CC(C)C[C@@H](NC(=O)C1(C(F)(F)F)CCCCC1)C(=O)Nc1nnc(Cc2ccc(C#N)cc2)s1 CHEMBL5279102 EC50 0.0166 nM
N#Cc1ccc(Cc2nnc(NC(=O)[C@@H](CO)NC(=O)C3(C(F)(F)F)CCCCC3)s2)cc1 CHEMBL5286335 Kd 5.8 nM
CC(NC(=O)C1CCCC1)C(=O)Nc1nnc(Cc2ccc([N+](=O)[O-])cc2)s1 CHEMBL5273043 Kd 7.87 nM
N#Cc1ccc(Cc2nnc(NC(=O)[C@H](NC(=O)C3(C(F)(F)F)CCCCC3)C3CCCC3)s2)cc1 CHEMBL5268828 IC50 8.0 nM
CCC1(C(=O)N[C@H](COC)C(=O)Nc2nnc(Cc3ccc(C#N)cc3)s2)CCCCC1 CHEMBL5277351 IC50 28.0 nM
COC[C@@H](NC(=O)C1(C)CCCCC1)C(=O)Nc1nnc(Cc2ccc(C#N)cc2)s1 CHEMBL5275560 IC50 32.0 nM
COC[C@@H](NC(=O)C1(C(F)F)CCCCC1)C(=O)Nc1nnc(Cc2ccc(C#N)cc2)s1 CHEMBL5267932 IC50 32.0 nM
COC[C@@H](NC(=O)C1(C(F)(F)F)CCCCC1)C(=O)Nc1nnc(Cc2ccc(C#N)cc2)s1 CHEMBL5271965 IC50 36.0 nM
CC(C)(O)[C@@H](NC(=O)C1(C(F)(F)F)CCCCC1)C(=O)Nc1nnc(Cc2ccc(C#N)cc2)s1 CHEMBL5266176 IC50 45.0 nM
COC[C@@H](NC(=O)C1(C)CCCCC1)C(=O)Nc1sc(Cc2ccc(C#N)cc2)nc1C CHEMBL5279700 IC50 65.0 nM
COC[C@@H](NC(=O)C1(C)CCCCC1)C(=O)Nc1nc(C)c(Cc2ccc(C#N)cc2)s1 CHEMBL5280287 IC50 72.0 nM
COCC(NC(=O)C1(C)CCCCC1)C(=O)Nc1nnc(Cc2ccc([N+](=O)[O-])cc2)s1 CHEMBL5274527 IC50 72.0 nM
COC[C@@H](NC(=O)C1(C)CCCCC1)C(=O)Nc1nnc(Cc2ccc([N+](=O)[O-])cc2)s1 CHEMBL5275910 IC50 74.0 nM
COCC(NC(=O)C1CCCCC1)C(=O)Nc1nnc(Cc2ccc([N+](=O)[O-])cc2)s1 CHEMBL5278034 IC50 221.0 nM