CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)N[C@@H](C)COC(F)(F)F)CC3)nc12 CHEMBL4785914 IC50 0.2 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)NCCOC(F)(F)F)CC3)nc12 CHEMBL4796521 IC50 0.4 nM
CC[C@H](C)NC(=O)OC1CCN(c2cc(C(F)(F)F)c3scc(C(=O)NC)c3n2)CC1 CHEMBL4787939 IC50 0.4 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)N[C@@H](C)C4CC4)CC3)nc12 CHEMBL4750073 IC50 0.9 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)NCC4CC4)CC3)nc12 CHEMBL4776963 IC50 1.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)N4CC(OC(F)(F)F)C4)CC3)nc12 CHEMBL4750432 IC50 1.7 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)NC(C)C)CC3)nc12 CHEMBL4765010 IC50 2.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(NC(=O)OCC4CC4)CC3)nc12 CHEMBL4755797 IC50 18.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CC(NC(=O)OCC4CC4)C3)nc12 CHEMBL4757982 IC50 43.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCN(CC(=O)NC(C)C)CC3)nc12 CHEMBL4760937 IC50 67.0 nM
CCC(=O)c1csc2c(C(F)(F)F)cc(N3CCN(CC(=O)NC(C)C)CC3)nc12 CHEMBL4795937 IC50 97.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCN(C(C)C(=O)NC4CC4)CC3)nc12 CHEMBL4799472 IC50 170.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCN(CC(O)COC(C)(C)C)CC3)nc12 CHEMBL4797076 IC50 190.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CC(OC(=O)NCC4CC4)C3)nc12 CHEMBL4764180 IC50 200.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCN(CCOC(C)C)CC3)nc12 CHEMBL4751927 IC50 200.0 nM
CC(C)NC(=O)CN1CCN(c2cc(C(F)(F)F)c3scc(C(=O)N4CCC4)c3n2)CC1 CHEMBL4747085 IC50 320.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCN(C(=O)COC(C)C)CC3)nc12 CHEMBL4745037 IC50 450.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)NCCN4CCCC4)CC3)nc12 CHEMBL4799203 IC50 510.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCN(CC(=O)C(C)(C)C)CC3)nc12 CHEMBL4791074 IC50 610.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)NCC4CC4)C3)nc12 CHEMBL4762406 IC50 610.0 nM
CNC(=O)c1csc2c(C(F)(F)F)cc(N3CCC(OC(=O)N4CC(CN(C)C)C4)CC3)nc12 CHEMBL4752928 IC50 980.0 nM