C#Cc1ccnc2c1c(C1CN(C(=O)C=C)C1)nn2-c1ccc(OC(F)(F)F)cc1 CHEMBL5411200 IC50 2.0 nM
C=CS(=O)(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 CHEMBL5419829 IC50 3.0 nM
C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncn(C)c3n2)C1 CHEMBL5401444 IC50 3.0 nM
C=C(Cl)C(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 CHEMBL5408536 IC50 3.0 nM
C#CC(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 CHEMBL5403826 IC50 3.0 nM
C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncsc3n2)C1 CHEMBL5422959 IC50 4.0 nM
Cn1cnc2c(-c3ccc(OC(F)(F)F)cc3)nc(C3CN(C(=O)C4=CCC4)C3)nc21 CHEMBL5400400 IC50 4.0 nM
C=CC(=O)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(CO)c23)C1 CHEMBL5432828 IC50 4.0 nM
C=CC(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncn(C)c2c1C#CCO CHEMBL5416415 IC50 6.0 nM
C=CC(=O)N(C)Cc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 CHEMBL5415215 IC50 6.0 nM
COc1c(C)cc(N2C[C@@H](O)[C@@H](O)C2=O)cc1/C=C/c1ccc(Cl)cc1 CHEMBL5440009 Kd 6.2 nM
CN(Cc1nn(-c2ccc(OC(F)(F)F)cc2)c2ccccc12)C(=O)CCl CHEMBL5438256 IC50 9.0 nM
O=C(/C=C/CO)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(Cl)c23)C1 CHEMBL5428867 IC50 17.0 nM
COc1ncc(NS(C)(=O)=O)cc1/C=C/C1CCC(F)(F)CC1 CHEMBL5417138 Kd 229.0 nM
O=C(CSc1nnc[nH]1)Nc1ccc(C23CC4CC(CC(C4)C2)C3)cc1 CHEMBL5397201 IC50 710.0 nM
N#CN1Cc2cccc(Nc3ccc(C(F)(F)F)cc3)c2C1 CHEMBL5434817 IC50 800.0 nM