C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncsc3n2)C1 CHEMBL5422959 IC50 3.0 nM
C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncn(C)c3n2)C1 CHEMBL5401444 IC50 4.0 nM
CN(Cc1nn(-c2ccc(OC(F)(F)F)cc2)c2ccccc12)C(=O)CCl CHEMBL5438256 IC50 4.0 nM
C=C(Cl)C(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 CHEMBL5408536 IC50 4.0 nM
C#Cc1ccnc2c1c(C1CN(C(=O)C=C)C1)nn2-c1ccc(OC(F)(F)F)cc1 CHEMBL5411200 IC50 5.0 nM
C=CC(=O)N(C)Cc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 CHEMBL5415215 IC50 7.0 nM
C=CS(=O)(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 CHEMBL5419829 IC50 8.0 nM
Cn1cnc2c(-c3ccc(OC(F)(F)F)cc3)nc(C3CN(C(=O)C4=CCC4)C3)nc21 CHEMBL5400400 IC50 9.0 nM
C=CC(=O)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(CO)c23)C1 CHEMBL5432828 IC50 9.0 nM
C#CC(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 CHEMBL5403826 IC50 10.0 nM
O=C(/C=C/CO)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(Cl)c23)C1 CHEMBL5428867 IC50 13.0 nM
C=CC(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncn(C)c2c1C#CCO CHEMBL5416415 IC50 93.0 nM
C=CC(=O)N1CCCN(CCCOCc2ccccc2)C1 CHEMBL5421419 IC50 160.0 nM
C=CC(=O)N1CCC(CCOc2ccccc2)CC1 CHEMBL5428462 IC50 610.0 nM
