CC(C)NCC(O)c1ccc(O)c(O)c1 CHEMBL434 EC50 4.9 nM
Cc1ccc(S(=O)(=O)N(Cc2ccccc2)CC2CCC(C(=O)O)CC2)cc1 CHEMBL3895068 IC50 14.0 nM
COc1cccc(CN(CC2CCC(C(=O)O)CC2)S(=O)(=O)c2ccc(C)cc2)c1 CHEMBL3909546 IC50 36.0 nM
Cc1ccc(S(=O)(=O)N(Cc2ccc(F)cc2)Cc2ccc(C(=O)O)cc2)cc1 CHEMBL3907785 IC50 54.0 nM
Cc1cc(C(F)(F)F)nc(Nc2ccccc2-c2nnn[nH]2)n1 CHEMBL5279691 EC50 72.0 nM
Cc1ccc(S(=O)(=O)N(Cc2ccc(F)cc2)CC2CCC(C(=O)O)CC2)cc1 CHEMBL3930803 IC50 83.0 nM
COc1ccc(S(=O)(=O)N(Cc2ccc(F)cc2)CC2CCC(C(=O)O)CC2)cc1 CHEMBL3905445 IC50 92.0 nM
FC(F)(F)c1cccc(Nc2ccccc2-c2nnn[nH]2)n1 CHEMBL5285591 EC50 98.0 nM
FC(F)(F)c1cc(Nc2ccccc2-c2nnn[nH]2)cc(C(F)(F)F)c1 CHEMBL5275180 EC50 100.0 nM
Cc1ccc(CN(CC2CCC(C(=O)O)CC2)S(=O)(=O)c2ccc(C)cc2)cc1 CHEMBL3904387 IC50 109.0 nM
C#Cc1cc(Nc2ccccc2C(=O)O)cc(C(F)(F)F)c1 CHEMBL5273955 EC50 150.0 nM
FC(F)(F)c1ccnc(Nc2ccccc2-c2nnn[nH]2)n1 CHEMBL5274304 EC50 160.0 nM
N#Cc1ccc(Nc2ccccc2C(=O)O)cc1C(F)(F)F CHEMBL5277615 EC50 170.0 nM
N#Cc1cc(Nc2ccccc2C(=O)O)cc(C(F)(F)F)c1 CHEMBL5280542 EC50 180.0 nM
COc1cccc(CN(Cc2ccc(C(=O)O)cc2)S(=O)(=O)c2ccc(O)cc2)c1 CHEMBL3901989 IC50 188.0 nM
O=C(O)c1ccccc1Nc1cccc(S(F)(F)(F)(F)F)c1 CHEMBL3623735 EC50 190.0 nM
Cc1cc(Nc2ccccc2C(=O)O)cc(C(F)(F)F)c1 CHEMBL5279381 EC50 190.0 nM
COc1ccc(CN(Cc2ccccc2)S(=O)(=O)c2ccc(C(=O)O)cc2)cc1 CHEMBL3092287 IC50 200.0 nM
O=C(O)c1ccccc1Nc1cc(Br)cc(C(F)(F)F)c1 CHEMBL3088246 EC50 230.0 nM
O=C(O)C1CCC(CN(Cc2ccc(F)cc2)S(=O)(=O)c2ccccc2)CC1 CHEMBL3946036 IC50 240.0 nM
Cn1c(=O)c2cc(S(=O)(=O)Nc3ccc4c(c3)OCO4)ccc2n(C)c1=O CHEMBL1401915 IC50 264.0 nM
Cc1nc(SCC(=O)N2CCCCC2)c2c(=O)n(C)c(=O)n(C)c2n1 CHEMBL3962122 IC50 292.0 nM
O=C(O)c1ccccc1Nc1ccc(Br)c(C(F)(F)F)c1 CHEMBL5278834 EC50 300.0 nM
N#Cc1cc(C(F)(F)F)nc(Nc2ccccc2-c2nnn[nH]2)n1 CHEMBL5277281 EC50 300.0 nM
Cc1ccc(Nc2ccccc2C(=O)O)cc1C(F)(F)F CHEMBL5278171 EC50 330.0 nM
CCOC(=O)C1CCC(CN(Cc2ccccc2)S(=O)(=O)c2ccc(NC(C)=O)cc2)CC1 CHEMBL3917592 IC50 334.0 nM
O=C(O)C1CCC(CN(Cc2ccc(F)cc2)S(=O)(=O)c2cccs2)CC1 CHEMBL3972175 IC50 342.0 nM
COc1cccc(CN(Cc2ccc(C(=O)O)cc2)S(=O)(=O)c2ccccc2)c1 CHEMBL3954153 IC50 345.0 nM
FC(F)(F)c1ccnc(Nc2ccccc2-c2nnn[nH]2)c1 CHEMBL5274470 EC50 360.0 nM
CC#Cc1cc(Nc2ccccc2C(=O)O)cc(C(F)(F)F)c1 CHEMBL5278477 EC50 380.0 nM
Cc1ccc(C(F)(F)F)cc1Nc1ccccc1C(=O)O CHEMBL5275001 EC50 390.0 nM
O=C(O)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 CHEMBL1082389 IC50 394.0 nM
O=C(O)c1ccc(CN(Cc2cccc(F)c2)S(=O)(=O)c2ccccc2)cc1 CHEMBL3892321 IC50 406.0 nM
N#Cc1ccc(C(F)(F)F)cc1Nc1ccccc1C(=O)O CHEMBL5289590 EC50 420.0 nM
O=C(O)c1ccc(CN(Cc2ccccc2F)S(=O)(=O)c2ccccc2)cc1 CHEMBL3907807 IC50 429.0 nM
O=C(O)c1ccccc1Nc1cccc(C(F)(F)F)c1 CHEMBL23588 EC50 430.0 nM
O=C(O)c1ccc(CN(Cc2cccc(F)c2)S(=O)(=O)c2ccc(O)cc2)cc1 CHEMBL3976457 IC50 459.0 nM
Cc1ccc(S(=O)(=O)N(Cc2ccc(C#N)cc2)CC2CCC(C(=O)O)CC2)cc1 CHEMBL3982886 IC50 499.0 nM
N#C/C(=C\c1ccco1)C(=O)Nc1nnc(-c2ccccc2)s1 CHEMBL3908011 IC50 499.0 nM
FC(F)(F)c1cc(Cl)nc(Nc2ccccc2-c2nnn[nH]2)n1 CHEMBL5280688 EC50 540.0 nM
COc1ccc(CN(Cc2ccco2)S(=O)(=O)c2ccc(C(=O)O)cc2)cc1 CHEMBL3894540 IC50 590.0 nM
O=C(O)c1ccccc1Nc1cc(C(F)(F)F)ccc1Br CHEMBL5286379 EC50 640.0 nM
CC(C)(C)c1cc(C(F)(F)F)nc(Nc2ccccc2-c2nnn[nH]2)n1 CHEMBL5268924 EC50 640.0 nM
O=C(O)c1ccccc1Nc1cccc(C(F)(F)F)n1 CHEMBL5279341 EC50 670.0 nM
CCOC(=O)C1CCC(CN(Cc2ccccc2)S(=O)(=O)c2ccc(Cl)cc2)CC1 CHEMBL1356858 IC50 672.0 nM
COc1ccc(CN(Cc2ccccc2)S(=O)(=O)c2ccc(C(=O)O)cc2)cc1OC CHEMBL3978302 IC50 678.0 nM
Cn1c(=O)c2cc(S(=O)(=O)Nc3ccc4c(c3)OCCO4)ccc2n(C)c1=O CHEMBL3945665 IC50 706.0 nM
Cn1c(=O)c2c(SCC(=O)NCc3ccccc3)ccnc2n(C)c1=O CHEMBL3965603 IC50 710.0 nM
CCc1nc(SCC(=O)N2CCC(C)CC2)c2c(=O)n(C)c(=O)n(C)c2n1 CHEMBL1499181 IC50 721.0 nM
FC(F)(F)c1cc(I)nc(Nc2ccccc2-c2nnn[nH]2)n1 CHEMBL5289980 EC50 750.0 nM
CCOC(=O)N1CCN(C(=O)CSc2nc(CC)nc3c2c(=O)n(C)c(=O)n3C)CC1 CHEMBL1711155 IC50 763.0 nM
CC(=O)Nc1ccc(S(=O)(=O)N(Cc2ccc(F)cc2)CC2CCC(C(=O)O)CC2)cc1 CHEMBL3976205 IC50 842.0 nM
CCN(C)C(=O)CSc1nc(C)nc2c1c(=O)n(C)c(=O)n2C CHEMBL3953366 IC50 861.0 nM
O=C(O)c1ccccc1Nc1cccc(OC(F)F)c1 CHEMBL5276181 EC50 930.0 nM
O=C(O)c1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2ccccc2)cc1 CHEMBL3916808 IC50 935.0 nM
Cc1c(F)cccc1NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C CHEMBL1419634 IC50 935.0 nM
O=C(O)c1ccccc1Nc1cccc(Cl)c1 CHEMBL22815 EC50 950.0 nM