CN1CC[C@@H](Oc2ccc(F)c(-c3nc4c(o3)C(=O)c3ccccc3C4=O)c2Cl)C1 CHEMBL5185273 IC50 0.28 nM
CN1CC[C@@H](Oc2ccc(Cl)c(-c3nc4c(o3)C(=O)c3ccccc3C4=O)c2)C1 CHEMBL5196686 IC50 1.27 nM
CN1CC[C@@H](Oc2ccc(Cl)c(-c3nc4c(o3)C(=O)c3ccccc3C4=O)c2F)C1 CHEMBL5173239 IC50 2.0 nM
O=C1c2ccccc2C(=O)c2oc(-c3cccnc3)nc21 CHEMBL5172138 IC50 2.7 nM
N#Cc1nc2c(nc1C#N)-c1ccc(Cl)cc1C2=O CHEMBL2398212 IC50 96.0 nM
N#Cc1nc2c(nc1C#N)-c1cc(Cl)ccc1C2=O CHEMBL3407548 IC50 133.0 nM
N#Cc1nc2c(nc1C#N)-c1ccc(F)cc1C2=O CHEMBL5281075 IC50 250.0 nM
CCO/N=C1/c2ccccc2-c2nc(C#N)c(C#N)nc21 CHEMBL5180195 IC50 280.0 nM
N#Cc1cc2c(cc1C#N)-c1ccccc1C2=O CHEMBL5170305 IC50 290.0 nM
N#Cc1nc2c(nc1C#N)-c1ccccc1C2=O CHEMBL4569978 IC50 290.0 nM
Cc1c(F)ccc2c1C(=O)c1nc(C#N)c(C#N)nc1-2 CHEMBL5269711 IC50 316.0 nM
C=CCO/N=C1\c2ccccc2-c2nc(C#N)c(C#N)nc21 CHEMBL5202404 IC50 560.0 nM
COc1ccc2c(c1OC)C(=O)c1nc(C#N)c(C#N)nc1-2 CHEMBL5276040 IC50 710.0 nM
COc1ccc(OC)c2c1C(=O)c1nc(C#N)c(C#N)nc1-2 CHEMBL4515695 IC50 810.0 nM
N#Cc1nc2c(nc1C#N)-c1ccccc1/C2=N\OCc1ccccc1 CHEMBL5208383 IC50 850.0 nM
Cc1ccc2c(c1)-c1nc(C#N)c(C#N)nc1C2=O CHEMBL4584162 IC50 930.0 nM
Cc1ccc(S(=O)(=O)Nc2cc(C(F)(F)F)ccc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 CHEMBL3392741 IC50 950.0 nM