CCOC(=O)N1CCC(c2cc(O)n3nc(C)c(-c4ccc(C(F)(F)F)cc4)c3n2)CC1 CHEMBL4085233 EC50 19.0 nM
CC1CCCN(C(=O)c2nc(Nc3cc4c(cc3F)OCO4)sc2Cl)C1C CHEMBL2418809 IC50 32.0 nM
CC1CCCN(C(=O)c2csc(Nc3ccc4c(c3)OCO4)n2)C1C CHEMBL2418807 IC50 80.0 nM
Cc1sc(Nc2ccc(Cl)cc2F)nc1C(=O)N1CCC[C@H](C)[C@@H]1C CHEMBL2418811 IC50 100.0 nM
Cc1nn2c(O)cc(C3CCN(C(=O)OCc4ccccc4)CC3)nc2c1-c1ccc(Cl)cc1 CHEMBL4060387 EC50 138.0 nM
Cc1sc(Nc2cc3c(cc2F)OCO3)nc1C(=O)N1CCCC(C)C1C CHEMBL2418808 IC50 160.0 nM
Cc1nn2c(O)cc(C3CCN(C(=O)OCc4ccccc4)CC3)nc2c1-c1ccc(F)cc1 CHEMBL4060400 EC50 236.0 nM
Cc1sc(Nc2ccc(Cl)cc2F)nc1C(=O)N1CCCC(C)C1C CHEMBL2418810 IC50 250.0 nM
Cc1ccc(Nc2nc(C(=O)N3CCCC(C)C3C)cs2)cc1 CHEMBL2418806 IC50 250.0 nM
N#Cc1ccc(O[C@@H]2c3ccccc3C[C@H]2N2CCC[C@@H](N)C2)c(Cl)c1 CHEMBL4129809 IC50 282.0 nM
Cc1sc(Nc2ccc3c(c2)OCO3)nc1C(=O)N1CCc2ccccc2C1C CHEMBL2418815 IC50 316.0 nM
CC1c2ccccc2CCN1C(=O)c1csc(Nc2ccc3c(c2)OCO3)n1 CHEMBL2418814 IC50 316.0 nM
CCNC(=O)c1cnn(-c2ccc(-n3ccc(Cl)c(Cl)c3=O)cc2)c1C(F)(F)F CHEMBL4761535 IC50 370.0 nM
CC1CCN(C(=O)c2csc(Nc3ccc4c(c3)OCO4)n2)CC1 CHEMBL2418823 IC50 400.0 nM
CCOC(=O)N1CCC(c2cc(O)n3nc(C)c(-c4ccc(F)cc4)c3n2)CC1 CHEMBL1496110 EC50 450.0 nM
CCOC(=O)c1cnn(-c2ccc(NC(=O)C(Cl)=C(Cl)Cl)cc2)c1C(F)(F)F CHEMBL4177187 IC50 470.0 nM
O=C(c1csc(Nc2ccc3c(c2)OCO3)n1)N1CCc2ccccc2C1 CHEMBL2418813 IC50 500.0 nM
Cc1ccc(Nc2nc(C(=O)N3CCC(C)CC3)cs2)cc1 CHEMBL2418818 IC50 630.0 nM
Cc1ccc(S(=O)(=O)Nc2ccc(-n3nc(C(F)(F)F)cc3C(F)(F)F)cc2)cc1 CHEMBL4460029 IC50 720.0 nM
Cc1ccc(Nc2nc(C(=O)N3CCCCC3C)cs2)cc1 CHEMBL2418824 IC50 800.0 nM
COc1ccc(Nc2nc(C(=O)N3CCC(C)CC3)cs2)cc1 CHEMBL2418820 IC50 800.0 nM
CC1CCN(C(=O)c2csc(Nc3ccc(Cl)cc3)n2)CC1 CHEMBL2418819 IC50 800.0 nM
Cc1sc(Nc2ccc(Cl)cc2F)nc1C(=O)N1CCC[C@@H](C)[C@H]1C CHEMBL2418812 IC50 1000.0 nM