C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N3CCNCC3)c(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5087368 EC50 9.9 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2CC(c3ccccc3)=CC2=O)C2(CCCC2)C1 CHEMBL5428753 IC50 49.0 nM
CC(CC1CCCCC1)C(=O)N1CCC(CN2Cc3c(C(=O)N(C)C)cccc3C2=O)C2(CCCC2)C1 CHEMBL5429248 IC50 58.0 nM
Cc1ccc2c(c1)CN(C[C@]1(O)CCN(C(=O)[C@H](C)CC3CCCCC3)CC13CCCC3)C2=O CHEMBL5396358 IC50 74.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2C[C@H](c3ccccc3)CC2=O)C2(CCCC2)C1 CHEMBL5433263 IC50 110.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2C[C@@H](c3ccc(Cl)cc3)CC2=O)C2(CCCC2)C1 CHEMBL5396766 IC50 110.0 nM
COc1cccc([C@H]2CC(=O)N(C[C@]3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)C2)c1 CHEMBL5417864 IC50 120.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2C[C@@H](c3ccccc3)CC2=O)C2(CCCC2)C1 CHEMBL5432985 IC50 140.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2Cc3c(C(=O)N(C)C)cccc3C2=O)C2(CCCC2)C1 CHEMBL5439024 IC50 150.0 nM
Cc1ccccc1[C@@H]1CC(=O)N(C[C@]2(O)CCN(C(=O)[C@H](C)CC3CCCCC3)CC23CCCC3)C1 CHEMBL5428250 IC50 150.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2Cc3cc(C(=O)N(C)C)ccc3C2=O)C2(CCCC2)C1 CHEMBL5439171 IC50 190.0 nM
COc1cccc([C@@H]2CC(=O)N(C[C@]3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)C2)c1 CHEMBL5431080 IC50 210.0 nM
Cc1ccc([C@H]2CC(=O)N(C[C@]3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)C2)cc1 CHEMBL5403806 IC50 220.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2Cc3c(cccc3-c3ncco3)C2=O)C2(CCCC2)C1 CHEMBL5429133 IC50 280.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2Cc3c(cccc3-n3cccn3)C2=O)C2(CCCC2)C1 CHEMBL5400910 IC50 280.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2C[C@H](c3ccc(Cl)cc3)CC2=O)C2(CCCC2)C1 CHEMBL5437136 IC50 290.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2C[C@@](C)(c3ccccc3)CC2=O)C2(CCCC2)C1 CHEMBL5421217 IC50 320.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2Cc3c(Cl)cccc3C2=O)C2(CCCC2)C1 CHEMBL5412764 IC50 440.0 nM
Cc1ccc([C@@H]2CC(=O)N(C[C@]3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)C2)cc1 CHEMBL5403412 IC50 450.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(-c3cccc(C(N)=O)c3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5092219 IC50 500.0 nM
CC(C)N(C)C(=O)c1cn(CC2(O)CCN(C(=O)C3(C)CCc4ccccc4C3)CC2)c(=O)cc1-c1ccccc1F CHEMBL5083472 IC50 500.0 nM
CC(C)C(CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccccc3F)cc2=O)C(C)(C)C1 CHEMBL5084401 IC50 500.0 nM
C[C@H](Cc1ccccc1)C(=O)N1C[C@H]2CC[C@@H](C1)C2(O)Cn1cnc(-c2ccccc2F)cc1=O CHEMBL5094385 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(C(=O)N3CCCCC3)c(-c3ccccc3)cc2=O)CC1 CHEMBL5080439 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccccc3F)cc2=O)C2(CCC2)C1 CHEMBL5087762 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3cccc(CN)c3)c(-c3ccccc3F)cc2=O)CC1 CHEMBL5089604 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C(C)(C)C1)c1ccccc1 CHEMBL5086698 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N3CCC(O)CC3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5073032 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N3CCCC3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5074955 IC50 500.0 nM
CCN(CC)C(=O)c1cn(CC2(O)CCN(C(=O)C[C@@H](C)c3ccccc3)CC2)c(=O)cc1-c1ccccc1 CHEMBL5078256 IC50 500.0 nM
CC(CC(=O)N1CCC(O)(Cn2cnc(-c3ccccc3F)cc2=O)C(C)(C)C1)C1CCCCC1 CHEMBL5084536 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N3CCOCC3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5079191 IC50 500.0 nM
CC1(C)CN(C(=O)CCC2CCCCC2)CCC1(O)Cn1cnc(-c2ccccc2F)cc1=O CHEMBL5071270 IC50 500.0 nM
CC(C)N(C)C(=O)c1cn(CC2(O)CCN(C(=O)CCC3CCC3)CC2(C)C)c(=O)cc1-c1ccccc1 CHEMBL5086699 IC50 500.0 nM
CC(C)N(C)C(=O)c1cn(CC2(O)CCN(C(=O)[C@H](C)CC3CCCCC3)CC2)c(=O)cc1-c1ccccc1 CHEMBL5092836 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N3CCCCC3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5080532 IC50 500.0 nM
COc1ccccc1-c1cc(=O)n(CC2(O)CCN(C(=O)C[C@@H](C)c3ccccc3)CC2)cc1C(=O)N(C)C(C)C CHEMBL5085024 IC50 500.0 nM
CC(C)N(C)C(=O)c1cn(CC2(O)CCN(C(=O)C[C@@H](C)c3ccccc3)CC2)c(=O)cc1-c1ccccc1F CHEMBL5084246 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(-c3ccccn3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5079208 IC50 500.0 nM
CC(C)N(C)C(=O)c1cn(CC2(O)CCN(C(=O)CCC3CCCCC3)CC2)c(=O)cc1-c1ccccc1 CHEMBL5092530 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N3CCNCC3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5091123 IC50 500.0 nM
Cc1cccc(-c2cc(=O)n(CC3(O)CCN(C(=O)C[C@@H](C)c4ccccc4)CC3)cc2C(=O)N(C)C(C)C)c1 CHEMBL5084479 IC50 500.0 nM
CC(n1cnc(-c2ccccc2)cc1=O)C1(O)CCN(C(=O)[C@H](C)Cc2ccccc2)CC1 CHEMBL5082843 IC50 500.0 nM
C=CC[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccccc3F)cc2=O)CC1 CHEMBL5088608 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N3CCC[C@@H]3C)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5086483 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N3CCC(CO)CC3)c(-c3ccccc3)cc2=O)CC1)c1ccccc1 CHEMBL5075341 IC50 500.0 nM
CCC(CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccccc3F)cc2=O)C(C)(C)C1 CHEMBL5092121 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(C(=O)N(C)C)ccc2=O)C2(CCCC2)C1 CHEMBL5086611 IC50 500.0 nM
C[C@H](CC1CCC1)C(=O)N1CCC(O)(Cn2cc(C(=O)N(C)C)c(-c3ccccc3)cc2=O)C(C)(C)C1 CHEMBL5077649 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3cncnc3)cc2=O)C(C)(C)C1 CHEMBL5086805 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccnn3C)cc2=O)C(C)(C)C1 CHEMBL5087065 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccn[nH]3)cc2=O)C(C)(C)C1 CHEMBL5088091 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3ncco3)c(-c3ccccc3)cc2=O)C(C)(C)C1 CHEMBL5085329 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccccc3CO)cc2=O)C(C)(C)C1 CHEMBL5074660 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3ccc(CN)cc3)cc2=O)C(C)(C)C1 CHEMBL5092525 IC50 500.0 nM
CN(C)C(=O)c1cn(CC2(O)CCN(C(=O)[C@H](COCc3ccccc3)CC3CCCCC3)CC2(C)C)c(=O)cc1-c1ccccc1 CHEMBL5093482 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc(-c3cccc(CN)c3)cc2=O)C(C)(C)C1 CHEMBL5083163 IC50 500.0 nM
CN(C)C(=O)c1cn(CC2(O)CCN(C(=O)C[C@H](c3ccccc3)C(F)F)CC23CCCC3)c(=O)cc1-c1ccccc1 CHEMBL5092302 IC50 500.0 nM
CN(C)C(=O)c1cn(CC2(O)CCN(C(=O)CCc3ccc(F)cc3)CC23CCCC3)c(=O)cc1-c1ccccc1 CHEMBL5085999 IC50 500.0 nM
C[C@H](CC(=O)N1CCC(O)(Cn2cc(C(=O)N(C)C)c(-c3ccccc3)cc2=O)C2(CCCC2)C1)c1ccccc1 CHEMBL5074806 IC50 500.0 nM
CN(C)C(=O)c1cn(CC2(O)CCN(C(=O)c3c[nH]nc3-c3ccccc3)CC23CCCC3)c(=O)cc1-c1ccccc1 CHEMBL5083450 IC50 500.0 nM
CN(C)C(=O)c1cn(CC2(O)CCN(C(=O)C3CCC(C(F)(F)F)C3)CC23CCCC3)c(=O)cc1-c1ccccc1 CHEMBL5077844 IC50 500.0 nM
CC1(C)CN(C(=O)[C@H](CO)CC2CCC2)CCC1(O)Cn1cnc(-c2ccccc2F)cc1=O CHEMBL5076530 IC50 500.0 nM
CN(C)C(=O)c1cn(CC2(O)CCN(C(=O)C(O)Cc3ccccc3)CC23CCCC3)c(=O)cc1-c1ccccc1 CHEMBL5084890 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N(C)C)c(-c3ccccc3)cc2=O)C(C)(C)C1 CHEMBL5092372 IC50 500.0 nM
CN(C)C(=O)c1cn(C[C@]2(O)CCN(C(=O)C(CC(F)(F)F)CC(F)(F)F)CC23CCCC3)c(=O)cc1-c1ccccc1 CHEMBL5078851 IC50 500.0 nM
O=C(c1cn(C[C@]2(O)CCN(C(=O)C(CC(F)(F)F)CC(F)(F)F)CC23CCCC3)c(=O)cc1-c1ccccc1)N1CCCCC1 CHEMBL5078396 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N(C)C)c(C3CC3)cc2=O)C(C)(C)C1 CHEMBL5090274 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N3CCNCC3)c(C3CC3)cc2=O)C(C)(C)C1 CHEMBL5079446 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N(C)C)c(-c3ccccc3F)cc2=O)C2(CCCC2)C1 CHEMBL5089266 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N3CCNCC3)c(-c3ccccc3F)cc2=O)C2(CCCC2)C1 CHEMBL5087406 IC50 500.0 nM
C[C@H](CC1CCC1)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N(C)C)c(C3CC3)cc2=O)C2(CCCC2)C1 CHEMBL5069760 IC50 500.0 nM
C[C@H](CC1CCC1)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N3CCNCC3)c(C3CC3)cc2=O)C2(CCCC2)C1 CHEMBL5087127 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N(C)C)c(-c3ccccc3)cc2=O)C2(CCOCC2)C1 CHEMBL5093308 IC50 500.0 nM
C[C@H](CC1CCC1)C(=O)N1CC[C@@](O)(Cn2cc(C(=O)N(C)C)c(-c3ccccc3F)cc2=O)C(C)(C)C1 CHEMBL5077081 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(C(=O)O)c(-c3ccccc3)cc2=O)C(C)(C)C1 CHEMBL5091404 IC50 500.0 nM
COc1cc(=O)n(CC2(O)CCN(C(=O)[C@H](C)CC3CCCCC3)CC23CCCC3)cc1C(=O)N(C)C CHEMBL5075817 IC50 500.0 nM
C[C@H](CC1CCC1)C(=O)N1CCC(O)(Cn2ccncc2=O)C2(CCCC2)C1 CHEMBL5086853 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3ccccc3)ncc2=O)C(C)(C)C1 CHEMBL5079633 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2ccncc2=O)C2(CCCC2)C1 CHEMBL5080732 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2ccncc2=O)C(C)(C)C1 CHEMBL5087664 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc3cc(Cl)ccc3c2=O)C2(CCCC2)C1 CHEMBL5091408 IC50 500.0 nM
Cc1nc2ccccc2c(=O)n1CC1(O)CCN(C(=O)[C@H](C)CC2CCCCC2)CC12CCCC2 CHEMBL5078047 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3ccccc3)c(N=S(C)(C)=O)cc2=O)C2(CCCC2)C1 CHEMBL5090357 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3cccnc3)ncc2=O)C2(CCCC2)C1 CHEMBL5088815 IC50 500.0 nM
COc1ccc2ccn(CC3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)c(=O)c2c1 CHEMBL5087099 IC50 500.0 nM
CNc1ncc2c(=O)n(CC3(O)CCN(C(=O)[C@H](C)CC(F)(F)F)CC34CCCC4)ccc2n1 CHEMBL5070748 IC50 500.0 nM
O=C1Cn2ccnc2CN1CC1(O)CCN(C(=O)N2CCNC[C@H]2c2ccccc2)CC12CCCC2 CHEMBL5083942 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2CCN(S(C)(=O)=O)CC2=O)C2(CCCC2)C1 CHEMBL5089640 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-n3cccn3)ncc2=O)C(C)(C)C1 CHEMBL5077418 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2Cc3ncccc3C2=O)C2(CCCC2)C1 CHEMBL5082237 IC50 500.0 nM
CSc1ncc2c(=O)n(CC3(O)CCN(C(=O)[C@H](C)CC(F)(F)F)CC34CCCC4)n(C)c2n1 CHEMBL5085350 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2CC(Cc3ccccc3)CC2=O)C2(CCCC2)C1 CHEMBL5087230 IC50 500.0 nM
O=C1COCCN1CC1(O)CCN(C(=O)N2CCNC[C@H]2c2ccccc2)CC12CCCC2 CHEMBL5093996 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3ccn[nH]3)ncc2=O)C(C)(C)C1 CHEMBL5087291 IC50 500.0 nM
Cc1cccc2c(=O)n(CC3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)cnc12 CHEMBL5075471 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2ccc3nc(N4CCNCC4)ncc3c2=O)C2(CCCC2)C1 CHEMBL5084125 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2C[C@H](c3ccccc3)CC2=O)C2(CCCC2)C1 CHEMBL5074476 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(C(=O)O)ncc2=O)C2(CCCC2)C1 CHEMBL5094075 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2CCN(C(=O)OCc3ccccc3)CC2=O)C2(CCCC2)C1 CHEMBL5092580 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-n3cc4ccccc4n3)ncc2=O)C(C)(C)C1 CHEMBL5086052 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2ccc3nc(N=S(C)(C)=O)ncc3c2=O)C2(CCCC2)C1 CHEMBL5080385 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2CCNCC2=O)C2(CCCC2)C1 CHEMBL5093660 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(N=S(C)(C)=O)c(Cl)cc2=O)C2(CCCC2)C1 CHEMBL5077632 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-n3ncc4ccccc43)ncc2=O)C(C)(C)C1 CHEMBL5078444 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2ccc3nc(N4CCN(C)CC4)ncc3c2=O)C2(CCCC2)C1 CHEMBL5079674 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2CC(Cc3ccccc3)CC2=O)C(C)(C)C1 CHEMBL5093270 IC50 500.0 nM
CC1(C)CCC(N2CCN(CC3(O)CCN(C(=O)NCc4ccccc4)CC34CCCC4)C(=O)C2)CC1 CHEMBL5085532 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(S(C)(=N)=O)c(-c3ccccc3)cc2=O)C(C)(C)C1 CHEMBL5083863 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(C3CC3)ncc2=O)C(C)(C)C1 CHEMBL5085165 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3ccncc3)ncc2=O)C(C)(C)C1 CHEMBL5078801 IC50 500.0 nM
O=C(N1CCC(O)(Cn2ccncc2=O)C2(CCCC2)C1)N1CCNC[C@H]1c1ccccc1 CHEMBL5085085 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2ccc3nc(N4CCOCC4)ncc3c2=O)C2(CCCC2)C1 CHEMBL5078760 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2C(=O)COc3c(N)cccc32)C2(CCCC2)C1 CHEMBL5082927 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2CCN(C)CC2=O)C2(CCCC2)C1 CHEMBL5089474 IC50 500.0 nM
COc1cc2ncn(CC3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)c(=O)c2cc1OC CHEMBL5074823 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc3sccc3c2=O)C2(CCCC2)C1 CHEMBL5086890 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc3c(F)cccc3c2=O)C2(CCCC2)C1 CHEMBL5091763 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2ccc3ccc(F)cc3c2=O)C2(CCCC2)C1 CHEMBL5081636 IC50 500.0 nM
O=C(N1CCC(O)(Cn2ccncc2=O)C2(CCCC2)C1)N1CCOC[C@H]1c1ccccc1 CHEMBL5090166 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(S(C)(=N)=O)c(Cl)cc2=O)C(C)(C)C1 CHEMBL5092855 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(N3CCCC3=O)ncc2=O)C(C)(C)C1 CHEMBL5083955 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc3ccccc3c2=O)C2(CCCC2)C1 CHEMBL5081352 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2Cc3ccccc3C2=O)C2(CCCC2)C1 CHEMBL5092718 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(Cn2cc(N=S(C)(C)=O)c(-c3ccccc3F)cc2=O)C(C)(C)C1 CHEMBL5092265 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2ccc3nc(N(C)C)ncc3c2=O)C2(CCCC2)C1 CHEMBL5083507 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(CN2C(=O)COc3cccnc32)C2(CCCC2)C1 CHEMBL5076801 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3ccncc3)ncc2=O)C2(CCCC2)C1 CHEMBL5093450 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(-c3cccnc3)ncc2=O)C(C)(C)C1 CHEMBL5084603 IC50 500.0 nM
COc1ccc2c(=O)n(CC3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)ccc2c1 CHEMBL5089033 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc3ccsc3c2=O)C2(CCCC2)C1 CHEMBL5076400 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cc(C(=O)N(C)C)c3ccccc3c2=O)C2(CCCC2)C1 CHEMBL5079040 IC50 500.0 nM
COc1cc2ccn(CC3(O)CCN(C(=O)[C@H](C)CC4CCCCC4)CC34CCCC4)c(=O)c2cc1OC CHEMBL5091440 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2cnc3ccc(Cl)cc3c2=O)C2(CCCC2)C1 CHEMBL5070567 IC50 500.0 nM
Cc1nc2cnccc2c(=O)n1CC1(O)CCN(C(=O)[C@H](C)CC2CCCCC2)CC12CCCC2 CHEMBL5077217 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2cnc3ccncc3c2=O)C2(CCCC2)C1 CHEMBL5078273 IC50 500.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CCC(O)(Cn2ccc3ncncc3c2=O)C2(CCCC2)C1 CHEMBL5082008 IC50 500.0 nM
CSc1ncc2c(=O)n(CC3(O)CCN(C(=O)[C@H](C)CC(F)(F)F)CC34CCCC4)cnc2n1 CHEMBL5086241 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2cnc3nc(N4CCOCC4)ncc3c2=O)C2(CCCC2)C1 CHEMBL5087735 IC50 500.0 nM
C[C@H](CC(F)(F)F)C(=O)N1CCC(O)(Cn2cnc3nc(N4CCN(C)CC4)ncc3c2=O)C2(CCCC2)C1 CHEMBL5084992 IC50 500.0 nM
O=C(N1CCC(O)(Cn2ccc3ccncc3c2=O)C2(CCCC2)C1)N1CCOC[C@H]1c1ccccc1 CHEMBL5075539 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc3c(cnn3Cc3ccccc3)c2=O)C2(CCCC2)C1)N1CCOC[C@H]1c1ccccc1 CHEMBL5082722 IC50 500.0 nM
O=C(NCc1ccccc1)N1CCC(O)(Cn2cnc(-c3ccncc3)cc2=O)C2(CCCC2)C1 CHEMBL5080362 IC50 500.0 nM
Cn1nccc1-c1cc(=O)n(CC2(O)CCN(C(=O)NCc3ccccc3)CC23CCCC3)cn1 CHEMBL5089311 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)N1CCCC1C(F)(F)F CHEMBL5088054 IC50 500.0 nM
O=C(N1CC(C(F)(F)F)C1)N1CC[C@@](O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5087232 IC50 500.0 nM
O=C(N1CCC(C(F)(F)F)C1)N1CC[C@@](O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5094146 IC50 500.0 nM
CN(Cc1ccoc1)C(=O)N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5094708 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)N1CCCC1c1cccnc1 CHEMBL5090588 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)N1CCCC1c1ccncc1 CHEMBL5093790 IC50 500.0 nM
CN(Cc1cccc(C#N)c1)C(=O)N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5081864 IC50 500.0 nM
CC(NC(=O)N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)c1ccoc1 CHEMBL5088028 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)N1CCCC1C1CC1 CHEMBL5093863 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)N1CCC[C@H]1c1ccon1 CHEMBL5090180 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)N1CCNCC1c1cccnc1 CHEMBL5078479 IC50 500.0 nM
CC(=O)N1CCN(C(=O)N2CC[C@@](O)(Cn3cnc(-c4ccccc4)cc3=O)C3(CCCC3)C2)[C@H](c2ccccc2)C1 CHEMBL5084923 IC50 500.0 nM
O=C(N1CCC(O)(Cn2cnc(-c3ccccc3)cc2=O)CC1)N1CCOC[C@H]1c1ccccc1 CHEMBL5091345 IC50 500.0 nM
O=C(N1CC[C@@](O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1)N1CCCN1c1ccccc1 CHEMBL5072989 IC50 500.0 nM
O=C(NC(C(F)(F)F)C(F)(F)F)N1CC[C@@](O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5075818 IC50 500.0 nM
O=C(NCC1(F)CC1)N1CC[C@@](O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5085008 IC50 500.0 nM
CN(CC1CC1)C(=O)N1CC[C@@](O)(Cn2cnc(-c3ccccc3)cc2=O)C2(CCCC2)C1 CHEMBL5094417 IC50 500.0 nM
O=C(N1CCC(O)(Cn2ccc(-c3ccccc3)c(F)c2=O)C2(CCCC2)C1)N1CCNC[C@H]1c1ccccc1 CHEMBL5070417 IC50 500.0 nM
COc1cccc2c1CN(C[C@]1(O)CCN(C(=O)[C@H](C)CC3CCCCC3)CC13CCCC3)C2=O CHEMBL5436433 IC50 500.0 nM
Cc1cccc2c1CN(C[C@]1(O)CCN(C(=O)[C@H](C)CC3CCCCC3)CC13CCCC3)C2=O CHEMBL5406382 IC50 530.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2C[C@@H](c3ccccc3)CC2=O)C(C)(C)C1 CHEMBL5403692 IC50 740.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2C[C@](C)(c3ccccc3)CC2=O)C2(CCCC2)C1 CHEMBL5408004 IC50 760.0 nM
Cc1ccccc1[C@H]1CC(=O)N(C[C@]2(O)CCN(C(=O)[C@H](C)CC3CCCCC3)CC23CCCC3)C1 CHEMBL5421949 IC50 800.0 nM
C[C@H](CC1CCCCC1)C(=O)N1CC[C@@](O)(CN2Cc3c(cccc3-c3cscn3)C2=O)C2(CCCC2)C1 CHEMBL5438285 IC50 940.0 nM