C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncn(C)c3n2)C1 CHEMBL5401444 IC50 3.0 nM
C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncsc3n2)C1 CHEMBL5422959 IC50 3.0 nM
CN(Cc1nn(-c2ccc(OC(F)(F)F)cc2)c2ccccc12)C(=O)CCl CHEMBL5438256 IC50 3.0 nM
C=C(Cl)C(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 CHEMBL5408536 IC50 3.0 nM
C=CS(=O)(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 CHEMBL5419829 IC50 4.0 nM
C=CC(=O)N(C)Cc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 CHEMBL5415215 IC50 4.0 nM
C#Cc1ccnc2c1c(C1CN(C(=O)C=C)C1)nn2-c1ccc(OC(F)(F)F)cc1 CHEMBL5411200 IC50 4.0 nM
C#CC(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 CHEMBL5403826 IC50 4.0 nM
C=CC(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncn(C)c2c1C#CCO CHEMBL5416415 IC50 6.0 nM
Cn1cnc2c(-c3ccc(OC(F)(F)F)cc3)nc(C3CN(C(=O)C4=CCC4)C3)nc21 CHEMBL5400400 IC50 7.0 nM
O=C(/C=C/CO)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(Cl)c23)C1 CHEMBL5428867 IC50 8.0 nM
C=CC(=O)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(CO)c23)C1 CHEMBL5432828 IC50 10.0 nM
CCCC[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc2cccc(Cl)c2)NC(C)[C@@H]2CCCN2C(=O)[C@@H](NC(C)=O)C(C)C)CCSSC[C@@H](C(=O)N[C@@H](CCCCN)C(=O)N2CCC[C@H]2C(=O)N2CCC[C@H]2C(=O)N[C@@H](CCC(=O)O)C(N)=O)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@@H]2CCCN2C1=O CHEMBL4130196 Kd 15.0 nM
O=C(CSc1nnc[nH]1)Nc1ccc(C2C3CC4CC(C3)CC2C4)cc1 CHEMBL4129172 IC50 83.0 nM
Cn1cc2c3cc(C(=O)O)ccc3n(-c3ccc(C(F)(F)F)cc3)c2n1 CHEMBL5170406 Kd 120.0 nM
N#CN1Cc2cccc(Nc3ccc(C(F)(F)F)cc3)c2C1 CHEMBL5434817 IC50 200.0 nM
N#CN1Cc2ccc(F)c(Nc3cccc(C(F)(F)F)c3)c2C1 CHEMBL5432067 IC50 200.0 nM
COc1ccc2c(c1Nc1cccc(C(F)(F)F)c1)CN(C#N)C2 CHEMBL5405832 IC50 300.0 nM
C=CC(=O)N1CCC(CCOc2ccccc2)CC1 CHEMBL5428462 IC50 580.0 nM
N#CN1Cc2cccc(Nc3cccc(C(F)(F)F)c3)c2C1 CHEMBL5394226 IC50 900.0 nM