O=C(Nc1snnc1C(=O)Nc1ccc(N2CCCC2)cc1)c1cncc(C(F)(F)F)c1 CHEMBL5303447 IC50 198.0 nM
CC(C)(C)[C@H]1CC[C@@H](NC(=O)c2nnsc2NC(=O)c2cncc(C(F)(F)F)c2)CC1 CHEMBL5402536 IC50 329.0 nM
O=C(Nc1snnc1C(=O)Nc1ccc(Oc2ccccc2)cc1)c1cncc(C(F)(F)F)c1 CHEMBL5425763 IC50 335.0 nM
O=C(Nc1snnc1C(=O)Nc1ccc(C(F)(F)F)cc1)c1cncc(C(F)(F)F)c1 CHEMBL5440446 IC50 340.0 nM
O=C(Nc1snnc1C(=O)Nc1cccc(Oc2ccccc2)c1)c1cncc(C(F)(F)F)c1 CHEMBL5395399 IC50 365.0 nM
O=C(Nc1snnc1C(=O)Nc1cccc(N2CCCC2)c1)c1cncc(C(F)(F)F)c1 CHEMBL5426200 IC50 407.0 nM
O=C(Nc1snnc1C(=O)Nc1ccc2c(c1)CCC2)c1cncc(C(F)(F)F)c1 CHEMBL5405199 IC50 507.0 nM
CC(C)c1ccc(NC(=O)c2nnsc2NC(=O)c2cncc(C(F)(F)F)c2)cc1 CHEMBL5430481 IC50 553.0 nM
O=C(Nc1snnc1C(=O)Nc1ccc(OC(F)(F)F)cc1)c1cncc(C(F)(F)F)c1 CHEMBL5398825 IC50 556.0 nM
O=C(Nc1nc(-c2ccccc2)ns1)c1ccccc1NS(=O)(=O)c1ccc(-c2ccccc2)cc1 CHEMBL5416528 IC50 560.0 nM
O=C(Nc1snnc1C(=O)Nc1cccc(Cl)c1)c1cncc(C(F)(F)F)c1 CHEMBL5419354 IC50 587.0 nM
O=C(Nc1snnc1C(=O)Nc1ccc2c(c1)OC(F)(F)O2)c1cncc(C(F)(F)F)c1 CHEMBL5398708 IC50 666.0 nM
CC(C)c1cccc(NC(=O)c2nnsc2NC(=O)c2cncc(C(F)(F)F)c2)c1 CHEMBL5424112 IC50 669.0 nM
O=C(Nc1snnc1C(=O)Nc1ccc(Cl)cc1)c1cncc(C(F)(F)F)c1 CHEMBL5431635 IC50 689.0 nM
O=C(Nc1snnc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cncc(C(F)(F)F)c1 CHEMBL5408990 IC50 749.0 nM
O=C(Nc1snnc1C(=O)N[C@@H](CN1CCCC1)c1ccc(Cl)cc1)c1cncc(C(F)(F)F)c1 CHEMBL5435107 IC50 764.0 nM
O=C(Nc1nc(-c2ccccc2)ns1)c1ccc(C(F)(F)F)cc1NS(=O)(=O)c1ccc(Cl)cc1 CHEMBL5400602 IC50 816.0 nM
CC(C)(NC(=O)c1nnsc1NC(=O)c1cccc(Cl)c1)c1cccc(Cl)c1 CHEMBL5399861 IC50 820.0 nM
O=C(Nc1snnc1C(=O)Nc1ccn(-c2cccc(Cl)c2)n1)c1cccc(Cl)c1 CHEMBL5431379 IC50 826.0 nM
CC(C)Oc1cccc(NC(=O)c2nnsc2NC(=O)c2cccc(Cl)c2)c1 CHEMBL5403255 IC50 849.0 nM
O=C(Nc1snnc1C(=O)NCC1CC12CCCCC2)c1cncc(C(F)(F)F)c1 CHEMBL5398678 IC50 868.0 nM
CC(C)(NC(=O)c1nnsc1NC(=O)c1cncc(Cl)c1)c1ccccc1 CHEMBL5436187 IC50 898.0 nM
O=C(Nc1snnc1C(=O)Nc1cccc(OC(F)F)c1)c1cncc(C(F)(F)F)c1 CHEMBL5416230 IC50 900.0 nM
O=C(Nc1snnc1C(=O)NCc1ccc(Cl)cc1)c1cccc(C(F)(F)F)c1 CHEMBL5432156 IC50 923.0 nM
O=C(Nc1snnc1C(=O)NC1Cc2ccc(Cl)cc2C1)c1cccc(C(F)(F)F)c1Cl CHEMBL5414618 IC50 961.0 nM
CC(C)n1ncc2cc(NC(=O)c3nnsc3NC(=O)c3cncc(C(F)(F)F)c3)ccc21 CHEMBL5408951 IC50 961.0 nM
Cc1ccc(C)c(NC(=O)c2nnsc2NC(=O)c2cccc(Cl)c2)c1 CHEMBL5423451 IC50 964.0 nM
CC(NC(=O)c1nnsc1NC(=O)c1cccc(Cl)c1)c1ccc(Cl)cc1 CHEMBL5436483 IC50 989.0 nM
