COc1cc(C2=N/C(=C\c3cc(Br)cc(Br)c3OC(C)=O)C(=O)NN2c2ncc(-c3ccccc3)s2)cc(OC)c1OC CHEMBL4161876 IC50 6.85 nM
COc1cc(C2=N/C(=C\c3cc(Br)cc(Br)c3OC(C)=O)C(=O)NN2c2ccccc2)cc(OC)c1OC CHEMBL4174756 IC50 12.6 nM
Cc1ccc2c(=O)n(Cc3ccccc3)c(SCc3cn(-c4ccc(C(=O)O)cc4)nn3)nc2c1 CHEMBL5266387 IC50 25.8 nM
O=C1c2ccccc2C(=O)c2c(NCCNCCO)ccc(NCCNCCO)c21 CHEMBL49442 IC50 30.0 nM
COc1cc(C2=N/C(=C\c3cc(Br)cc(Br)c3OC(C)=O)C(=O)NN2C(N)=S)cc(OC)c1OC CHEMBL4160802 IC50 31.68 nM
COc1cc([C@@H]2c3cc4c(cc3[C@@H](O[C@@H]3O[C@@H]5CO[C@@H](C)O[C@H]5[C@H](O)[C@H]3O)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O CHEMBL44657 IC50 69.8 nM
COc1cc(C(=O)N/C(=C/c2cc(Br)cc(Br)c2OC(C)=O)C(=O)NNC(N)=S)cc(OC)c1OC CHEMBL4172196 IC50 81.42 nM
COc1cc(C2=N/C(=C\c3cc(Br)cc(Br)c3OC(C)=O)C(=O)n3c(C)nc(=S)n32)cc(OC)c1OC CHEMBL4169404 IC50 110.45 nM
Cc1cc(NC2=NC(=O)/C(=C\c3c4ccccc4cc4ccccc34)S2)no1 CHEMBL4751362 IC50 130.0 nM
CC[C@@](C)(Nc1ccnc(-c2c[nH]c3ncccc23)n1)C(=O)NCC(F)(F)F CHEMBL3039513 Kd apparent 148.0 nM
C[n+]1c2ccccc2cc2[n-]c3ccccc3c21 CHEMBL119096 MIC 250.0 nM
CCCCNc1c2ccccc2[n+](C)c2c1[nH]c1ccccc12 CHEMBL5194065 MIC 500.0 nM
Cc1[nH]c(C(=O)Nc2ccc(C(N)=O)cc2OCc2ccc(C(=O)NCCN)cc2)c(Cl)c1Cl CHEMBL5408150 IC50 550.0 nM
O=C(CN1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)cn3C2CC2)CC1)N/N=C/c1ccccc1O CHEMBL4213218 IC50 580.0 nM
COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(=O)CO)C[C@@H]3O[C@H]1C[C@H](N)[C@H](O)[C@H](C)O1 CHEMBL53463 IC50 727.0 nM
O=C(CN1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)cn3C2CC2)CC1)N/N=C/c1cc2ccccc2[nH]1 CHEMBL4205327 IC50 860.0 nM
Cc1cc(-c2c(F)cc3c4nn(CCN(C)C)c(=O)c-4cn(C4CC4)c3c2F)cc(C)n1 CHEMBL130381 EC50 930.0 nM
C[C@@H](Nc1cc(F)cc(F)c1)c1cc(C(=O)N(C)C)cc2c(=O)cc(N3CCOCC3)oc12 CHEMBL3408248 Kd apparent 936.0 nM
CN(C)CCNc1nc2c3ccc(O)cc3ccc2c2ccccc12 CHEMBL123828 MIC 1000.0 nM
COc1cc2c(NCCN(C)C)nc3c4cc5c(cc4ccc3c2cc1OC)OCO5 CHEMBL121582 MIC 1000.0 nM