CC(=O)Nc1ncc(Cc2csc(CCO)c2C)c(N)n1 CHEMBL255138 Kd 3.0 nM
CC(=O)OCCc1sc[n+](Cc2ccc(C)nc2N)c1C CHEMBL403691 EC50 4.7 nM
Cc1c(CCO)sc[n+]1Cc1ccc(N)nc1 CHEMBL255603 Kd 7.0 nM
CC(=O)OCC/C(SC(C)=O)=C(\C)N(C=O)Cc1ccc(C)nc1N CHEMBL252843 EC50 8.0 nM
C/C(=C(\CCO)SS/C(CCO)=C(/C)N(C=O)Cc1ccc(Cl)nc1N)N(C=O)Cc1ccc(Cl)nc1N CHEMBL402594 EC50 8.0 nM
Cc1cc(C)c(C[n+]2csc(CCO)c2C)c(N)n1 CHEMBL271044 EC50 8.3 nM
CCc1ccc(C[n+]2csc(CCO)c2C)c(N)n1 CHEMBL256627 EC50 8.7 nM
Cc1c(CCO)sc[n+]1Cc1ccc(Cl)nc1N CHEMBL401948 EC50 9.0 nM
Cc1c(CCO)sc[n+]1Cc1ccc(Cl)nc1N CHEMBL270613 EC50 9.0 nM
C/C(=C(\CCO)SS/C(CCO)=C(/C)N(C=O)Cc1ccc(C)nc1N)N(C=O)Cc1ccc(C)nc1N CHEMBL440237 EC50 12.0 nM
Cc1ncc(Cc2csc(CCO)c2C)c(N)n1 CHEMBL401772 Kd 12.0 nM
C/C(=C(\CCO)SSCCO)N(C=O)Cc1ccc(C)nc1N CHEMBL253045 EC50 13.0 nM
C/C(=C1\CCOC(=O)S1)N(C=O)Cc1ccc(C)nc1N CHEMBL252845 EC50 15.0 nM
Cc1ncc(Cn2c(C)c(CCOP(=O)(O)OP(=O)(O)O)sc2=O)c(N)n1 CHEMBL403021 Kd 16.0 nM
Cc1ccc(C[n+]2csc(CCO)c2C)c(N)n1 CHEMBL252086 EC50 18.0 nM
CCc1sc(CCO)c(C)[n+]1Cc1ccc(C)nc1N CHEMBL403212 EC50 21.0 nM
Cc1ccc(C[n+]2csc(CCOP(=O)(O)OP(=O)(O)O)c2C)c(N)n1 CHEMBL401817 Kd 22.0 nM
CC(=O)Nc1ccc(C[n+]2csc(CCO)c2C)c(N)n1 CHEMBL256831 Kd 23.0 nM
Cc1ccc(C[n+]2c(C)sc(CCO)c2C)c(N)n1 CHEMBL402329 Kd 25.0 nM
Cc1ccc(C[n+]2csc(CCO)c2CO)c(N)n1 CHEMBL402566 Kd 25.0 nM
Cc1ccc(C[n+]2csc([C@@H](O)CO)c2C)c(N)n1 CHEMBL255340 Kd 27.0 nM
C/C(=C(\CCOC(=O)c1ccccc1)SC(=O)c1ccccc1)N(C=O)Cc1ccc(C)nc1N CHEMBL252844 EC50 28.0 nM
Cc1ccc(C[n+]2c(C)sc(CCO)c2C)c(N)n1 CHEMBL252441 EC50 28.0 nM
Cc1ccc(C[n+]2csc([C@H](O)CO)c2C)c(N)n1 CHEMBL258077 Kd 28.0 nM
Cc1ccc(C[n+]2csc(CCO)c2)c(N)n1 CHEMBL256454 Kd 29.0 nM
Cc1ccc(C[n+]2c(C(C)O)sc(CCO)c2C)c(N)n1 CHEMBL255339 EC50 30.0 nM
CC(=O)N(Cc1ccc(C)nc1N)/C(C)=C(/CCO)SS/C(CCO)=C(/C)N(Cc1ccc(C)nc1N)C(C)=O CHEMBL251888 EC50 32.0 nM
Cc1ccc(C[n+]2cc(CCO)sc2C)c(N)n1 CHEMBL270632 Kd 36.0 nM
Cc1c(CCO)sc[n+]1Cc1cccnc1N CHEMBL403365 Kd 36.0 nM
CCc1c(CCO)sc[n+]1Cc1ccc(C)nc1N CHEMBL255541 Kd 40.0 nM
C/C(=C(\CCO)SSCCC(=O)O)N(C=O)Cc1ccc(C)nc1N CHEMBL401965 EC50 52.0 nM
Cc1ccc(C[n+]2csc(C(O)CO)c2C)c(N)n1 CHEMBL255542 Kd 53.0 nM
Cc1c(CCO)sc[n+]1Cc1ccc(C#N)nc1N CHEMBL429246 Kd 57.0 nM
Cc1c(Cc2cnc(C3CC3)nc2N)csc1CCO CHEMBL256177 Kd 60.0 nM
Cc1c(Cc2cnc(C(F)(F)F)nc2N)csc1CCO CHEMBL401572 Kd 63.0 nM
Cc1c(Cc2cnc(C(C)C)nc2N)csc1CCO CHEMBL255550 Kd 64.0 nM
Cc1c(CCO)sc[n+]1Cc1cnccc1N CHEMBL271521 Kd 64.0 nM
Cc1c(CCO)sc[n+]1Cc1ccc(C(F)(F)F)nc1N CHEMBL270168 Kd 104.0 nM
Cc1c(CCO)sc[n+]1Cc1cc(I)cnc1N CHEMBL270384 Kd 109.0 nM
Cc1c(CCO)sc[n+]1Cc1cccnc1N CHEMBL252637 EC50 110.0 nM
C/C(=C(\CCO)SCOC(=O)C(C)(C)C)N(C=O)Cc1ccc(C)nc1N CHEMBL253044 EC50 116.0 nM
Cc1c(CCO)sc[n+]1Cc1ccc(C(=O)c2ccccc2C(=O)O)nc1 CHEMBL402065 Kd 140.0 nM
Cc1ncc(C[n+]2csc(CCOP(C)(=O)OP(=O)(O)O)c2C)c(N)n1 CHEMBL430409 Kd 170.0 nM
Cc1cncc(C[n+]2csc(CCO)c2C)c1 CHEMBL256267 Kd 220.0 nM
Cc1c(Cc2cnc(-c3ccccc3)nc2N)csc1CCO CHEMBL255548 Kd 230.0 nM
Cc1c(CCO)sc[n+]1Cc1ccc(C(F)(F)F)nc1 CHEMBL257929 Kd 310.0 nM
C/C(=C(\CCO)SS/C(CCO)=C(/C)N(C=O)Cc1cccnc1N)N(C=O)Cc1cccnc1N CHEMBL251889 EC50 479.0 nM
Cc1ccc(C[n+]2c(Cc3cccnc3)sc(CCO)c2C)c(N)n1 CHEMBL404163 EC50 840.0 nM