O[C@H](c1ccccn1)[C@]1(c2cccc(OC(F)(F)F)c2)C[C@H](O)C1 CHEMBL3828010 Kb 40.0 nM
O[C@H](c1ccccn1)C1(c2ccc(OC(F)(F)F)cc2)CC(F)(F)C1 CHEMBL3827928 Kb 40.0 nM
O[C@H](c1ccccn1)[C@@]1(c2ccc(Cl)c(Cl)c2)CCCO1 CHEMBL3828066 Kb 43.0 nM
O[C@H](c1ccccn1)[C@]1(c2ccnc(C(F)(F)F)c2)C[C@H](O)C1 CHEMBL3827855 Kb 60.0 nM
O[C@H](c1ccccn1)[C@]1(c2cccc(OC(F)(F)F)c2)C[C@@H](O)C1 CHEMBL3827746 Kb 80.0 nM
O[C@H](c1ccccn1)C1(c2ccc(Cl)c(Cl)c2)CC(F)(F)C1 CHEMBL3828442 Kb 80.0 nM
O[C@H](c1ccccn1)C1(c2cccc(OC(F)(F)F)c2)CCC1 CHEMBL3828083 Kb 80.0 nM
O[C@H](c1ccccn1)C1(c2ccc(Cl)c(Cl)c2)CCC1 CHEMBL3828278 Kb 80.0 nM
CC(C)[C@H](CO)NCc1nc(C2=CCC(C(F)(F)F)CC2)ccc1F CHEMBL3696391 IC50 80.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc(F)cc(F)c2)ccc1F CHEMBL3696410 IC50 80.0 nM
O[C@H](c1ccccn1)[C@]1(c2cccc(C(F)(F)F)c2)C[C@H](O)C1 CHEMBL3827049 Kb 90.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCc3c(F)cccc3C2)ccc1F CHEMBL3692308 IC50 110.0 nM
CC(C)[C@H](CO)NCc1nc(N2Cc3cccc(F)c3C2)ccc1F CHEMBL3692305 IC50 120.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc3ccccc3n2C(=O)OC(C)(C)C)ccc1F CHEMBL3696433 IC50 120.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(F)c(Cl)c2)ccc1F CHEMBL3696452 IC50 120.0 nM
O[C@]1(c2ccccn2)CC[C@@H](c2ccc(C(F)(F)F)cc2)C1 CHEMBL3828290 Kb 130.0 nM
CC(C)[C@H](CO)NCc1nc(C#Cc2ccccc2)ccc1F CHEMBL3696448 IC50 130.0 nM
O[C@H](c1ccccn1)C1(c2ccc(OC(F)(F)F)cc2)CCC1 CHEMBL3827389 Kb 140.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)cn2)ccc1F CHEMBL3692284 IC50 140.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCc3cccc(F)c3C2)ccc1F CHEMBL3692310 IC50 140.0 nM
CC(C)[C@H](CO)NCc1nc(C2=CCC(F)(F)CC2)ccc1F CHEMBL3696392 IC50 140.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(F)c(F)c2)ccc1F CHEMBL3696396 IC50 140.0 nM
O[C@H](c1ccccn1)[C@]1(c2ccc(Cl)c(Cl)c2)CCO1 CHEMBL3827109 Kb 150.0 nM
CC(CCO)CNCc1nc(N2Cc3ccccc3C2)ccc1F CHEMBL3696458 IC50 160.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc(F)c(F)c(F)c2)ccc1F CHEMBL3696407 IC50 160.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(F)c(F)c2F)ccc1F CHEMBL3696408 IC50 160.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc(F)c(F)cc2F)ccc1F CHEMBL3696409 IC50 160.0 nM
CC(C)[C@@H](CO)NCc1nc(-c2ccc(C(F)(F)F)s2)ccc1F CHEMBL3696474 IC50 170.0 nM
CC(C)[C@H](CO)NCc1cccc(C#Cc2ccc(F)cc2)n1 CHEMBL3696426 IC50 170.0 nM
CC(C)[C@H](CO)NCc1nc(C#CCCC2CCCCC2)ccc1F CHEMBL3696447 IC50 170.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCc3ccccc3C2)ccc1F CHEMBL3692282 IC50 180.0 nM
CC(C)[C@H](CO)NCc1cccc(-c2ccc(F)c(C(F)(F)F)c2)n1 CHEMBL3696429 IC50 180.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(S(=O)(=O)N(C)C(C)(C)C)c2)ccc1F CHEMBL3692275 IC50 190.0 nM
CC(C)[C@H](CO)NCc1cccc(C#Cc2ccc(F)c(F)c2)n1 CHEMBL3696427 IC50 190.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F CHEMBL3692233 IC50 200.0 nM
O[C@H](c1ccccn1)[C@]1(c2cccc(C(F)(F)F)c2)C[C@@H](O)C1 CHEMBL3827938 Kb 210.0 nM
OCC1(NCc2cccc(-c3cc(C(F)(F)F)cc(C(F)(F)F)c3)n2)CCCC1 CHEMBL3696473 IC50 220.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCC(C(F)(F)F)CC2)ccc1F CHEMBL3692279 IC50 220.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(OC(F)(F)F)cc2)ccc1F CHEMBL3692235 IC50 230.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc3sccc3c2)ccc1F CHEMBL3696418 IC50 230.0 nM
O[C@@]1(c2ccccn2)CC[C@@H](c2ccc(C(F)(F)F)cc2)C1 CHEMBL3828640 Kb 240.0 nM
Cc1cc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)ccc1F CHEMBL3696439 IC50 250.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCc3ccc(C(F)(F)F)cc3C2)ccc1F CHEMBL3692313 IC50 260.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc3ccccc3[nH]2)ccc1F CHEMBL3696434 IC50 260.0 nM
COc1cc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)cc(F)c1F CHEMBL3696442 IC50 260.0 nM
O[C@H](c1ccccn1)[C@]1(c2cc(C(F)(F)F)ccn2)C[C@H](O)C1 CHEMBL3828720 Kb 270.0 nM
CC(C)[C@H](CO)NCc1nc(N2Cc3ccc(F)cc3C2)ccc1F CHEMBL3692304 IC50 270.0 nM
C[C@]1(O)C[C@@](c2cccc(OC(F)(F)F)c2)([C@H](O)c2ccccn2)C1 CHEMBL3828294 Kb 280.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cncc(C(F)(F)F)c2)ccc1F CHEMBL3696450 IC50 280.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)c(Cl)c2)ccc1F CHEMBL3692261 IC50 290.0 nM
OCC1(NCc2nc(-c3ccc(C(F)(F)F)cc3)ccc2F)CCCC1 CHEMBL3692291 IC50 290.0 nM
CC(C)[C@H](CO)NCc1nc(C#Cc2ccc(F)cc2)ccc1F CHEMBL3696403 IC50 290.0 nM
CC(C)[C@H](CO)NCc1nc([C@H]2CC[C@H](C(F)(F)F)CC2)ccc1F CHEMBL3696421 IC50 290.0 nM
C[C@]1(O)C[C@@](c2cccc(C(F)(F)F)c2)([C@H](O)c2ccccn2)C1 CHEMBL3827863 Kb 300.0 nM
CC(O)C(C)NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F CHEMBL3692297 IC50 300.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(-n3cccn3)c2)ccc1F CHEMBL3696423 IC50 300.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCC(C(F)(F)F)CC2)ccc1F CHEMBL3696384 IC50 310.0 nM
O[C@H](c1ccccn1)[C@]1(c2cc(C(F)(F)F)ccn2)C[C@@H](O)C1 CHEMBL3828190 Kb 320.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(F)cc2)ccc1F CHEMBL3692242 IC50 320.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCCC(C(F)(F)F)C2)ccc1F CHEMBL3639911 IC50 320.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCc3ccc(F)cc3C2)ccc1F CHEMBL3692309 IC50 320.0 nM
C[C@]1(O)C[C@@](c2ccc(OC(F)(F)F)cc2)([C@H](O)c2ccccn2)C1 CHEMBL3828134 Kb 330.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(S(=O)(=O)N3CCCCC3)c2)ccc1F CHEMBL3692262 IC50 330.0 nM
CC(C)[C@H](CO)NCc1nc(N2Cc3ccc(C(F)(F)F)cc3C2)ccc1F CHEMBL3692307 IC50 330.0 nM
CC(C)[C@H](CO)NCc1nc(N2Cc3cccc(Cl)c3C2)ccc1F CHEMBL3692306 IC50 340.0 nM
CC(C)[C@H](CO)NCc1nc([C@H]2CC[C@@H](C(F)(F)F)CC2)ccc1F CHEMBL3696420 IC50 340.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCc3c(cccc3C(F)(F)F)C2)ccc1F CHEMBL3692312 IC50 350.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCc3ccccc3C2)ccc1F CHEMBL3696385 IC50 350.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc3ccccc3n2C)ccc1F CHEMBL3696412 IC50 350.0 nM
CC(O)CC(C)CNCc1nc(C2CCCCC2)ccc1F CHEMBL3696459 IC50 360.0 nM
O[C@H](c1ncccn1)C1(c2ccc(Cl)c(Cl)c2)CCC1 CHEMBL3827447 Kb 370.0 nM
CC(C)[C@@H](CO)NCc1nc(CCc2ccc(F)c(F)c2)ccc1F CHEMBL3696469 IC50 370.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc3ccccc3s2)ccc1F CHEMBL3696397 IC50 370.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc(C(F)(F)F)ccc2F)ccc1F CHEMBL3696441 IC50 370.0 nM
O[C@H](c1ccccn1)[C@@]1(c2ccc(Cl)c(Cl)c2)CCO1 CHEMBL3827001 Kb 380.0 nM
C[C@]1(O)C[C@](c2cc(C(F)(F)F)ccn2)([C@H](O)c2ccccn2)C1 CHEMBL3828340 IC50 380.0 nM
CC(C)[C@H](CO)NCc1nc(/C=C/c2cccc(F)c2)ccc1F CHEMBL3696399 IC50 380.0 nM
Cc1ccc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)s1 CHEMBL3696406 IC50 380.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(Cl)cc2)ccc1F CHEMBL3692256 IC50 390.0 nM
OCC1(NCc2cccc(-c3ccc(F)c(Cl)c3)n2)CCCC1 CHEMBL3696428 IC50 390.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(F)c(C(F)(F)F)c2)ccc1F CHEMBL3696440 IC50 390.0 nM
OC[C@@H](NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F)C1CC1 CHEMBL3696456 IC50 410.0 nM
CC(C)[C@@H](CO)NCc1nc(-c2ccc(Cl)s2)ccc1F CHEMBL3696470 IC50 410.0 nM
C[C@]1(c2ccc(OC(F)(F)F)cc2)C[C@](O)(c2ccccn2)CO1 CHEMBL3828376 Kb 420.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCC(C(F)(F)F)C2)ccc1F CHEMBL3692280 IC50 420.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc3occc3c2)ccc1F CHEMBL3696419 IC50 420.0 nM
OCC1(NCc2cccc(-c3ccc(F)c(C(F)(F)F)c3)n2)CCCC1 CHEMBL3696430 IC50 420.0 nM
CC(C)[C@H](CO)NCc1cccc(-c2ccc(F)c(C#N)c2)n1 CHEMBL3696431 IC50 440.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(N(C)C)c2)ccc1F CHEMBL3692257 IC50 460.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(OCC(F)(F)F)cc2)ccc1F CHEMBL3692267 IC50 460.0 nM
CCC[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F CHEMBL3692294 IC50 460.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)cc2)ncc1F CHEMBL3692338 IC50 460.0 nM
O[C@H](c1ccccn1)[C@]1(c2ccc(Cl)c(Cl)c2)CCCO1 CHEMBL3827886 Kb 470.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(N3CCCC3)c2)ccc1F CHEMBL3692263 IC50 480.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc3ccn(C)c3c2)ccc1F CHEMBL3692278 IC50 480.0 nM
CC(c1ccc(F)cc1)c1ccc(F)c(CN[C@@H](CO)C(C)C)n1 CHEMBL3692337 IC50 480.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCCC2)ccc1F CHEMBL3696388 IC50 480.0 nM
C[C@]1(O)C[C@](c2ccnc(C(F)(F)F)c2)([C@H](O)c2ccccn2)C1 CHEMBL3827043 Kb 500.0 nM
CCN(CC)S(=O)(=O)c1cccc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)c1 CHEMBL3692265 IC50 500.0 nM
CC(C)Oc1ccc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)cn1 CHEMBL3692271 IC50 500.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCc3cc(Cl)ccc3C2)ccc1F CHEMBL3692311 IC50 500.0 nM
CC(C)(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)nc2)ccc1F CHEMBL3692300 IC50 510.0 nM
CC[C@@H](NCc1nc(-c2ccc(C(F)(F)F)nc2)ccc1F)C(C)O CHEMBL3692324 IC50 510.0 nM
CC(C)[C@H](CO)NCc1nc(C#CC2CCCCC2)ccc1F CHEMBL3696404 IC50 510.0 nM
CC(C)(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F CHEMBL3692296 IC50 520.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc3c(OCc4ccccc4)cccc3n2C(=O)OC(C)(C)C)ccc1F CHEMBL3696422 IC50 520.0 nM
CC(C)[C@H](CO)NCc1cccc(C#Cc2ccc(F)cc2F)n1 CHEMBL3696443 IC50 520.0 nM
CC(C)[C@H](CO)NCc1cccc(C#Cc2ccc(Cl)cc2)n1 CHEMBL3696445 IC50 520.0 nM
O[C@H](c1ccccn1)[C@]1(c2ccnc(C(F)(F)F)c2)C[C@@H](O)C1 CHEMBL3828220 Kb 530.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCC(F)(F)CC2)ccc1F CHEMBL3696372 IC50 530.0 nM
O[C@]1(c2ccccn2)CC[C@H](c2ccc(C(F)(F)F)cc2)C1 CHEMBL3827263 Kb 540.0 nM
CC[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F CHEMBL3692288 IC50 540.0 nM
CC(C)[C@@H](NCc1nc(-c2ccc(C(F)(F)F)nc2)ccc1F)C(C)O CHEMBL3692317 IC50 540.0 nM
OC(c1ccccn1)C1(c2ccccc2OC(F)(F)F)CCC1 CHEMBL3828484 Kb 550.0 nM
CC(C)[C@H](CO)NCc1cccc(-c2ccc(C(F)(F)F)cc2C(F)(F)F)n1 CHEMBL3696432 IC50 550.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)cc2C(F)(F)F)ccc1F CHEMBL3696451 IC50 550.0 nM
OC[C@H](NCc1nc(-c2ccc(C(F)(F)F)nc2)ccc1F)C1CCCCC1 CHEMBL3692299 IC50 570.0 nM
OCC1(NCc2cccc(-c3ccc(C(F)(F)F)cc3C(F)(F)F)n2)CCCC1 CHEMBL3696472 IC50 580.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccoc2)ccc1F CHEMBL3696414 IC50 580.0 nM
CC(CCO)CNCc1ccc(F)c(-c2ccc(OCC(F)(F)F)nc2)n1 CHEMBL3696457 IC50 590.0 nM
CC(C)[C@H](CO)NCc1cccc(-c2cccc([Si](C)(C)C)c2)n1 CHEMBL3696394 IC50 600.0 nM
O[C@@]1(c2ccccn2)CC[C@H](c2ccc(C(F)(F)F)cc2)C1 CHEMBL3827897 Kb 610.0 nM
OC(c1ncccc1F)C1(c2ccc(Cl)c(Cl)c2)CCC1 CHEMBL3827600 Kb 610.0 nM
COc1ccc(-c2cc(=O)c3c(O)cc(O)cc3o2)cc1 CHEMBL243664 IC50 620.0 nM
OC(c1ccccn1)C1(c2ccc(Cl)c(Cl)c2)CCOC1 CHEMBL3828719 Kb 630.0 nM
Cc1ccc(S(=O)(=O)C(F)(F)F)cc1-c1ccc(F)c(CN[C@@H](CO)C(C)C)n1 CHEMBL3692273 IC50 630.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)nc2)ccc1Cl CHEMBL3692319 IC50 630.0 nM
OC(c1cc(F)ccn1)C1(c2ccc(Cl)c(Cl)c2)CCC1 CHEMBL3827217 Kb 640.0 nM
CC(C)Oc1ccc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)cc1F CHEMBL3692241 IC50 650.0 nM
CCCN(CCC)C(=O)c1ccc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)cc1 CHEMBL3639953 IC50 650.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCCN(C(=O)OC(C)(C)C)C2)ccc1F CHEMBL3696387 IC50 660.0 nM
OCC1(NCc2nc(-c3ccc(C(F)(F)F)cc3)ccc2F)CCCCC1 CHEMBL3692292 IC50 680.0 nM
CC(C)[C@H](CO)NCc1ccnc(-c2ccc(S(=O)(=O)C(F)(F)F)cc2)n1 CHEMBL3696375 IC50 680.0 nM
CC(C)Oc1ccc(F)c(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)c1 CHEMBL3692239 IC50 700.0 nM
OCC1(NCc2nc(-c3ccc(C(F)(F)F)cc3)ccc2F)CCC1 CHEMBL3692290 IC50 700.0 nM
OC[C@H](NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F)C1CCCCC1 CHEMBL3692295 IC50 700.0 nM
CC(C)[C@@H](NCc1nc(-c2ccc(C(F)(F)F)cc2)ccc1F)C(C)O CHEMBL3692316 IC50 700.0 nM
Cc1cc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)cnc1N1CCOCC1 CHEMBL3696416 IC50 700.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCN(C(=O)OC(C)(C)C)C2)ccc1F CHEMBL3696390 IC50 710.0 nM
COc1cccc(CNC(=O)CC2CC3(CCC3)Oc3ccc(Cl)cc32)c1OC1CCCC1 CHEMBL3664218 IC50 725.3 nM
C[C@]1(O)C[C@@](c2cc(C(F)(F)F)ccn2)([C@H](O)c2ccccn2)C1 CHEMBL3828557 Kb 730.0 nM
Cc1nc(-c2ccccc2)sc1-c1ccc(F)c(CN[C@@H](CO)C(C)C)n1 CHEMBL3696446 IC50 730.0 nM
CC(C)[C@H](CO)NCc1nc(C2=CCCCC2)ccc1F CHEMBL3692335 IC50 740.0 nM
CC(C)Oc1cccc(-c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)c1 CHEMBL3692240 IC50 750.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cnc(N(C)C)nc2)ccc1F CHEMBL3696424 IC50 750.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(S(=O)(=O)N3CCOCC3)c2)ccc1F CHEMBL3692268 IC50 760.0 nM
CCC1CCC(c2ccc(F)c(CN[C@@H](CO)C(C)C)n2)CC1 CHEMBL3696370 IC50 770.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCC(C)(C)CC2)ccc1F CHEMBL3696371 IC50 790.0 nM
CC(C)[C@H](CO)NCc1nc(C2CCC(C(C)(C)C)CC2)ccc1F CHEMBL3696381 IC50 790.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cc(C(F)(F)F)nn2C)ccc1F CHEMBL3696449 IC50 790.0 nM
CCCCOc1ccc(-c2cccc(CN[C@H](CO)C(C)C)n2)cc1Cl CHEMBL3696471 IC50 810.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(F)c2)ccc1F CHEMBL3692230 IC50 810.0 nM
CC(C)[C@H](CO)NCc1nc(-c2cccc(N3CCOCC3)c2)ccc1F CHEMBL3692258 IC50 830.0 nM
C[C@]1(O)C[C@@](c2ccc(C(F)(F)F)cc2)([C@H](O)c2ccccn2)C1 CHEMBL3828490 Kb 840.0 nM
OC(c1ccc(F)cn1)C1(c2ccc(Cl)c(Cl)c2)CCC1 CHEMBL3828433 Kb 910.0 nM
CC(C)[C@H](CO)NCc1cccc(OCc2ccccc2)n1 CHEMBL3692228 IC50 910.0 nM
C=C(c1ccccc1)c1ccc(F)c(CN[C@@H](CO)C(C)C)n1 CHEMBL3692333 IC50 920.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(F)c(C#N)c2)ccc1F CHEMBL3696438 IC50 940.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(C(F)(F)F)nc2)ccc1F CHEMBL3692243 IC50 950.0 nM
CC(C)[C@H](CO)NCc1nc(-c2ccc(F)cn2)ccc1F CHEMBL3692250 IC50 950.0 nM
CC(C)[C@H](CO)NCc1nc(N2CCC(F)(F)CC2)ccc1F CHEMBL3692303 IC50 960.0 nM
CC(C)[C@H](CO)NCc1nc(C#CCC2CCCCC2)ccc1F CHEMBL3696401 IC50 980.0 nM
CC(C)[C@H](CO)NCc1cccc(C#Cc2ccccc2F)n1 CHEMBL3696444 IC50 990.0 nM
CCCCCc1cc(O)c(C/C=C(\C)CCC=C(C)C)c(O)c1 CHEMBL497318 EC50 1000.0 nM