHEMBL55076 IC50 0.13 nM
COc1ccc(C(=O)N2CC[C@@H](NC(=O)c3ccccc3Cl)[C@@H](c3ccccc3)C2)cc1OC CHEMBL4228416 IC50 0.36 nM
COc1cc(C(=O)N2CC[C@H](NC(=O)c3ccccc3OC(F)(F)F)c3c2cnn3C(C)C)cnc1OC CHEMBL4225519 IC50 0.54 nM
Cn1nc(C(F)(F)F)cc1C(=O)N[C@@H]1CCN(C(=O)c2cc(Cl)c3nccnc3c2)C[C@@H]1c1ccccc1 CHEMBL4228472 IC50 0.71 nM
COc1cc(C(=O)N2CCC(NC(=O)c3ccccc3OC(F)(F)F)c3c2cnn3C(C)C)cnc1OC CHEMBL4225462 IC50 1.2 nM
COc1ccc(C(=O)N2CCC(NC(=O)c3ccccc3Cl)C(c3ccccc3)C2)cc1OC CHEMBL4225764 IC50 1.2 nM
COc1ccc(C(=O)N2CC[C@@H](NC(=O)c3ccccc3Cl)[C@H](c3ccccc3)C2)cc1OC CHEMBL4229253 IC50 5.0 nM
COc1ccc(C(=O)N2CCC(NC(=O)c3ccccc3Cl)c3ccc(Cl)cc32)cc1OC CHEMBL4225192 IC50 5.1 nM
COc1ccc(C(=O)N2CCC(NC(=O)c3ccccc3Cl)c3c2cnn3C)cc1OC CHEMBL4226297 IC50 7.7 nM
CCCCCCCC(=O)CCCCCC/C=C/[C@H](C(=O)N[C@@H](Cc1ccc(OCC=C(C)C)cc1)C(=O)O)[C@@](O)(CC(=O)O)C(=O)O CHEMBL1241090 IC50 10.0 nM
COc1ccc(C(=O)N2CC[C@H](NC(=O)c3ccccc3Cl)[C@H](c3ccccc3)C2)cc1OC CHEMBL4228993 IC50 220.0 nM
COc1ccc(C(=O)N2CCC(Nc3ccc(Cl)cc3)c3ccc(Cl)cc32)cc1OC CHEMBL4226045 IC50 650.0 nM