N#CN1CC[C@H](C(=O)Nc2nc3c(s2)CN(C(=O)CN=[N+]=[N-])CC3)C1 CHEMBL4802050 IC50 230.0 nM
N#CN1CCC(C(=O)Nc2ncc(N3CCOCC3)s2)C1 CHEMBL5191704 IC50 230.0 nM
CC(=O)O/N=C1\C(=O)N(Cc2cc(Cl)ccc2Cl)c2ccc(Cl)cc21 CHEMBL3407553 Ki 400.0 nM
N#CN1CC[C@H](C(=O)Nc2ncc(-c3ccccc3)s2)C1 CHEMBL5169766 IC50 550.0 nM
C#Cc1ccc(-c2cnc(NC(=O)[C@H]3CCN(C#N)C3)s2)cc1 CHEMBL5192316 IC50 600.0 nM
N#CN1CCCC1C(=O)n1ccc2c(-c3cn[nH]c3C(F)(F)F)cccc21 CHEMBL5175498 IC50 670.0 nM
Nc1c(C(=O)c2ccc3ccccc3c2)sc2[nH]c(=O)c(C(=O)O)cc12 CHEMBL540117 Ki app 740.0 nM
CC(=O)O/N=C1/C(=O)N(Cc2ccc(Cl)c(Cl)c2)c2ccc(Br)cc21 CHEMBL1241672 IC50 810.0 nM
CC(=O)O/N=C1/C(=O)N(Cc2cc(Cl)ccc2Cl)c2ccc(Br)cc21 CHEMBL1241673 IC50 880.0 nM
Cc1ccc(C(=O)c2sc3[nH]c(=O)c(C(=O)O)cc3c2N)cc1 CHEMBL553923 Ki app 910.0 nM
CC(=O)O/N=C1/C(=O)N(Cc2ccc(Cl)c(Cl)c2)c2ccc(I)cc21 CHEMBL1241765 IC50 940.0 nM
