CCc1ccccc1-n1nc(C)c(C(=O)Nc2ccc3ccccc3n2)c1C CHEMBL5174802 IC50 1.3 nM
Cc1ccccc1-n1nc(C)c(C(=O)Nc2ccc3ccccc3n2)c1C CHEMBL5200990 IC50 1.5 nM
Cc1c(C(=O)Nc2ccc3ccccc3n2)cnn1-c1ccccc1Br CHEMBL4555217 IC50 2.3 nM
COc1ccc(C(=O)C2CCN(CC(=O)N(Cc3nc4c(c(=O)[nH]3)COCC4)CC3CC3)CC2)cc1 CHEMBL2419706 IC50 3.5 nM
O=C(c1ccc(F)cc1)C1CCN(CC(=O)N(Cc2nc3c(c(=O)[nH]2)COCC3)Cc2cccs2)CC1 CHEMBL2419698 IC50 3.6 nM
Cc1ccccc1-n1nnc(C(=O)Nc2ccc3ccccc3n2)c1C CHEMBL4454905 IC50 4.1 nM
Cn1cc(-c2ccc(-c3cncc(Cl)c3N3CCC4(CCNC4=O)CC3)cc2)cn1 CHEMBL3408213 IC50 7.0 nM
O=C(c1ccc(F)cc1)C1CCN(CC(=O)N(Cc2nc3c(c(=O)[nH]2)COCC3)CC2CC2)CC1 CHEMBL2419705 IC50 17.0 nM
CC(C)CN(Cc1nc2c(c(=O)[nH]1)COCC2)C(=O)CN1CCC(C(=O)c2ccc(F)cc2)CC1 CHEMBL2419701 IC50 17.0 nM
Cc1nn(-c2ccccc2Br)c(C)c1C(=O)Nc1ccc2ccccc2n1 CHEMBL5199170 IC50 21.0 nM
CCCN(Cc1nc2c(c(=O)[nH]1)COCC2)C(=O)CN1CCC(C(=O)c2ccc(F)cc2)CC1 CHEMBL2419702 IC50 34.0 nM
O=C(CN1CCC(C(=O)c2ccc(F)cc2)CC1)NCc1nc2c(c(=O)[nH]1)COCC2 CHEMBL2419697 IC50 40.0 nM
Cc1nn(-c2ccccc2C(C)C)c(C)c1C(=O)Nc1ccc2ccccc2n1 CHEMBL5197208 IC50 48.0 nM
Cc1nn(-c2c(F)cccc2Br)c(C)c1C(=O)Nc1ccc2ccccc2n1 CHEMBL5205399 IC50 50.0 nM
O=C(c1ccc(F)cc1)C1CCN(CC(=O)N(Cc2ccccn2)Cc2nc3c(c(=O)[nH]2)COCC3)CC1 CHEMBL2419700 IC50 52.0 nM
O=C(c1ccc(F)cc1)C1CCN(CC(=O)N(Cc2ccccc2)Cc2nc3c(c(=O)[nH]2)COCC3)CC1 CHEMBL2419699 IC50 65.0 nM
CCN(Cc1nc2c(c(=O)[nH]1)COCC2)C(=O)CN1CCC(C(=O)c2ccc(F)cc2)CC1 CHEMBL2419703 IC50 70.0 nM
Oc1nc(-c2ccc(C(F)(F)F)cc2)nc2c1CSCC2 CHEMBL1086580 IC50 78.0 nM
Cc1nn(-c2ccccc2F)c(C)c1C(=O)Nc1ccc2ccccc2n1 CHEMBL5188822 IC50 87.0 nM
Cc1ccc(C)c(-n2nc(C)c(C(=O)Nc3ccc4ccccc4n3)c2C)c1 CHEMBL5201010 IC50 96.0 nM
Cc1nn(-c2ccccc2)c(C)c1C(=O)Nc1ccc2ccccc2n1 CHEMBL5201325 IC50 135.0 nM
CN(Cc1nc2c(c(=O)[nH]1)COCC2)C(=O)CN1CCC(C(=O)c2ccc(F)cc2)CC1 CHEMBL2419704 IC50 193.0 nM
O=C(CCc1ccccc1F)N(Cc1nc2c(c(=O)[nH]1)COCC2)Cc1cccs1 CHEMBL2419718 IC50 304.0 nM
Cc1nn(-c2ccccc2Cl)c(C)c1C(=O)Nc1ccc2ccccc2n1 CHEMBL5195176 IC50 305.0 nM
O=C(CCc1ccc(F)cc1)N(Cc1nc2c(c(=O)[nH]1)COCC2)Cc1cccs1 CHEMBL2419692 IC50 483.0 nM
O=C(CCc1cccc(O)c1)N(Cc1nc2c(c(=O)[nH]1)COCC2)Cc1cccs1 CHEMBL2419694 IC50 812.0 nM
O=C(CCc1ccccc1)N(Cc1nc2ccccc2c(=O)[nH]1)Cc1cccs1 CHEMBL2419711 IC50 937.0 nM