CCNC(=O)c1ccc2c(C3CCN(CC4(O)C5CC6CC(C5)CC4C6)CC3)c(C)nn2c1 CHEMBL5397585 Ki 21.0 nM
CCNC(=O)c1ccc2c([C@H]3CCN(CC4(O)CCOCC4)C[C@@H]3C)c(C)nn2c1 CHEMBL5439842 Kd 30.0 nM
CCNC(=O)c1ccc2c(c1)nc(-c1cccn(C)c1=O)n2[C@H]1CCN(CC2(O)CCCCC2)C[C@@H]1C CHEMBL5414722 Ki 33.0 nM
CCNC(=O)c1ccc2c([C@H]3CCN(CC4(O)CCCCC4)C[C@@H]3C)c(C)nn2c1 CHEMBL5428051 Ki 33.0 nM
Cc1nn2cc(C(=O)NCC3CC3)ccc2c1[C@H]1CCN(CC2(O)CCOCC2)C[C@@H]1C CHEMBL5432565 Ki 43.0 nM
CCNC(=O)c1ccc2c(c1)nc(C(F)F)n2[C@H]1CCN(CC2(O)CCCCC2)C[C@@H]1C CHEMBL5434894 Kd 45.0 nM
CCNC(=O)c1ccc2c(C3CCN(CC4(O)CCCCC4)CC3)c(C)nn2c1 CHEMBL5439506 Ki 56.0 nM
COC1(CN2CC[C@H](c3c(C)nn4cc(C(=O)NCC5CC5)ccc34)[C@@H](C)C2)CCOCC1 CHEMBL5426169 Ki 57.0 nM
CCNC(=O)c1ccc2c(c1)nc(C)n2[C@H]1CCN(CC2(O)CCCCC2)C[C@@H]1C CHEMBL5411016 Ki 63.0 nM
CCNC(=O)c1ccc2c(C3CCN(CC4(O)CCCCC4)CC3)c(-c3cccn(C)c3=O)nn2c1 CHEMBL5432083 Ki 69.0 nM
O=C(Nc1ccc(C(=O)N2CC(c3nc4ccccc4s3)C2)s1)[C@@H]1C[C@@H](OCCCCCO[C@H]2CN[C@H](C(=O)Nc3ccc(C(=O)N4CC(c5nc6ccccc6s5)C4)s3)C2)CN1 CHEMBL5409682 IC50 96.0 nM
CCNC(=O)c1ccc2c(c1)nc(C)n2C1CCN(CC2(O)CCCCC2)CC1 CHEMBL5429949 Ki 141.0 nM
CCNC(=O)c1ccc2c(c1)[nH]c(=O)n2C1CCN(CC2(O)CCCCC2)CC1 CHEMBL5435884 Ki 284.0 nM
CCNC(=O)c1ccc2c(c1)[nH]c(=O)n2C1CCN(C[C@@H](O)c2ccc(Cl)cc2)CC1 CHEMBL5439514 Ki 540.0 nM